Synthesis of 1-Acyl-3-isopropenylbenzimidazolone Derivatives and Their Activity against Botrytis cinerea

被引：25

作者：

Li, Sheng-Kun ^{[1
]}

Ji, Zhi-Qin ^{[1
]}

Zhang, Ji-Wen ^{[1
]}

Guo, Zheng-Yan ^{[1
]}

Wu, Wen-Jun ^{[1
,2
]}

机构：

[1] NW A&F Univ, Inst Pesticide Sci, Yangling 712100, Shaanxi, Peoples R China

[2] Nankai Univ, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China

来源：

JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | 2010年 / 58卷 / 05期

基金：

中国国家自然科学基金;

关键词：

Benzimidazolone derivatives; synthesis; fungicidal activities; BENZIMIDAZOLONE DERIVATIVES; ACTIVATORS;

D O I：

10.1021/jf903855y

中图分类号：

S [农业科学];

学科分类号：

09 ;

摘要：

A series of 1-acyl-3-isopropenylbenzimidazolone derivatives were synthesized, and their structures were characterized by H-1 and C-13 NMR and elemental analysis. Their fungicidal activities against Botrytis cinerea were also evaluated by spore germination assay. The acrylic acid, methacrylic acid, 4-chlorophenyl acetic acid, and 2-chlorobenzoic acid derivatives exhibited strong fungicidal activity. This implied that benzimidazolones might be potential fungicide leading compounds.

引用

页码：2668 / 2672

页数：5

共 50 条

[31] Semisynthesis and Antifungal Activity of Novel Oxime Ester Derivatives of Carabrone Modified at C(4) against Botrytis cinerea
Wang, Delong
Ren, Shuangxi
Wang, Hao
Yan, He
Feng, Juntao
Zhang, Xing
CHEMISTRY & BIODIVERSITY, 2014, 11 (06) : 886 - 903
[32] Antifungal activity of thymol and carvacrol against postharvest pathogens Botrytis cinerea
Jihong Zhang
Shuang Ma
Shenglong Du
Shaoyang Chen
Helong Sun
Journal of Food Science and Technology, 2019, 56 : 2611 - 2620
[33] Phytotoxic Activity and Metabolism of Botrytis cinerea and Structure-Activity Relationships of Isocaryolane Derivatives
Ascari, Jociani
Diamantino Boaventura, Maria Amelia
Takahashi, Jacqueline Aparecida
Duran-Patron, Rosa
Hernandez-Galan, Rosario
Macias-Sanchez, Antonio J.
Collado, Isidro G.
JOURNAL OF NATURAL PRODUCTS, 2013, 76 (06): : 1016 - 1024
[34] Synthesis, Fungicidal Activity and SAR of 2-Thiazolamide/Pyrazolamide-Cyclohexylsulfonamides against Botrytis cinerea
Zhang, Shen
Meng, Siqi
Xie, Yong
Yang, Yonggui
Zhang, Yumeng
He, Lu
Wang, Kai
Qi, Zhiqiu
Ji, Mingshan
Qin, Peiwen
Li, Xinghai
MOLECULES, 2019, 24 (14):
[35] Synthesis and Fungistatic Activity of Bicyclic Lactones and Lactams against Botrytis cinerea, Penicillium citrinum, and Aspergillus glaucus
Walczak, Paulina
Pannek, Jakub
Boratynski, Filip
Janik-Polanowicz, Agata
Olejniczak, Teresa
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2014, 62 (34) : 8571 - 8578
[36] Activity and metabolism of cyano-oxime derivatives in various strains of Botrytis cinerea
Tellier, F
Carlin-Sinclair, A
Fritz, R
Cherton, JC
Leroux, P
PESTICIDE BIOCHEMISTRY AND PHYSIOLOGY, 2004, 78 (03) : 151 - 160
[37] Synthesis, Bioactivity, and QSAR Study of 3,4-Dichlorophenyl Isoxazole-Substituted Stilbene Derivatives against the Phytopathogenic Fungus Botrytis cinerea
Lin, Xingdong
Li, Yan
Zhong, Weiqiang
Hong, Tian
Li, Lihuang
Song, Shaoyun
He, Daohang
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2021, 69 (33) : 9520 - 9528
[38] Synthesis, Bioactivity, and QSAR Study of 3,4-Dichlorophenyl Isoxazole-Substituted Stilbene Derivatives against the Phytopathogenic Fungus Botrytis cinerea
He, Daohang (cehdh@scut.edu.cn), 1600, American Chemical Society (69):
[39] Synthesis and antifungal property of N-(aryl) and quaternary N-(aryl) chitosan derivatives against Botrytis cinerea
Badawy, Mohamed E. I.
Rabea, Entsar I.
CELLULOSE, 2014, 21 (04) : 3121 - 3137
[40] Global Antifungal Profile Optimization of Chlorophenyl Derivatives against Botrytis cinerea and Colletotrichum gloeosporioides
Saiz-Urra, Liane
Bustillo Perez, Antonio J.
Cruz-Monteagudo, Maykel
Pinedo-Rivilla, Cristina
Aleu, Josefina
Hernandez-Galan, Rosario
Collado, Isidro G.
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY, 2009, 57 (11) : 4838 - 4843

← 1 2 3 4 5 →