共 50 条
- [41] Synthesis of 2′-O,4′-C-alkylene-bridged ribonucleosides and their evaluation as inhibitors of HCV NS5B polymeraseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2014, 24 (12) : 2699 - 2702Chapron, Christopher论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USAGlen, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Peakdale Mol Ltd, Chapel En Le Frith SK23 0PG, Derby, England Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USALa Colla, Massimiliano论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USAMayes, Benjamin A.论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, CMC Dept, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USAMcCarville, Joseph F.论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USAMoore, Stephen论文数: 0 引用数: 0 h-index: 0机构: Peakdale Mol Ltd, Chapel En Le Frith SK23 0PG, Derby, England Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USAMoussa, Adel论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, CMC Dept, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USASarkar, Ruhul论文数: 0 引用数: 0 h-index: 0机构: Peakdale Mol Ltd, Chapel En Le Frith SK23 0PG, Derby, England Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USASeifer, Maria论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USASerra, Ilaria论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USAStewart, Alistair论文数: 0 引用数: 0 h-index: 0机构: Idenix Pharmaceut, CMC Dept, Cambridge, MA 02141 USA Idenix Pharmaceut, Dept Biol, Cambridge, MA 02141 USA
- [42] 2-(3-Thienyl)-5,6-dihydroxypyrimidine-4-carboxylic acids as inhibitors of HCV NS5B RdRpBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (21) : 6245 - 6249Pacini, Barbara论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyAvolio, Salvatore论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyErcolani, Caterina论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyKoch, Uwe论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyMigliaccio, Giovanni论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyNarjes, Frank论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyPacini, Laura论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyTomei, Licia论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, ItalyHarper, Steven论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs Rome, IRBM, I-00040 Rome, Italy Merck Res Labs Rome, IRBM, I-00040 Rome, Italy
- [43] Non-nucleoside inhibitors of HCV polymerase NS5B. Part 2: Synthesis and structure-activity relationships of benzothiazine-substituted quinolinedionesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (13) : 3642 - 3646de Vicente, Javier论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAHendricks, Robert T.论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USASmith, David B.论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAFell, Jay B.论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAFischer, John论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USASpencer, Stacey R.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAStengel, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAMohr, Peter论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USARobinson, John E.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USABlake, James F.论文数: 0 引用数: 0 h-index: 0机构: Array BioPharma Inc, Boulder, CO 80301 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAHilgenkamp, Ramona K.论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAYee, Calvin论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAAdjabeng, George论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAElworthy, Todd R.论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USATracy, Jahari论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAChin, Elbert论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USALi, Jim论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAWang, Beihan论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USABamberg, Joe T.论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAStephenson, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAOshiro, Connie论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAHarris, Seth F.论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAGhate, Manjiri论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USALeveque, Vincent论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USANajera, Isabel论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USALe Pogam, Sophie论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USARajyaguru, Sonal论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAAo-Ieong, Gloria论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAAlexandrova, Ludmila论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USALarrabee, Susan论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USABrandl, Michael论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USABriggs, Andrew论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USASukhtankar, Sunil论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAFarrell, Robert论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USAXu, Brian论文数: 0 引用数: 0 h-index: 0机构: Roche Palo Alto LLC, Palo Alto, CA 94304 USA Roche Palo Alto LLC, Palo Alto, CA 94304 USA
- [44] Novel HCV NS5B polymerase inhibitors: Discovery of indole 2-carboxylic acids with C3-heterocyclesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2011, 242Anilkumar, Gopinadhan N.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USALesburg, Charles论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USASelyutin, Oleg论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USARosenblum, Stuart B.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAZeng, Qingbei论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAJiang, Yueheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAChan, Tin-Yau论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAPu, Haiyan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAVaccaro, Henry论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAWang, Li论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USABennet, Frank论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAChen, Kevin X.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USADuca, Jose论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAGavalas, Stephen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAHuang, Yuhua论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAPinto, Patrick论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USASannigrahi, Mousumi论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAVelazquez, Francisco论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAVenkatraman, Srikanth论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAVibulbhan, Bancha论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAAgrawal, Sony论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAButkiewicz, Nancy论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAFerrari, Eric论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAFeld, Boris论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAHe, Zhiqing论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAJiang, Chuan-kui论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAPalermo, Robert E.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAHuang, H. -C.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAShih, Neng-Yang论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USANjoroge, George论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USAKozlowski, Joseph A.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Kenilworth, NJ 07033 USA Merck Res Labs, Kenilworth, NJ 07033 USA
- [45] A 2′-DEOXY-2′-FLUORO-2′-C-METHYL URIDINE CYCLOPENTYL CARBOCYCLIC ANALOG AND ITS PHOSPHORAMIDATE PRODRUG AS INHIBITORS OF HCV NS5B POLYMERASENUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS, 2012, 31 (04): : 277 - 285Liu, Jian论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USADu, Jinfa论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USAWang, Peiyuan论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USANagarathnam, Dhanapalan论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USAEspiritu, Christine L.论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USABao, Haiying论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USAMurakami, Eisuke论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USAFurman, Phillip A.论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USASofia, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Pharmasset Inc, Princeton, NJ USA Pharmasset Inc, Princeton, NJ USA
- [46] Design, synthesis, and structure-activity relationships of novel imidazo [4,5-c] pyridine derivatives as potent non-nucleoside inhibitors of hepatitis C virus NS5BBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (09) : 2621 - 2631Liu, Moyi论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaXu, Qiaoling论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaGuo, Su论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaZuo, Ruixi论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaHong, Yue论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaLuo, Yong论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaLi, Yingxiu论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaGong, Ping论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R ChinaLiu, Yajing论文数: 0 引用数: 0 h-index: 0机构: Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China Shenyang Pharmaceut Univ, Minist Educ, Key Lab Struct Based Drug Design & Discovery, 103 Wenhua Rd, Shenyang 110016, Liaoning, Peoples R China
- [47] Synthesis of 2′-deoxy-2′-fluoro-2′-C-methyl spiro cyclopentyl carbocyclic uridine analog as potential inhibitors of HCV NS5B polymeraseNUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS, 2020, 39 (1-3): : 52 - 68Singh, Uma S.论文数: 0 引用数: 0 h-index: 0机构: Univ Georgia, Coll Pharm, Dept Pharmaceut & Biomed Sci, Athens, GA 30602 USA Univ Georgia, Coll Pharm, Dept Pharmaceut & Biomed Sci, Athens, GA 30602 USAChu, Chung K.论文数: 0 引用数: 0 h-index: 0机构: Univ Georgia, Coll Pharm, Dept Pharmaceut & Biomed Sci, Athens, GA 30602 USA Univ Georgia, Coll Pharm, Dept Pharmaceut & Biomed Sci, Athens, GA 30602 USA
- [48] 5,5′- and 6,6′-Dialkyl-5,6-dihydro-1H-pyridin-2-ones as potent inhibitors of HCV NS5B polymeraseBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (21) : 6047 - 6052Ellis, David A.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USABlazel, Julie K.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USATran, Chinh V.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USARuebsam, Frank论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAMurphy, Douglas E.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USALi, Lian-Sheng论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAZhao, Jingjing论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAZhou, Yuefen论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAMcGuire, Helen M.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAXiang, Alan X.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAWebber, Stephen E.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAZhao, Qiang论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAHan, Qing论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAKissinger, Charles R.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USALardy, Matthew论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAGobbi, Alberto论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAShowalter, Richard E.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAShah, Amit M.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USATsan, Mei论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAPatel, Rupal A.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USALeBrun, Laurie A.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAKamran, Ruhi论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USABartkowski, Darian M.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USANolan, Thomas G.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USANorris, Daniel A.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USASergeeva, Maria V.论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USAKirkovsky, Leo论文数: 0 引用数: 0 h-index: 0机构: Anadys Pharmaceut Inc, San Diego, CA 92121 USA Anadys Pharmaceut Inc, San Diego, CA 92121 USA
- [49] Discovery of thiophene-2-carboxylic acids as potent inhibitors of HCVNS5B polymerase and HCV subgenomic RNA replication.: Part 2:: Tertiary amidesBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (03) : 797 - 800Chan, L论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaPereira, O论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaReddy, TJ论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaDas, SK论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaPoisson, C论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaCourchesne, M论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaProulx, M论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaSiddiqui, A论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaYannopoulos, CG论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaNguyen-Ba, N论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaRoy, C论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaNasturica, D论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaMoinet, C论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaBethell, R论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaHamel, M论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaL'Heureux, L论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaDavid, M论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaNicolas, O论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaCourtemanche-Asselin, P论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaBrunette, S论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaBilimoria, D论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, CanadaBédard, J论文数: 0 引用数: 0 h-index: 0机构: Shire BioChem Inc, Laval, PQ H7V 4A7, Canada Shire BioChem Inc, Laval, PQ H7V 4A7, Canada
- [50] Discovery of thienoimidazole-based HCV NS5A inhibitors. Part 2: Non-symmetric inhibitors with potent activity against genotype 1a and 1bBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2015, 25 (04) : 940 - 943Giroux, Simon论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USABilimoria, Darius论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USACadilhac, Caroline论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USACottrell, Kevin M.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USADenis, Francois论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USADietrich, Evelyne论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USAEwing, Nigel论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAHenderson, James A.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAL'Heureux, Lucille论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USAMani, Nagraj论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAMorris, Mark论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USANicolas, Olivier论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USAReddy, T. Jagadeeswar论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USASelliah, Subajini论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USAShawgo, Rebecca S.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAXu, Jinwang论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAChauret, Nathalie论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USABerlioz-Seux, Francoise论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAChan, Laval C.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USADas, Sanjoy K.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Canada Inc, Laval, PQ H7V 4A7, Canada Vertex Pharmaceut Inc, Boston, MA 02210 USAGrillot, Anne-Laure论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USABennani, Youssef L.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USAMaxwell, John P.论文数: 0 引用数: 0 h-index: 0机构: Vertex Pharmaceut Inc, Boston, MA 02210 USA Vertex Pharmaceut Inc, Boston, MA 02210 USA