Palladium-catalyzed synthesis of 5-and 5,7-substituted indole derivatives

被引：0

作者：

Yang, SC ^{[1
]}

Chung, WH ^{[1
]}

机构：

[1] Kaohsiung Med Univ, Grad Inst Pharmaceut Sci, Kaohsiung 80708, Taiwan

来源：

INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 1999年 / 38卷 / 08期

关键词：

D O I：

暂无

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

The reaction of IPy2BF4 with anilines give the corresponding 2-iodoanilines regioselectively in high yields. N-Allyl-2-iodoanilines undergo cyclization to give 5- and 5,7-substituted indole derivatives in the presence of palladium catalysts and bases. The procedure do not require protective groups on nitrogen.

引用

页码：897 / 904

页数：8

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