Fragment-Based Lead Discovery

被引:19
|
作者
Congreve, Miles [1 ]
Murray, Christopher W. [1 ]
Carr, Robin [1 ]
Rees, David C. [1 ]
机构
[1] Astex Therapeut, Cambridge CB4 0QA, England
关键词
D O I
10.1016/S0065-7743(07)42028-0
中图分类号
R914 [药物化学];
学科分类号
100701 ;
摘要
[No abstract available]
引用
收藏
页码:431 / 448
页数:18
相关论文
共 50 条
  • [21] Integrated biophysical approach to fragment screening and validation for fragment-based lead discovery
    Silvestre, Hernani Leonardo
    Blundell, Thomas L.
    Abell, Chris
    Ciulli, Alessio
    PROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2013, 110 (32) : 12984 - 12989
  • [22] Fragment-based lead discovery and optimization using the SHAPES strategy
    Lepre, CA
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 230 : U2762 - U2762
  • [23] Capitalizing on Fragment-Based Discovery
    Liszewski, Kathy
    GENETIC ENGINEERING & BIOTECHNOLOGY NEWS, 2009, 29 (08): : 18 - +
  • [24] Fragment-based drug discovery
    Erlanson, DA
    McDowell, RS
    O'Brien, T
    JOURNAL OF MEDICINAL CHEMISTRY, 2004, 47 (14) : 3463 - 3482
  • [25] Fragment-based drug discovery
    Wendy A. Warr
    Journal of Computer-Aided Molecular Design, 2009, 23 : 453 - 458
  • [26] fragment-based ligand discovery
    Fischer, Marcus
    Hubbard, Roderick E.
    MOLECULAR INTERVENTIONS, 2009, 9 (01) : 22 - 30
  • [27] Fragment-based drug discovery
    Warr, Wendy A.
    JOURNAL OF COMPUTER-AIDED MOLECULAR DESIGN, 2009, 23 (08) : 453 - 458
  • [28] Fragment-Based Drug Discovery
    Norton, Raymond S.
    AUSTRALIAN JOURNAL OF CHEMISTRY, 2013, 66 (12) : 1463 - 1464
  • [29] Fragment-based discovery in spotlight
    Lipp, Elizabeth
    GENETIC ENGINEERING & BIOTECHNOLOGY NEWS, 2007, 27 (19): : 22 - +
  • [30] Fragment-based lead design
    Tarasova, Olga A.
    Poroikov, V. V.
    RUSSIAN CHEMICAL REVIEWS, 2012, 81 (02) : 158 - 174