A ONE-POT SYNTHESIS OF PHAITANTHRIN E THROUGH INTERMOLECULAR CONDENSATION/INTRAMOLECULAR ARYL C-H AMINATION CASCADE

被引：13

作者：

Itoh, Tomoki ^{[1
]}

Abe, Takumi ^{[1
]}

Choshi, Tominari ^{[2
]}

Nishiyama, Takashi ^{[2
]}

Ishikura, Minoru ^{[1
]}

机构：

[1] Hlth Sci Univ Hokkaido, Sch Pharmaceut Sci, Ishikari, Hokkaido 0610293, Japan

[2] Fukuyama Univ, Fac Pharm & Pharmaceut Sci, Fukuyama, Hiroshima 7290292, Japan

来源：

HETEROCYCLES | 2016年 / 92卷 / 06期

关键词：

Indoloquinazoline; Phaitanthrin E; Condensation/Aryl CH Amination Cascade; One-Pot Synthesis; TRYPTANTHRIN; DERIVATIVES; CHEMISTRY;

D O I：

10.3987/COM-16-13465

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

A one-pot synthesis of phaitanthrin E starting from methyl indole-3-carboxylate and isatoic anhydride through intermolecular condensation/intramolecular aryl C-H amination cascade was developed.

引用

页码：1132 / 1136

页数：5

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