Tetrahydrobenzothiophenone derivatives as a novel class of adenosine receptor antagonists.

被引:0
|
作者
vanRhee, AM
Siddiqi, SM
Melman, N
Shi, D
Padgett, WL
Daly, JW
Jacobson, KA
机构
[1] NIDDK,NIH,LBC,MOL RECOGNIT SECT,BETHESDA,MD 20892
[2] NIDDK,NIH,LBC,PHARMACODYNAM SECT,BETHESDA,MD 20892
来源
FASEB JOURNAL | 1996年 / 10卷 / 03期
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:784 / 784
页数:1
相关论文
共 50 条
  • [31] Novel 2-benzyl-piperidine derivatives as selective M2 muscarinic receptor antagonists.
    Zhao, SH
    Berger, J
    Miller, AK
    Flippin, L
    Clark, R
    Maag, H
    Stepane, G
    Watson, N
    Shetty, SG
    Cefalu, JS
    Dawson, MW
    Rocha, C
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2001, 221 : U200 - U200
  • [32] Novel small molecule bradykinin B1 receptor antagonists. Part 3: Hydroxyurea derivatives
    Schnatbaum, Karsten
    Schaudt, Marco
    Stragies, Roland
    Pfeifer, Jochen R.
    Gibson, Christoph
    Locardi, Elsa
    Scharn, Dirk
    Richter, Uwe
    Kalkhof, Holger
    Dinkel, Klaus
    Zischinsky, Gunther
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (03) : 1233 - 1236
  • [33] Novel potent substance P and neurokinin A receptor antagonists.: Conception, synthesis and biological evaluation indolizine derivatives
    Millet, R
    Domarkas, J
    Rigo, B
    Goossens, L
    Goossens, JF
    Houssin, R
    Hénichart, JP
    BIOORGANIC & MEDICINAL CHEMISTRY, 2002, 10 (09) : 2905 - 2912
  • [34] Benzylidene ketal derivatives as M2 muscarinic receptor antagonists.
    Boyle, CD
    Chackalamannil, S
    Chen, LY
    Dugar, S
    Pushpavanam, P
    Billard, W
    Binch, H
    Crosby, G
    Coffin, VL
    Cohen-Williams, M
    Duffy, RA
    Ruperto, V
    Taylor, LA
    McQuade, RD
    Lachowicz, JE
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 220 : U556 - U556
  • [35] Sar and molecular modeling studies of pyridine derivatives as selective A3 adenosine antagonists.
    Li, AH
    Moro, S
    Melman, N
    Ji, XD
    Jacobson, KA
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1998, 216 : U229 - U229
  • [36] Design, synthesis and pharmacological evaluation of a novel class of potent, selective, orally active oxytocin receptor antagonists.
    Schwarz, MK
    Quattropani, A
    Page, P
    Thomas, RJ
    Baxter, A
    Dorbais, J
    Pomel, V
    Maio, M
    Mannino, C
    Covini, D
    Pittet, PA
    Jorand-Lebrun, C
    Valognes, D
    Halazy, S
    Scheer, A
    Missotten, M
    Ayala, G
    Cirillo, R
    Tos, EG
    Marinelli, P
    Giacchetti, C
    Barberis, C
    Chollet, A
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2003, 226 : U69 - U69
  • [37] Novel adenosine antagonists: A(3) receptor-selective flavonoid and dihydropyridine derivatives.
    Jacobson, KA
    vanRhee, AM
    Jiang, L
    Ji, XD
    Karton, Y
    vonLubitz, DKJE
    Olah, ME
    Stiles, GL
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1996, 212 : 99 - MEDI
  • [38] Novel urea derivatives that are highly potent VLA-4 antagonists.
    Kassir, JL
    Grabbe, VO
    Biediger, RJ
    Scott, IL
    Market, RV
    Raju, BG
    Lin, SQ
    Dupre, B
    Kogan, TP
    Chan, Q
    Yu, T
    Holland, GW
    Maxwell, DC
    Vanderslice, P
    West, H
    Decker, ER
    Bourgoyne, A
    Tilton, R
    Munsch, CL
    Dixon, RAF
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 220 : U568 - U568
  • [39] Novel small molecule GLP-1 receptor antagonists: A comparison with peptide antagonists.
    Kiel, D
    Lakis, JN
    Gonzalez, J
    Rajapakse, R
    May, JM
    FASEB JOURNAL, 2000, 14 (08): : A1351 - A1351
  • [40] Diamine derivatives containing imidazolidinylidene propanedinitrile as a new class of histamine H3 receptor antagonists.: Part I
    Sasho, Setsuya
    Seishi, Takashi
    Kawamura, Mariko
    Hirose, Ryo
    Toki, Shinichiro
    Shimada, Jun-ich
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2008, 18 (07) : 2288 - 2291