Synthesis and preclinical evaluation of two novel radioligands for PDE7 imaging in the brain

被引：0

作者：

Thomae, David ^{[1
,2
]}

Servaes, Sijn ^{[1
]}

Vazquez, Naiara ^{[1
,3
]}

Wyffels, Leonie ^{[4
]}

Dedeurwaerdere, Stefanie ^{[3
]}

Van der Veken, Pieter ^{[2
]}

Joossens, Jurgen ^{[2
]}

Augustyns, Koen ^{[2
]}

Stroobants, Sigrid ^{[1
,4
]}

Staelens, Steven ^{[1
]}

机构：

[1] Univ Antwerp, Mol Imaging Ctr Antwerp, Antwerp, Belgium

[2] Univ Antwerp, Univ Antwerp Med Chem, Antwerp, Belgium

[3] Univ Antwerp, Dept Translat Neurosci, Antwerp, Belgium

[4] Univ Antwerp Hosp, Nucelar Med, Edegem, Belgium

来源：

JOURNAL OF LABELLED COMPOUNDS & RADIOPHARMACEUTICALS | 2015年 / 58卷

关键词：

D O I：

暂无

中图分类号：

Q5 [生物化学];

学科分类号：

071010 ; 081704 ;

摘要：

295

引用

页码：S295 / S295

页数：1

共 50 条

[1] Synthesis and preclinical evaluation of a novel carbon-11 radiolabeled PDE7 ligand
Xiao, Zhiwei
Sun, Jiyun
Fujinaga, Masayuki
Zhao, Chunyu
Haider, Ahmed
Rong, Jian
Shao, Yihan
Xu, Ying
Lloyd, K. C. Kent
Wang, Lu
Zhang, Ming-Rong
Liang, Steven
JOURNAL OF NUCLEAR MEDICINE, 2022, 63
[2] Development of a novel PET ligand for imaging phosphodiesterase 7 (PDE7)
Rong, Jian
Zhao, Chunyu
Chaudhary, Ahmad
Yuan, Hongjie
Liang, Steven
JOURNAL OF NUCLEAR MEDICINE, 2024, 65
[3] Synthesis and preclinical evaluation of an 18F labeled PDE7 inhibitor for PET neuroimaging
Thomae, David
Servaes, Stijn
Vazquez, Naiara
Wyffels, Leonie
Dedeurwaerdere, Stefanie
Van der Veken, Pieter
Joossens, Jurgen
Augustyns, Koen
Stroobants, Sigrid
Staelens, Steven
NUCLEAR MEDICINE AND BIOLOGY, 2015, 42 (12) : 975 - 981
[4] Synthesis and preclinical evaluation of 18-Flabeled radioligands for imaging rhoassociated protein kinase 2 in the brain
Zheng, Chao
Mennie, William
Gravel, Paul
Balayeva, Tutukhanim
Chen, Baosheng
Holden, Daniel
Kapinos, Michael
Felchner, Zachary
Nicholson, LaShae
Toyonaga, Takuya
Zheng, MingQiang
Fowles, Krista
Ropchan, Jim
Nabulsi, Nabeel
Strittmatter, Stephen M.
Carson, Richard
Huang, Yiyun
Cai, Zhengxin Jason
JOURNAL OF NUCLEAR MEDICINE, 2023, 64
[5] Spiroquinazolinones as novel, potent, and selective PDE7 inhibitors. Part 1
Lorthiois, E
Bernardelli, P
Vergne, F
Oliveira, C
Mafroud, AK
Proust, E
Heuze, L
Moreau, F
Idrissi, M
Tertre, A
Bertin, B
Coupe, M
Wrigglesworth, R
Descours, A
Soulard, P
Berna, P
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2004, 14 (18) : 4623 - 4626
[6] Synthesis and evaluation of two novel 2-nitroimidazole derivatives as potential PET radioligands for tumor imaging
Zha, Zhihao
Zhu, Lin
Liu, Yajing
Du, Fenghua
Gan, Hongmei
Qiao, Jinping
Kung, Hank F.
NUCLEAR MEDICINE AND BIOLOGY, 2011, 38 (04) : 501 - 508
[7] Isothiazole and isoxazole fused pyrimidones as PDE7 inhibitors: SAR and pharmacokinetic evaluation
Banerjee, Abhisek
Yadav, Pravin S.
Bajpai, Malini
Sangana, Ramachandra Rao
Gullapalli, Srinivas
Gudi, Girish S.
Gharat, Laxmikant A.
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (09) : 3223 - 3228
[8] Synthesis and structure-activity relationships of guan analogues as phosphodiesterase 7 (PDE7) inhibitors
Barnes, MJ
Cooper, N
Davenport, RJ
Dyke, HJ
Galleway, FP
Galvin, FCA
Gowers, L
Haughan, AF
Lowe, C
Meissner, JWG
Montana, JG
Morgan, T
Picken, CL
Watson, RJ
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2001, 11 (08) : 1081 - 1083
[9] Synthesis and preclinical evaluation of serotonin 5-HT6 receptor radioligands for PET imaging
Becker, G.
Colomb, J.
Billard, T.
Zimmer, L.
EUROPEAN JOURNAL OF NUCLEAR MEDICINE AND MOLECULAR IMAGING, 2013, 40 : S198 - S198
[10] Synthesis and structure-activity relationship studies of dihydronaphthyridinediones as a novel structural class of potent and selective PDE7 inhibitors
Gewald, Rainer
Rueger, Carla
Grunwald, Christian
Egerland, Ute
Hoefgen, Norbert
BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2011, 21 (22) : 6652 - 6656

← 1 2 3 4 5 →