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- [31] Synthesis and [4+2] cycloaddition of (2R,2′R)-N,N′-fumaroylbis[fenchane-8,2-sultam] (= (2E)-1,4-bis[(3aS,6S,7aR)-1,4,5,6,7,7a-hexahydro-7,7-dimethyl-2,2-dioxido-3H-3a,6-methano-2,1-benzothiazol-1-yl]but-2-ene-1,4-dione) to cyclopentadieneHELVETICA CHIMICA ACTA, 2005, 88 (09) : 2441 - 2453Piatek, AM论文数: 0 引用数: 0 h-index: 0机构: Warsaw Univ, Dept Chem, PL-02093 Warsaw, PolandChojnacka, A论文数: 0 引用数: 0 h-index: 0机构: Warsaw Univ, Dept Chem, PL-02093 Warsaw, PolandChapuis, C论文数: 0 引用数: 0 h-index: 0机构: Warsaw Univ, Dept Chem, PL-02093 Warsaw, PolandJurczak, J论文数: 0 引用数: 0 h-index: 0机构: Warsaw Univ, Dept Chem, PL-02093 Warsaw, Poland
- [32] Safety and efficacy of AveMix (R) XG 10 (endo-1,4-beta-xylanase and endo1,3(4)-beta-glucanase) for use as feed additive for chickens for fattening1 2 Scientific Opinion of the Panel on Additives and Products or Substances used in Animal FeedEFSA JOURNAL, 2009, 7 (06):Bories, Georges论文数: 0 引用数: 0 h-index: 0Brantom, Paul论文数: 0 引用数: 0 h-index: 0de Barbera, Joaquim Brufau论文数: 0 引用数: 0 h-index: 0Chesson, Andrew论文数: 0 引用数: 0 h-index: 0Cocconcelli, Pier Sandro论文数: 0 引用数: 0 h-index: 0Debski, Bogdan论文数: 0 引用数: 0 h-index: 0Dierick, Noel论文数: 0 引用数: 0 h-index: 0Gropp, Juergen论文数: 0 引用数: 0 h-index: 0Halle, Ingrid论文数: 0 引用数: 0 h-index: 0Hogstrand, Christer论文数: 0 引用数: 0 h-index: 0de Knecht, Joop论文数: 0 引用数: 0 h-index: 0Leng, Lubomir论文数: 0 引用数: 0 h-index: 0Lindgren, Sven论文数: 0 引用数: 0 h-index: 0Haldorsen, Anne-Katrine Lundebye论文数: 0 引用数: 0 h-index: 0Mantovani, Alberto论文数: 0 引用数: 0 h-index: 0Mezes, Miklos论文数: 0 引用数: 0 h-index: 0Nebbia, Carlo论文数: 0 引用数: 0 h-index: 0Rambeck, Walter论文数: 0 引用数: 0 h-index: 0Rychen, Guido论文数: 0 引用数: 0 h-index: 0von Wright, Atte论文数: 0 引用数: 0 h-index: 0Wester, Pieter论文数: 0 引用数: 0 h-index: 0
- [33] Overcoming Preclinical Safety Obstacles to Discover (S)-N-((1,2,3,5,6,7-Hexahydro-s-indacen-4-yl)carbamoyl)-6-(methylamino)-6,7-dihydro-5H-pyrazolo[5,1-b][1,3]oxazine-3-sulfonamide (GDC-2394): A Potent and Selective NLRP3 InhibitorJOURNAL OF MEDICINAL CHEMISTRY, 2022, 65 (21) : 14721 - 14739Townsend, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAStivala, Craig E.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAMcBride, Christopher论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA 858 Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USATrzoss, Lynnie论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USAPovero, Davide论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USALazic, Milos论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA 858 Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USAAmbrus-Aikelin, Geza论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USASantini, Angelina论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA 858 Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USAPranadinata, Rama论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USABain, Gretchen论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA 858 Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USAStansfield, Ryan论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA 858 Therapeut, San Diego, CA 92121 USA Denali Therapeut, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAStafford, Jeffrey A.论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA 858 Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USAVeal, James论文数: 0 引用数: 0 h-index: 0机构: Jecure Therapeut, San Diego, CA 92121 USA 858 Therapeut, San Diego, CA 92121 USA Genentech Inc, South San Francisco, CA 94080 USATakahashi, Ryan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USALy, Justin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAChen, Shu论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USALiu, Liling论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USANespi, Marika论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USABlake, Robert论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAKatewa, Arna论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAKleinheinz, Tracy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USASujatha-Bhaskar, Swathi论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USARamamoorthi, Nandhini论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USASims, Jessica论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAMcKenzie, Brent论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Sonoma Biotherapeut, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAChen, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAUltsch, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAJohnson, Matthew论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAMurray, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USACiferri, Claudio论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USAStaben, Steven T. .论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, South San Francisco, CA 94080 USA Lycia Therapeut, South San Francisco, CA 94080 USA Genentech Inc, South San Francisco, CA 94080 USA
- [34] Discovery of 6-(2,4-Dichlorophenyl)-5-[4-[(3S)-1-(3-fluoropropyl)pyrrolidin-3-yl]oxyphenyl]-8,9-dihydro-7H-benzo[7]annulene-2-carboxylic acid (SAR439859), a Potent and Selective Estrogen Receptor Degrader (SERD) for the Treatment of Estrogen-Receptor-Positive Breast CancerJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (02) : 512 - 528El-Ahmad, Youssef论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceTabart, Michel论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceHalley, Frank论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceCertal, Victor论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceThompson, Fabienne论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceFiloche-Romme, Bruno论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceGruss-Leleu, Florence论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceMuller, Claire论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceBrollo, Maurice论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceFabien, Laurence论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceLoyau, Veronique论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceBertin, Luc论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceRichepin, Patrick论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FrancePilorge, Fabienne论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceDesmazeau, Pascal论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceGirardet, Chrystelle论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceBeccari, Sylvie论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, 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FranceVallee, Francois论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceSteier, Valerie论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceMathieu, Magali论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceRak, Alexey论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, France Sanofi, Integrated Drug Discovery, 13 Quai Jules Guesde, F-94403 Vitry Sur Seine, FranceAbecassis, Pierre-Yves论文数: 0 引用数: 0 h-index: 0机构: Sanofi, Drug Metab & Pharmacokinet DMPK, 13 Quai Jules Guesde, 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