Solid-phase synthesis of peptoid-like oligomers containing diverse diketopiperazine units

被引：17
|
作者：
Suwal, Sujit [1 ]
Kodadek, Thomas [1 ]
机构：
[1] Scripps Res Inst, Dept Chem & Canc Biol, Jupiter, FL 33458 USA
来源：
ORGANIC & BIOMOLECULAR CHEMISTRY | 2014年 / 12卷 / 31期
关键词：
COMBINATORIAL LIBRARIES; 2,5-DIKETOPIPERAZINES;
D O I：
10.1039/c4ob00829d
中图分类号：
O62 [有机化学];
学科分类号：
070303 ; 081704 ;
摘要：
Diketopiperazine (DKP) units are found in many bioactive small molecules. Here we report facile chemistry for incorporating diverse DKP units within peptoid and peptoid-like libraries made by solid-phase split and pool synthesis.
引用
收藏
页码：5831 / 5834
页数：4
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