Palladium-catalyzed synthesis of 5-and 5,7-substituted indole derivatives

被引：0
|
作者：
Yang, SC [1 ]
Chung, WH [1 ]
机构：
[1] Kaohsiung Med Univ, Grad Inst Pharmaceut Sci, Kaohsiung 80708, Taiwan
来源：
INDIAN JOURNAL OF CHEMISTRY SECTION B-ORGANIC CHEMISTRY INCLUDING MEDICINAL CHEMISTRY | 1999年 / 38卷 / 08期
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中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
The reaction of IPy2BF4 with anilines give the corresponding 2-iodoanilines regioselectively in high yields. N-Allyl-2-iodoanilines undergo cyclization to give 5- and 5,7-substituted indole derivatives in the presence of palladium catalysts and bases. The procedure do not require protective groups on nitrogen.
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页码：897 / 904
页数：8
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