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- [32] Identification of C-2 Hydroxyethyl Imidazopyrrolopyridines as Potent JAK1 Inhibitors with Favorable Physicochemical Properties and High Selectivity over JAK2JOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (11) : 4764 - 4785Zak, Mark论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHurley, Christopher A.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAWard, Stuart I.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABergeron, Philippe论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABarrett, Kathy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABalazs, Mercedesz论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABlair, Wade S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USABull, Richard论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAChakravarty, Paroma论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Small Mol Pharmaceut Sci, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAChang, Christine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USACrackett, Peter论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADeshmukh, Gauri论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADeVoss, Jason论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USADragovich, Peter S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAEigenbrot, Charles论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAEllwood, Charles论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGaines, Simon论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGhilardi, Nico论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGibbons, Paul论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGradl, Stefan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAGribling, Peter论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHamman, Chris论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHarstad, Eric论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Safety Assessment, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAHewitt, Peter论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJohnson, Adam论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAJohnson, Tony论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKenny, Jane R.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKoehler, Michael F. T.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKohli, Pawan Bir论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALabadie, Sharada论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALee, Wyne P.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Immunol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALiao, Jiangpeng论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USALiimatta, Marya论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAMendonca, Rohan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USANarukulla, Raman论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAPulk, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAReeve, Austin论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USASavage, Scott论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Small Mol Proc Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAShia, Steven论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USASteffek, Micah论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biol Struct, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAUbhayakar, Savita论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Drug Metab & Pharmacokinet, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAvan Abbema, Anne论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Biochem & Cellular Pharmacol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAAliagas, Ignacio论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAAvitabile-Woo, Barbara论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAXiao, Yisong论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAYang, Jing论文数: 0 引用数: 0 h-index: 0机构: WuXi AppTec Co Ltd, Shanghai 200131, Peoples R China Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USAKulagowski, Janusz J.论文数: 0 引用数: 0 h-index: 0机构: Argenta, Spire Green Ctr 8 9, Harlow CM19 5TR, Essex, England Genentech Inc, Dept Discovery Chem, San Francisco, CA 94080 USA
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- [34] Different CALR mutation subtypes in essential thrombocythemia and primary myelofibrosis patients without JAK2 mutationmemo - Magazine of European Medical Oncology, 2020, 13 : 235 - 243Layla M. Saleh论文数: 0 引用数: 0 h-index: 0机构: Mansoura University,Hematology Laboratory, Oncology CenterReem Algamal论文数: 0 引用数: 0 h-index: 0机构: Mansoura University,Hematology Laboratory, Oncology CenterHanaa Abd Elmasseh论文数: 0 引用数: 0 h-index: 0机构: Mansoura University,Hematology Laboratory, Oncology CenterEmily Barber论文数: 0 引用数: 0 h-index: 0机构: Mansoura University,Hematology Laboratory, Oncology CenterHasan Abdel-ghaffar论文数: 0 引用数: 0 h-index: 0机构: Mansoura University,Hematology Laboratory, Oncology Center
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- [36] Long-term outcomes of 107 patients with myelofibrosis receiving JAK1/JAK2 inhibitor ruxolitinib: survival advantage in comparison to matched historical controlsBLOOD, 2012, 120 (06) : 1202 - 1209Verstovsek, Srdan论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAKantarjian, Hagop M.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAEstrov, Zeev论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USACortes, Jorge E.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAThomas, Deborah A.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAKadia, Tapan论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAPierce, Sherry论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAJabbour, Elias论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USABorthakur, Gautham论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USARumi, Elisa论文数: 0 引用数: 0 h-index: 0机构: Univ Pavia, Dept Hematol Oncol, Fdn IRCCS Policlin San Matteo, I-27100 Pavia, Italy Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAPungolino, Ester论文数: 0 引用数: 0 h-index: 0机构: Osped Niguarda Ca Granda, Milan, Italy Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAMorra, Enrica论文数: 0 引用数: 0 h-index: 0机构: Osped Niguarda Ca Granda, Milan, Italy Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USACaramazza, Domenica论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Osped Circolo & Fdn Macchi, Dept Internal Med, Div Hematol, Varese, Italy Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USACazzola, Mario论文数: 0 引用数: 0 h-index: 0机构: Univ Pavia, Dept Hematol Oncol, Fdn IRCCS Policlin San Matteo, I-27100 Pavia, Italy Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USAPassamonti, Francesco论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Osped Circolo & Fdn Macchi, Dept Internal Med, Div Hematol, Varese, Italy Univ Texas MD Anderson Canc Ctr, Leukemia Dept, Houston, TX 77030 USA
- [37] Structure-based discovery of C-2 substituted imidazo-pyrrolopyridine JAK1 inhibitors with improved selectivity over JAK2ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 246Labadie, Sharada S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA 94080 USA Genentech Inc, San Francisco, CA 94080 USA
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- [40] Structure-based discovery of C-2 substituted imidazo-pyrrolopyridine JAK1 inhibitors with improved selectivity over JAK2BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (24) : 7627 - 7633Labadie, Sharada论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USADragovich, Peter S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USABarrett, Kathy论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USABlair, Wade S.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USABergeron, Philippe论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USAChang, Christine论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USADeshmukh, Gauri论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USAEigenbrot, Charles论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USAGhilardi, Nico论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USAGibbons, Paul论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 USA Genentech Inc, Small Mol Discovery Chem, San Francisco, CA 94080 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