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- [31] Rapid approach to identification of a PDE10A tracer to support development of PDE10A inhibitors in preclinical and clinical studiesABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 246Harrington, Essa Hu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAMa, Ji论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USABiorn, Christopher论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USALester-Zeiner, Dianna论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USACho, Robert论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USARumfelt, Shannon论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAKunz, Roxanne论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USANixey, Thomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAMichelsen, Klaus论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAMiller, Silke论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAShi, Jianxia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USADella Puppa, Geraldine Hill论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USATalreja, Santosh论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAAble, Jessica论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAHwang, Dah-Ren论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USASlifstein, Mark论文数: 0 引用数: 0 h-index: 0机构: Columbia Univ, Dept Psychiat, New York, NY 10032 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAEaswaramoorthy, Balu论文数: 0 引用数: 0 h-index: 0机构: Columbia Univ, Dept Psychiat, New York, NY 10032 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAHitchcock, Stephen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Envoy Therapeut, Jupiter, FL 33458 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAPorter, Amy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAAllen, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAImmke, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USATreanor, James论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USAChen, Hang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Dept PKDM, San Francisco, CA 94080 USA Amgen Inc, Dept Small Mol Chem, Dept Neurosci,Dept PKDM,Dept Mol Struct, Dept Med Sci, Thousand Oaks, CA 91320 USA
- [32] Novel benzimidazole derivatives as phosphodiesterase 10A (PDE10A) inhibitors with improved metabolic stabilityBIOORGANIC & MEDICINAL CHEMISTRY, 2014, 22 (13) : 3515 - 3526Chino, Ayaka论文数: 0 引用数: 0 h-index: 0机构: Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanMasuda, Naoyuki论文数: 0 引用数: 0 h-index: 0机构: Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanAmano, Yasushi论文数: 0 引用数: 0 h-index: 0机构: Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanHonbou, Kazuya论文数: 0 引用数: 0 h-index: 0机构: Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanMihara, Takuma论文数: 0 引用数: 0 h-index: 0机构: Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanYamazaki, Mayako论文数: 0 引用数: 0 h-index: 0机构: Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, JapanTomishima, Masaki论文数: 0 引用数: 0 h-index: 0机构: Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan Inst Drug Discovery Res, Tsukuba, Ibaraki 3058585, Japan
- [33] Discovery of Potent, Selective, and Peripherally Restricted Pan-Trk Kinase Inhibitors for the Treatment of PainJOURNAL OF MEDICINAL CHEMISTRY, 2018, 61 (15) : 6779 - 6800Bagal, Sharan K.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandAndrews, Mark论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Sandwich CT13 9NJ, Kent, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandBechle, Bruce M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Groton Labs, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandBian, Jianwei论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Groton Labs, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandBilsland, James论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandBlakemore, David C.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandBraganza, John F.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandBungay, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Pharmacokinet Dynam & Metab, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandCorbett, Matthew S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Groton Labs, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandCronin, Ciaran N.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandCui, Jingrong Jean论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandDias, Rebecca论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandFlanagan, Neil J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandGreasley, Samantha E.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandGrimley, Rachel论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandJames, Kim论文数: 0 引用数: 0 h-index: 0机构: Peakdale Mol, Discovery Pk House,Ramsgate Rd, Sandwich CT13 9ND, Kent, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandJohnson, Eric论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandKitching, Linda论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandKraus, Michelle L.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandMcAlpine, Indrawan论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandNagata, Asako论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandNinkovic, Sacha论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, 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La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandWaldron, Gareth J.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D UK, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandWang, Fen论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, La Jolla Labs, 10770 Sci Ctr Dr, San Diego, CA 92121 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, EnglandWarmus, Joseph S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Worldwide R&D, Groton Labs, Eastern Point Rd, Groton, CT 06340 USA Pfizer Worldwide R&D UK, Worldwide Med Chem, Portway Bldg,Granta Pk, Cambridge CB21 6GS, England
- [34] Quetiapine and novel PDE10A inhibitors potentiate the anti-BuChE activity of donepezilJOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2020, 35 (01) : 1743 - 1750Sikora, Joanna论文数: 0 引用数: 0 h-index: 0机构: Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, PolandPodsiedlik, Maria论文数: 0 引用数: 0 h-index: 0机构: Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lodz, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, PolandPietras, Tadeusz论文数: 0 引用数: 0 h-index: 0机构: Med Univ Lodz, Dept Clin Pharmacol, Lodz, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, PolandKosmalski, Marcin论文数: 0 引用数: 0 h-index: 0机构: Med Univ Lodz, Dept Clin Pharmacol, Lodz, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, PolandMatloka, Mikolaj论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, Res & Dev Dept, Lomianki, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, PolandMoszczynski-Petkowski, Rafal论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, Res & Dev Dept, Lomianki, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, PolandWieczorek, Maciej论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, Res & Dev Dept, Lomianki, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, PolandMarkowicz-Piasecka, Magdalena论文数: 0 引用数: 0 h-index: 0机构: Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, Poland Med Univ Lodz, Dept Pharmaceut Chem Drug Anal & Radiopharm, Lab Bioanal, Ul Muszynskiego 1, PL-90151 Lodz, Poland
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