共 50 条
- [1] Discovery of novel potent imidazo[1,2-b]pyridazine PDE10a inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2016, 26 (17) : 4216 - 4222Meegalla, Sanath K.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAHuang, Hui论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAIllig, Carl R.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAParks, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAChen, Jinsheng论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USALee, Yu-Kai论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAWilson, Kenneth J.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAPatel, Sharmila K.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USACheung, Wing S.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USALu, Tianbao论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAKirchner, Thomas论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAAskari, Hossein B.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAGeisler, John论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAPatch, Raymond J.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAGibbs, Alan C.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USARady, Brian论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAConnelly, Margery论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USAPlayer, Mark R.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA Janssen Res & Dev, Welsh & McKean Rd, Spring House, PA 19477 USA
- [2] Novel quinazolines: Potent CNS-penetrable inhibitors of PDE10AABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Yang, Edward X.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USA Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USAChappie, Thomas A.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USA Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USAHumphrey, John M.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USA Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USAMenniti, Frank S.论文数: 0 引用数: 0 h-index: 0机构: Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USA Pfizer Inc, Neurosci Med Chem, Groton, CT 06340 USA
- [3] The discovery of potent, selective, and orally active pyrazoloquinolines as PDE10A inhibitors for the treatment of SchizophreniaBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (02) : 1019 - 1022Ho, Ginny D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAYang, Shu-Wei论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USASmotryski, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USABercovici, Ana论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USANechuta, Terry论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USASmith, Elizabeth M.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAMcElroy, William论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USATan, Zheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USATulshian, Deen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAMcKittrick, Brian论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAGreenlee, William J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAHruza, Alan论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Struct Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAXiao, Li论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Struct Chem, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USARindgen, Diane论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Drug Metab & Pharmacokinet, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAMullins, Deborra论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAGuzzi, Mario论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAZhang, Xiaoping论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USABleickardt, Carina论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USAHodgson, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Neurosci, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Med Chem, Kenilworth, NJ 07033 USA
- [4] Pyrazoloquinolines as PDE10A inhibitors: Discovery of a tool compoundBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (03) : 1335 - 1339McElroy, William T.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USATan, Zheng论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USABasu, Kallol论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USAYang, Shu-Wei论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USASmotryski, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USAHo, Ginny D.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USATulshian, Deen论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USAGreenlee, William J.论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USAMullins, Deborra论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurobiol Dept Biol Res, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USAGuzzi, Mario论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurobiol Dept Biol Res, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USAZhang, Xiaoping论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurobiol Dept Biol Res, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USABleickardt, Carina论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurobiol Dept Biol Res, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USAHodgson, Robert论文数: 0 引用数: 0 h-index: 0机构: Merck Res Labs, Neurobiol Dept Biol Res, Kenilworth, NJ 07033 USA Merck Res Labs, Dept Chem Res CV & CNS, Kenilworth, NJ 07033 USA
- [5] Discovery and quantitative pharmacology of novel azetidine-containing PDE10A inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2016, 252Liu, Qingyian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAAmegadzie, Albert论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAChen, Jian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAChen, Ning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAFrohn, Michael论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAHu, Essa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAKaller, Matthew论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAMa, Vu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USANguyen, Tom论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAPickrell, Alex论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAQian, Wenyuan论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USARumfelt, Shannon论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USARzasa, Robert论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAAndrews, Kristin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAZhao, Sharon论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USADavis, Carl论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAAble, Jessica论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAShi, Jianxia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USADella Puppa, Geraldine Hill论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USADovlatyan, Mary论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAChen, Hang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAMiller, Silke论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USATreanor, James论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAKornecook, Thomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAZhong, Wenge论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USAAllen, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Thousand Oaks, CA 91320 USA Amgen Inc, Thousand Oaks, CA 91320 USA
- [6] Discovery of Novel Imidazo[4,5-b]pyridines as Potent and Selective Inhibitors of Phosphodiesterase 10A (PDE10A)ACS MEDICINAL CHEMISTRY LETTERS, 2014, 5 (06): : 700 - 705Hu, Essa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAAndrews, Kristin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAChmait, Samer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USADavis, Carl论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAMiller, Silke论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USADella Puppa, Geraldine Hill论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USADovlatyan, Mary论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAChen, Hang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USALester-Zeiner, Dianna论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAAble, Jessica论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USABiorn, Christopher论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAMa, Ji论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAShi, Jianxia论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Pharmacokinet & Drug Metab, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USATreanor, James论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USAAllen, Jennifer R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA Amgen Inc, Dept Med Chem, One Amgen Ctr Dr, Thousand Oaks, CA 93012 USA
- [7] Discovery and synthesis of novel 3-alkoxy azetidines as PDE10A inhibitorsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2013, 246Rzasa, Robert M.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAFrohn, Michael J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAHorne, Daniel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAAndrews, Kristin L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAChmait, Samer论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USANguyen, Thomas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAKaller, Matthew R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAKunz, Roxanne K.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAChen, Ning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAHu, Essa论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAJones, Adrie D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAPickrell, Alex论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAReichelt, Andreas论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAPorter, Amy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAZhao, Xiaoning论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, San Francisco, CA 94080 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAEastwood, Heather论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Mol Struct & Characterizat, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAMiller, Silke论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USATreanor, James J. S.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Neurosci, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USAAllen, Jennifer R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA Amgen Inc, Dept Med Chem, Thousand Oaks, CA 91320 USA
- [8] New potent and selective PDE10A inhibitors for the treatment of schizophreniaABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240Malamas, Michael S.论文数: 0 引用数: 0 h-index: 0Ni, Yike论文数: 0 引用数: 0 h-index: 0Erdei, James论文数: 0 引用数: 0 h-index: 0Fan, Kristi论文数: 0 引用数: 0 h-index: 0Hoefgen, Norbert论文数: 0 引用数: 0 h-index: 0Stange, Hans论文数: 0 引用数: 0 h-index: 0Schindler, Rudolf论文数: 0 引用数: 0 h-index: 0Grunwald, Christian论文数: 0 引用数: 0 h-index: 0Egerland, Ute论文数: 0 引用数: 0 h-index: 0Langen, Barbara论文数: 0 引用数: 0 h-index: 0Hage, Thorsten论文数: 0 引用数: 0 h-index: 0Kronbach, Thomas论文数: 0 引用数: 0 h-index: 0Grauer, Steven论文数: 0 引用数: 0 h-index: 0Harrison, Boyd论文数: 0 引用数: 0 h-index: 0Robichaud, Albert论文数: 0 引用数: 0 h-index: 0Marquis, Karen论文数: 0 引用数: 0 h-index: 0Comery, Thomas论文数: 0 引用数: 0 h-index: 0Dunlop, John论文数: 0 引用数: 0 h-index: 0Pangalos, Menelas论文数: 0 引用数: 0 h-index: 0Brandon, Nicholas论文数: 0 引用数: 0 h-index: 0
- [9] PDE10A Inhibitors: Novel Therapeutic Drugs for SchizophreniaCURRENT PHARMACEUTICAL DESIGN, 2011, 17 (02) : 137 - 150Kehler, Jan论文数: 0 引用数: 0 h-index: 0机构: H Lundbeck & Co AS, Dept Biomol Chem, DK-2500 Valby, Denmark DMPK, DK-2500 Valby, Denmark H Lundbeck & Co AS, Dept Biomol Chem, DK-2500 Valby, DenmarkNielsen, Jacob论文数: 0 引用数: 0 h-index: 0机构: H Lundbeck & Co AS, Dept Synapt Transmiss 2, DK-2500 Valby, Denmark H Lundbeck & Co AS, Dept Biomol Chem, DK-2500 Valby, Denmark
- [10] Novel potent and selective PDE10A inhibitors show activity in animal models of psychosis and anxietySCHIZOPHRENIA BULLETIN, 2007, 33 (02) : 479 - 479Siuciak, J. A.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAChapin, D. S.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAMcCarthy, S. A.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAMartin, A. N.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAHarms, J. F.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAFox, C. B.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAChappie, T. A.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAHumphrey, J. M.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAProulx, C. A.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USAVerhoest, P. R.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USASchmidt, C. J.论文数: 0 引用数: 0 h-index: 0机构: CNS Discovery, Groton, CT USA CNS Discovery, Groton, CT USA