Synthesis and preclinical evaluation of two novel radioligands for PDE7 imaging in the brain

被引:0
|
作者
Thomae, David [1 ,2 ]
Servaes, Sijn [1 ]
Vazquez, Naiara [1 ,3 ]
Wyffels, Leonie [4 ]
Dedeurwaerdere, Stefanie [3 ]
Van der Veken, Pieter [2 ]
Joossens, Jurgen [2 ]
Augustyns, Koen [2 ]
Stroobants, Sigrid [1 ,4 ]
Staelens, Steven [1 ]
机构
[1] Univ Antwerp, Mol Imaging Ctr Antwerp, Antwerp, Belgium
[2] Univ Antwerp, Univ Antwerp Med Chem, Antwerp, Belgium
[3] Univ Antwerp, Dept Translat Neurosci, Antwerp, Belgium
[4] Univ Antwerp Hosp, Nucelar Med, Edegem, Belgium
关键词
D O I
暂无
中图分类号
Q5 [生物化学];
学科分类号
071010 ; 081704 ;
摘要
295
引用
收藏
页码:S295 / S295
页数:1
相关论文
共 50 条
  • [31] Synthesis and evaluation of novel radioligands for positron emission tomography imaging of central orexin-2 receptor
    Oi, Norihito
    Suzuki, Michiyuki
    Terauchi, Taro
    Tokunaga, Masaki
    Zhang, Ming-Rong
    Suhara, Tetsuya
    Higuchi, Makoto
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2014, 248
  • [32] Synthesis, in vitro and in vivo evaluation of novel radioligands for asynuclein PET
    Korat, Spela
    Pereira, Pedro
    Saw, Ran Sing
    Herfert, Kristina
    Beaino, Wissam
    Bang-Andersen, Benny
    de Esch, Iwan
    Vugts, Danielle
    Windhorst, Albert
    NUCLEAR MEDICINE AND BIOLOGY, 2023, 126 : S130 - S131
  • [33] SYNTHESIS AND EVALUATION OF TWO CANDIDATE 11C-LABELED RADIOLIGANDS FOR BRAIN PERIPHERAL BENZODIAZEPINE RECEPTORS
    Briard, E.
    Hong, J.
    Musachio, J. L.
    Zoghbi, S. S.
    Fujita, M.
    Imaizumi, M.
    Cropley, V.
    Innis, R. B.
    Pike, V. W.
    JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS, 2005, 48 : S71 - S71
  • [34] Synthesis and preclinical evaluation of [11C]MTP38 as a novel PET ligand for phosphodiesterase 7 in the brain
    Naoyuki Obokata
    Chie Seki
    Takeshi Hirata
    Jun Maeda
    Hideki Ishii
    Yuji Nagai
    Takehiko Matsumura
    Misae Takakuwa
    Hajime Fukuda
    Takafumi Minamimoto
    Kazunori Kawamura
    Ming-Rong Zhang
    Tatsuo Nakajima
    Takeaki Saijo
    Makoto Higuchi
    European Journal of Nuclear Medicine and Molecular Imaging, 2021, 48 : 3101 - 3112
  • [35] Synthesis and preclinical evaluation of [11C]MTP38 as a novel PET ligand for phosphodiesterase 7 in the brain
    Obokata, Naoyuki
    Seki, Chie
    Hirata, Takeshi
    Maeda, Jun
    Ishii, Hideki
    Nagai, Yuji
    Matsumura, Takehiko
    Takakuwa, Misae
    Fukuda, Hajime
    Minamimoto, Takafumi
    Kawamura, Kazunori
    Zhang, Ming-Rong
    Nakajima, Tatsuo
    Saijo, Takeaki
    Higuchi, Makoto
    EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2021, 48 (10) : 3101 - 3112
  • [36] Longitudinal evaluation of a preclinical model of Huntington disease using molecular imaging techniques and selected radioligands
    Moresco, Rosa Maria
    Belloli, S.
    Todde, S.
    Matarrese, M.
    Carpinelli, A.
    Turolla, E.
    Popoli, P.
    Pezzola, A.
    Carpinelli, A.
    Lecchi, M.
    Simonelli, P.
    Fazio, F.
    NEUROIMAGE, 2006, 31 : T34 - T34
  • [37] Synthesis and In Vitro Evaluation of Oxindole Derivatives as Potential Radioligands for 5-HT7 Receptor Imaging with PET
    Herth, Matthias M.
    Volk, Balazs
    Pallagi, Katalin
    Bech, Lasse Kofoed
    Antoni, Ferenc A.
    Knudsen, Gitte M.
    Kristensen, Jesper
    ACS CHEMICAL NEUROSCIENCE, 2012, 3 (12): : 1002 - 1007
  • [38] Synthesis and Evaluation of Radioligands for Imaging Brain Nociceptin/Orphanin FQ Peptide (NOP) Receptors with Positron Emission Tomography
    Pike, Victor W.
    Rash, Karen S.
    Chen, Zhaogen
    Pedregal, Concepcion
    Statnick, Michael A.
    Kimura, Yasuyuki
    Hong, Jinsoo
    Zoghbi, Sami S.
    Fujita, Masahiro
    Toledo, Miguel A.
    Diaz, Nuria
    Gackenheimer, Susan L.
    Tauscher, Johannes T.
    Barth, Vanessa N.
    Innis, Robert B.
    JOURNAL OF MEDICINAL CHEMISTRY, 2011, 54 (08) : 2687 - 2700
  • [39] Radionuclide labeling and evaluation of candidate radioligands for PET imaging of histone deacetylase in the brain
    Seo, Young Jun
    Muench, Lisa
    Reid, Alicia
    Chen, Jinzhu
    Kang, Yeona
    Hooker, Jacob M.
    Volkow, Nora D.
    Fowler, Joanna S.
    Kim, Sung Won
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2013, 23 (24) : 6700 - 6705
  • [40] Synthesis and Preclinical Evaluation of Fluorinated 5-Azaindoles as CB2 PET Radioligands
    Kallinen, Annukka
    Mardon, Karine
    Lane, Samuel
    Montgomery, Andrew P.
    Bhalla, Rajiv
    Stimson, Damion H. R.
    Ahamed, Muneer
    Cowin, Gary J.
    Hibbs, David
    Werry, Eryn L.
    Fulton, Roger
    Connor, Mark
    Kassiou, Michael
    ACS CHEMICAL NEUROSCIENCE, 2023, 14 (16): : 2902 - 2921