Synthesis of 1-Acyl-3-isopropenylbenzimidazolone Derivatives and Their Activity against Botrytis cinerea

被引：25
|
作者：
Li, Sheng-Kun [1 ]
Ji, Zhi-Qin [1 ]
Zhang, Ji-Wen [1 ]
Guo, Zheng-Yan [1 ]
Wu, Wen-Jun [1 ,2 ]
机构：
[1] NW A&F Univ, Inst Pesticide Sci, Yangling 712100, Shaanxi, Peoples R China
[2] Nankai Univ, State Key Lab Elementoorgan Chem, Tianjin 300071, Peoples R China
来源：
JOURNAL OF AGRICULTURAL AND FOOD CHEMISTRY | 2010年 / 58卷 / 05期
基金：
中国国家自然科学基金;
关键词：
Benzimidazolone derivatives; synthesis; fungicidal activities; BENZIMIDAZOLONE DERIVATIVES; ACTIVATORS;
D O I：
10.1021/jf903855y
中图分类号：
S [农业科学];
学科分类号：
09 ;
摘要：
A series of 1-acyl-3-isopropenylbenzimidazolone derivatives were synthesized, and their structures were characterized by H-1 and C-13 NMR and elemental analysis. Their fungicidal activities against Botrytis cinerea were also evaluated by spore germination assay. The acrylic acid, methacrylic acid, 4-chlorophenyl acetic acid, and 2-chlorobenzoic acid derivatives exhibited strong fungicidal activity. This implied that benzimidazolones might be potential fungicide leading compounds.
引用
收藏
页码：2668 / 2672
页数：5
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