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- [31] Discovery of DS42450411 as a potent orally active hepcidin production inhibitor: Design and optimization of novel 4-aminopyrimidine derivativesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2018, 28 (20) : 3333 - 3337Fukuda, Takeshi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanIshiyama, Takashi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanKatagiri, Takahiro论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanUeda, Kenjiro论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Pain & Neurosci Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanMuramatsu, Sumie论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Pain & Neurosci Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanHashimoto, Masami论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Med Informat Dept, Chuo Ku, 3-5-1 Nihombashihoncyo, Tokyo 1038426, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanAki, Anri论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Biol & Immunooncol Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanBaba, Daichi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Postmkt Regulatory Affairs Dept, Chuo Ku, 3-5-1 Nihombashihoncyo, Tokyo 1038426, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanWatanabe, Kengo论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Drug Metab & Pharmacokinet Res Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, JapanTanaka, Naoki论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, Oncol Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, Rare Dis Labs, Shinagawa Ku, 1-2-58 Hiromachi, Tokyo 1408710, Japan
- [32] Discovery of potent, orally active benzimidazole glucagon receptor antagonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (13) : 3701 - 3705Kim, Ronald M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChang, Jiang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USALins, Ashley R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USABrady, Ed论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USACandelore, Mari R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADallas-Yang, Qing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADing, Victor论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USADragovic, Jasminka论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAIliff, Susan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAJiang, Guoqiang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAMock, Steven论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAQureshi, Sajjad论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASaperstein, Richard论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Pharmacol, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USASzalkowski, Deborah论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATamvakopoulos, Constantin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATota, Laurie论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAWright, Michael论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAYang, Xiaodong论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USATata, James R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAChapman, Kevin论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAZhang, Bei B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Metab Disorders, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USAParmee, Emma R.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA Merck Res Labs, Dept Med Chem, Rahway, NJ 07065 USA
- [33] Discovery of potent and orally active farnesyltransferase (FT) inhibitors.ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2002, 224 : U29 - U29Tong, YS论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAWang, L论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAHasvold, L论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALeonard, N论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALi, TM论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALi, Q论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAWang, WB论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USACohen, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAGu, WZ论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAZhang, HY论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USABauch, J论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USAMarsh, K论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USARosenberg, SH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USALin, NH论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USASham, HL论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA Abbott Labs, Global Pharmaceut R&D, Canc Res, Abbott Pk, IL 60064 USA
- [34] Discovery of novel tetracyclic tetrahydrofuran derivatives as potent, orally active, broad spectrum psychotropic agentsProceedings of the Joint Meeting on Medicinal Chemistry, 2005, : 63 - 66Alonso, JM论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainAndrés, JI论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainCid, JM论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainDíaz, A论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainFernández, J论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainIturrino, L论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainGil, P论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainMegens, A论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainSipido, VK论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, SpainTrabanco, AA论文数: 0 引用数: 0 h-index: 0机构: Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain Johnson & Johnson Pharmaceut Res & Dev, Drug Discovery CNS, Toledo 45007, Spain
- [35] Discovery of novel quinoline sulphonamide derivatives as potent, selective and orally active RORγ inverse agonistsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (14) : 1799 - 1806Amaudrut, Jerome论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceArgiriadi, Maria A.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBarth, Martine论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBreinlinger, Eric C.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBressac, Didier论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceBroqua, Pierre论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceCalderwood, David J.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceChatar, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceCusack, Kevin P.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 381 Plantat St, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceGauld, Stephen B.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 1 North Waukegan Rd, N Chicago, IL 60064 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceJacquet, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceKamath, Rajesh, V论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceKort, Michael E.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 1 North Waukegan Rd, N Chicago, IL 60064 USA Inventiva, 50 Rue Dijon, F-21121 Daix, FranceLepais, Valerie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceLuccarini, Jean-Michel论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMasson, Philippe论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMontalbetti, Christian论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceMounier, Laurent论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FrancePotin, Dominique论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FrancePoupardin, Olivia论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceRouaud, Sylvie论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceSpitzer, Luc论文数: 0 引用数: 0 h-index: 0机构: Inventiva, 50 Rue Dijon, F-21121 Daix, France Inventiva, 50 Rue Dijon, F-21121 Daix, FranceWallace, Craig D.论文数: 0 引用数: 0 h-index: 0机构: AbbVie, 100 Res Dr, Worcester, MA 01605 USA Inventiva, 50 Rue Dijon, F-21121 Daix, France
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