Synthesis and biological activity of cyanopyridine, isoxazole and pyrazoline derivatives having thymol moiety

被引：0
|
作者：
Desai, JM [1 ]
Shah, VH [1 ]
机构：
[1] Saurashtra Univ, Dept Chem, Rajkot 360005, Gujarat, India
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 2003年 / 42卷 / 02期
关键词：
D O I：
暂无
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
New 4-acetoacetamido thymol 1, 4-(substituted benzalacetoacetamido)-thymols 2a-j, 4-(2'-amino-3'-cyano-4'-arylpyridin-6'-yl-acetamido) thymols 3a-j, 4-(5'-arylisoxazol-3'-yl-acetamido) thymols 4a-j and 4-(1'-N(H)/acetyl-5'-arylpyrazolin-3'-yl-acetamido) thymols 5a-t have been synthesised and screened for their antimicrobial activity. The products display moderate to good activities. The structures of the products 1, 2a-j, 3a-j, 4a-j and 5a-t have been elucidated by elemental analyses and spectral data.
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页码：382 / 385
页数：4
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