Diarylcyclohexanones: synthons for new bicyclic compounds

被引：1
|
作者：
Ahmad, Sarfraz [1 ]
Weis, Robert [1 ]
Faist, Johanna [1 ]
Wolkinger, Volker [1 ]
Saf, Robert [2 ]
Belaj, Ferdinand [3 ]
Brun, Reto [4 ]
Kaiser, Marcel [4 ]
Seebacher, Werner [1 ]
机构：
[1] Graz Univ, Inst Pharmaceut Sci, Graz, Austria
[2] Graz Univ Technol, ICTM, A-8010 Graz, Austria
[3] Graz Univ, Inst Chem, Graz, Austria
[4] Swiss Trop & Publ Hlth Inst, Basel, Switzerland
来源：
MONATSHEFTE FUR CHEMIE | 2012年 / 143卷 / 01期
关键词：
Cyclizations; Crystal structure; Drug research; Michael addition; Antiprotozoals; TRYPANOSOMA-BRUCEI-RHODESIENSE; ALPHA; BETA-UNSATURATED KETONES; GAMBIENSE; NONANES;
D O I：
10.1007/s00706-011-0679-z
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
We used 4-acetyl-3,5-diarylcyclohexanones bearing two different aromatic rings as synthons for the preparation of 6,7-diaryl-4-(dialkylamino)bicyclo[2.2.2]octanones, starting materials for new antiprotozoals.
引用
收藏
页码：145 / 152
页数：8
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