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- [1] Phase II multicenter proof of concept study of AZD4547 in FGFR amplified tumours.JOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (15)Smyth, Elizabeth Catherine论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandTurner, Nicholas C.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandPeckitt, Clare论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandPearson, Alex论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandBrown, Gina论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandChua, Sue论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandGillbanks, Angela论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandJohnston, Stephen R. D.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandTarazona, Noelia论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandCutts, Ros论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandKilgour, Elaine论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandRooney, Claire论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandSmith, Neil R.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandSumpter, Katherine Anne论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandAjaz, Mazhar A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandThomas, Anne L.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandWatkins, David论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandChau, Ian论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandPopat, Sanjay论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandCunningham, David论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, England
- [2] FGFR2 Gene Amplification in Gastric Cancer Predicts Sensitivity to the Selective FGFR Inhibitor AZD4547CLINICAL CANCER RESEARCH, 2013, 19 (09) : 2572 - 2583Xie, Liang论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaSu, Xinying论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaZhang, Lin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaYin, Xiaolu论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaTang, Lili论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaZhang, Xiuhua论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaXu, Yanping论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaGao, Zeren论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaLiu, Kunji论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaZhou, Minhua论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaGao, Beirong论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaShen, Danping论文数: 0 引用数: 0 h-index: 0机构: Shanghai Jiao Tong Univ, Sch Med, Renji Hosp, Shanghai 200030, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaZhang, Lianhai论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Surg, Key Lab Carcinogenesis & Translat Res, Beijing Inst Canc Res,Canc Hosp,Minist Educ, Beijing 100871, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaJi, Jiafu论文数: 0 引用数: 0 h-index: 0机构: Peking Univ, Dept Surg, Key Lab Carcinogenesis & Translat Res, Beijing Inst Canc Res,Canc Hosp,Minist Educ, Beijing 100871, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaGavine, Paul R.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaZhang, Jingchuan论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaKilgour, Elaine论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca Oncol, Macclesfield, Cheshire, England AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaZhang, Xiaolin论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R ChinaJi, Qunsheng论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China AstraZeneca R&D, Innovat Ctr China, Shanghai, Peoples R China
- [3] Structural Insights into FGFR Kinase Isoform Selectivity: Diverse Binding Modes of AZD4547 and Ponatinib in Complex with FGFR1 and FGFR4STRUCTURE, 2014, 22 (12) : 1764 - 1774Tucker, Julie A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, EnglandKlein, Tobias论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, EnglandBreed, Jason论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, EnglandBreeze, Alexander L.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, EnglandOverman, Ross论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, EnglandPhillips, Chris论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, EnglandNorman, Richard A.论文数: 0 引用数: 0 h-index: 0机构: AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England AstraZeneca, Discovery Sci, Macclesfield SK10 4TG, Cheshire, England
- [4] FGFR1 and FGFR2 in fibrolamellar carcinomaHISTOPATHOLOGY, 2016, 68 (05) : 686 - 692Graham, Rondell P.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USA Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USAGarcia, Joaquin J.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USA Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USAGreipp, Patricia T.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USA Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USAFritcher, Emily G. Barr论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USA Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USAKipp, Benjamin R.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USA Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USATorbenson, Michael S.论文数: 0 引用数: 0 h-index: 0机构: Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USA Mayo Clin, Dept Lab Med & Pathol, 200 First St SW, Rochester, MN 55905 USA
- [5] Inactivation of fgfr1 and fgfr2 in Postnatal AstrocytesINTEGRATIVE AND COMPARATIVE BIOLOGY, 2017, 57 : E392 - E392Rubin, L. B.论文数: 0 引用数: 0 h-index: 0机构: Univ Louisiana Lafayette, Lafayette, LA 70504 USA Univ Louisiana Lafayette, Lafayette, LA 70504 USASmith, K.论文数: 0 引用数: 0 h-index: 0机构: Univ Louisiana Lafayette, Lafayette, LA 70504 USA Univ Louisiana Lafayette, Lafayette, LA 70504 USA
- [6] FGFR1 and FGFR2 Mutations in Pfeiffer SyndromeJOURNAL OF CRANIOFACIAL SURGERY, 2013, 24 (01) : 150 - 152Chokdeemboon, Chayanin论文数: 0 引用数: 0 h-index: 0机构: Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, Thailand Chulalongkorn Univ, Ctr Excellence Med Genet, Dept Pediat, Fac Med, Bangkok 10330, Thailand Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, ThailandMahatumarat, Charan论文数: 0 引用数: 0 h-index: 0机构: King Chulalongkorn Mem Hosp, Dept Surg, Fac Med, Bangkok, Thailand Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, ThailandRojvachiranonda, Nond论文数: 0 引用数: 0 h-index: 0机构: King Chulalongkorn Mem Hosp, Dept Surg, Fac Med, Bangkok, Thailand Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, ThailandTongkobpetch, Siraprapa论文数: 0 引用数: 0 h-index: 0机构: Chulalongkorn Univ, Ctr Excellence Med Genet, Dept Pediat, Fac Med, Bangkok 10330, Thailand King Chulalongkorn Mem Hosp, Clin Excellence Ctr Med Genet, Bangkok, Thailand Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, ThailandSuphapeetiporn, Kanya论文数: 0 引用数: 0 h-index: 0机构: Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, Thailand Chulalongkorn Univ, Ctr Excellence Med Genet, Dept Pediat, Fac Med, Bangkok 10330, Thailand King Chulalongkorn Mem Hosp, Clin Excellence Ctr Med Genet, Bangkok, Thailand Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, ThailandShotelersuk, Vorasuk论文数: 0 引用数: 0 h-index: 0机构: Chulalongkorn Univ, Ctr Excellence Med Genet, Dept Pediat, Fac Med, Bangkok 10330, Thailand King Chulalongkorn Mem Hosp, Clin Excellence Ctr Med Genet, Bangkok, Thailand Chulalongkorn Univ, Fac Grad Sch, Interdept Biomed Sci, Bangkok 10330, Thailand
- [7] Mechanisms of Efficacy of the FGFR1–3 Inhibitor AZD4547 in Pediatric Solid Tumor ModelsInvestigational New Drugs, 2020, 38 : 1677 - 1686Nikki Phanhthilath论文数: 0 引用数: 0 h-index: 0机构: University of California San Diego,Department of Pediatrics, Division of HematologySara Hakim论文数: 0 引用数: 0 h-index: 0机构: University of California San Diego,Department of Pediatrics, Division of HematologyCatherine Su论文数: 0 引用数: 0 h-index: 0机构: University of California San Diego,Department of Pediatrics, Division of HematologyAndrea Liu论文数: 0 引用数: 0 h-index: 0机构: University of California San Diego,Department of Pediatrics, Division of HematologyDivya Subramonian论文数: 0 引用数: 0 h-index: 0机构: University of California San Diego,Department of Pediatrics, Division of HematologyJacqueline Lesperance论文数: 0 引用数: 0 h-index: 0机构: University of California San Diego,Department of Pediatrics, Division of HematologyPeter E. Zage论文数: 0 引用数: 0 h-index: 0机构: University of California San Diego,Department of Pediatrics, Division of Hematology
- [8] Phase II study of AZD4547 in FGFR amplified tumours: gastroesophageal cancer (GC) cohort clinical and translational resultsANNALS OF ONCOLOGY, 2015, 26 : 44 - 44Smyth, E. C.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandTurner, N.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Breast Oncol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandPearson, A.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res ICR, Inst Canc Res, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandPeckitt, C.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandChau, I.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandWatkins, D.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandKilgour, E.论文数: 0 引用数: 0 h-index: 0机构: Astra Zeneca, Innovat Med, Cheshire, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandSmith, N. R.论文数: 0 引用数: 0 h-index: 0机构: Astra Zeneca, Innovat Med, Cheshire, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandGillbanks, A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandChua, S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Nucl Med, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandBrown, G.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Radiol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandCutts, R.论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res ICR, Inst Canc Res, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandRooney, C.论文数: 0 引用数: 0 h-index: 0机构: Astra Zeneca, Innovat Med, Cheshire, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandLlavero, N. Tarazona论文数: 0 引用数: 0 h-index: 0机构: Inst Canc Res ICR, Inst Canc Res, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandThomas, A.论文数: 0 引用数: 0 h-index: 0机构: Leicester Royal Infirm, Univ Hosp Leicester NHS Trust, Gastrointestinal Oncol, Leicester, Leics, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandPopat, S.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Dept Med, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, EnglandCunningham, D.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, England Royal Marsden Hosp NHS Fdn Trust, Gastrointestinal Oncol, London, England
- [9] Phase II study of AZD4547 in FGFR amplified tumours: Gastroesophageal cancer (GC) cohort pharmacodynamic and biomarker results.JOURNAL OF CLINICAL ONCOLOGY, 2016, 34 (04)Smyth, Elizabeth Catherine论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandTurner, Nicholas C.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandPearson, Alex论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandPeckitt, Clare论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandChau, Ian论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandWatkins, David J.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandStarling, Naureen论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandRao, Sheela论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandGillbanks, Angela论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandKilgour, Elaine论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandSumpter, Katherine Anne论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandSmith, Neil R.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandCutts, Ros论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandRooney, Claire论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandThomas, Anne L.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandAjaz, Mazhar A.论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandChua, Sue论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandBrown, Gina论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandPopat, Sanjay论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, EnglandCunningham, David论文数: 0 引用数: 0 h-index: 0机构: Royal Marsden, London, England
- [10] The resistance mechanism of FGFR2 amplified gastric cancer cells against AZD4547, a fibroblast growth factor receptor inhibitorANNALS OF ONCOLOGY, 2016, 27Lee, S. Y.论文数: 0 引用数: 0 h-index: 0机构: Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South Korea Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South KoreaJeong, Y.论文数: 0 引用数: 0 h-index: 0机构: Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South Korea Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South KoreaNa, Y.论文数: 0 引用数: 0 h-index: 0机构: Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South Korea Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South KoreaKim, J. L.论文数: 0 引用数: 0 h-index: 0机构: Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South Korea Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South KoreaLee, D. H.论文数: 0 引用数: 0 h-index: 0机构: Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South Korea Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South KoreaOh, S. C.论文数: 0 引用数: 0 h-index: 0机构: Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South Korea Korea Univ, Guro Hosp, Oncol Hematol, Seoul, South Korea