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- [41] Novel Microtubule Polymerization Inhibitor with Potent Antiproliferative and Antitumor ActivityCANCER RESEARCH, 2009, 69 (05) : 1910 - 1915Arora, Sonia论文数: 0 引用数: 0 h-index: 0机构: Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USAWang, Xin I.论文数: 0 引用数: 0 h-index: 0机构: Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USAKeenan, Susan M.论文数: 0 引用数: 0 h-index: 0机构: Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USAAndaya, Christina论文数: 0 引用数: 0 h-index: 0机构: Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USAZhang, Qiang论文数: 0 引用数: 0 h-index: 0机构: Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USAPeng, Youyi论文数: 0 引用数: 0 h-index: 0机构: Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USAWelsh, William J.论文数: 0 引用数: 0 h-index: 0机构: Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USA Univ Med & Dent New Jersey, Robert Wood Johnson Med Sch, Dept Pharmacol, Piscataway, NJ 08854 USA
- [42] Discovery of Novel Potent VEGFR-2 Inhibitors Exerting Significant Antiproliferative Activity against Cancer Cell LinesJOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (01) : 140 - 157Zhang, Yanmin论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaChen, Yadong论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaZhang, Danfeng论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaWang, Lu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaLu, Tao论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, State Key Lab Nat Med, 24 Tongjiaxiang, Nanjing 210009, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R ChinaJiao, Yu论文数: 0 引用数: 0 h-index: 0机构: China Pharmaceut Univ, Sch Sci, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China China Pharmaceut Univ, Sch Sci, Lab Mol Design & Drug Discovery, 639 Longmian Ave, Nanjing 211198, Jiangsu, Peoples R China
- [43] Discovery of a potent and selective Bcl-2 inhibitor using SAR by NMRBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2010, 20 (22) : 6587 - 6591Petros, Andrew M.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAHuth, Jeffrey R.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAOost, Thorsten论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAPark, Cheol-Min论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USADing, Hong论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAWang, Xilu论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAZhang, Haichao论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USANimmer, Paul论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMendoza, Renaldo论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USASun, Chaohong论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAMack, Jamey论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAWalter, Karl论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USADorwin, Sarah论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAGramling, Emily论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USALadror, Uri论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USARosenberg, Saul H.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAElmore, Steven W.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAFesik, Stephen W.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USAHajduk, Philip J.论文数: 0 引用数: 0 h-index: 0机构: Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA Abbott Labs, Dept R460, Global Pharmaceut Res & Dev, Abbott Pk, IL 60064 USA
- [44] Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279JOURNAL OF MEDICINAL CHEMISTRY, 2023, 66 (15) : 10473 - 10496Leit, Silvana论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAGreenwood, Jeremy论文数: 0 引用数: 0 h-index: 0机构: Schrodinger Inc, New York, NY 10036 USA Nimbus Therapeut, Boston, MA 02210 USACarriero, Samantha论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAMondal, Sayan论文数: 0 引用数: 0 h-index: 0机构: Schrodinger Inc, New York, NY 10036 USA Nimbus Therapeut, Boston, MA 02210 USAAbel, Robert论文数: 0 引用数: 0 h-index: 0机构: Schrodinger Inc, New York, NY 10036 USA Nimbus Therapeut, Boston, MA 02210 USAAshwell, Mark论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USABlanchette, Heather论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USABoyles, Nicholas A. A.论文数: 0 引用数: 0 h-index: 0机构: Schrodinger Inc, New York, NY 10036 USA Nimbus Therapeut, Boston, MA 02210 USACartwright, Mark论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USACollis, Alan论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAFeng, Shulu论文数: 0 引用数: 0 h-index: 0机构: Schrodinger Inc, New York, NY 10036 USA Nimbus Therapeut, Boston, MA 02210 USAGhanakota, Phani论文数: 0 引用数: 0 h-index: 0机构: Schrodinger Inc, New York, NY 10036 USA Nimbus Therapeut, Boston, MA 02210 USAHarriman, Geraldine C. C.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAHosagrahara, Vinayak论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAKaila, Neelu论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAKapeller, Rosanna论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USARafi, Salma B. B.论文数: 0 引用数: 0 h-index: 0机构: Schrodinger Inc, New York, NY 10036 USA Nimbus Therapeut, Boston, MA 02210 USARomero, Donna L. L.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USATarantino, Paul M. M.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USATimaniya, Jignesh论文数: 0 引用数: 0 h-index: 0机构: Piramal Pharm Solut, Ahmadabad 382215, Gujarat, India Nimbus Therapeut, Boston, MA 02210 USAToms, Angela V. V.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAWester, Ronald T. T.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAWestlin, William论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USASrivastava, Bhaskar论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAMiao, Wenyan论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USATummino, Peter论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAMcElwee, Joshua J. J.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAEdmondson, Scott D. D.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USAMasse, Craig E. E.论文数: 0 引用数: 0 h-index: 0机构: Nimbus Therapeut, Boston, MA 02210 USA Nimbus Therapeut, Boston, MA 02210 USA
- [45] Discovery of remogliflozin etabonate: A potent and highly selective SGLT2 inhibitorBIOORGANIC & MEDICINAL CHEMISTRY, 2021, 34Shimizu, Kazuo论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Toho Univ, Fac Pharmaceut Sci, 2-2-1 Miyama, Funabashi, Chiba 2748510, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanFujikura, Hideki论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanFushimi, Nobuhiko论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanNishimura, Toshihiro论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanTatani, Kazuya论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanKatsuno, Kenji论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanFujimori, Yoshikazu论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanWatanabe, Shinjiro论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanHiratochi, Masahiro论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanNakabayashi, Takeshi论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanKamada, Noboru论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanArakawa, Koichi论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanHikawa, Hidemasa论文数: 0 引用数: 0 h-index: 0机构: Toho Univ, Fac Pharmaceut Sci, 2-2-1 Miyama, Funabashi, Chiba 2748510, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanAzumaya, Isao论文数: 0 引用数: 0 h-index: 0机构: Toho Univ, Fac Pharmaceut Sci, 2-2-1 Miyama, Funabashi, Chiba 2748510, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, JapanIsaji, Masayuki论文数: 0 引用数: 0 h-index: 0机构: Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan Kissei Pharmaceut Co Ltd, Cent Res Lab, 4365-1 Hotakakashiwabara, Azumino, Nagano 3998304, Japan
- [46] Selective ALK inhibitor alectinib with potent antitumor activity in models of crizotinib resistanceCANCER LETTERS, 2014, 351 (02) : 215 - 221Kodama, Tatsushi论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanTsukaguchi, Toshiyuki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanYoshida, Miyuki论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanKondoh, Osamu论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, JapanSakamoto, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan Chugai Pharmaceut Co Ltd, Div Res, Kamakura, Kanagawa 2478530, Japan
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