Solid-phase synthesis of peptoid-like oligomers containing diverse diketopiperazine units

被引：17

作者：

Suwal, Sujit ^{[1
]}

Kodadek, Thomas ^{[1
]}

机构：

[1] Scripps Res Inst, Dept Chem & Canc Biol, Jupiter, FL 33458 USA

来源：

ORGANIC & BIOMOLECULAR CHEMISTRY | 2014年 / 12卷 / 31期

关键词：

COMBINATORIAL LIBRARIES; 2,5-DIKETOPIPERAZINES;

D O I：

10.1039/c4ob00829d

中图分类号：

O62 [有机化学];

学科分类号：

070303 ; 081704 ;

摘要：

Diketopiperazine (DKP) units are found in many bioactive small molecules. Here we report facile chemistry for incorporating diverse DKP units within peptoid and peptoid-like libraries made by solid-phase split and pool synthesis.

引用

页码：5831 / 5834

页数：4

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