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- [21] Concurrent HER or PI3K Inhibition Potentiates the Antitumor Effect of the ERK Inhibitor Ulixertinib in Preclinical Pancreatic Cancer ModelsMOLECULAR CANCER THERAPEUTICS, 2018, 17 (10) : 2144 - 2155Jiang, Hongmei论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USAXu, Mai论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USALi, Lin论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA论文数: 引用数: h-index:机构:Dodhiawala, Paarth论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USAHighkin, Maureen论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USAZhang, Daoxiang论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USALi, Qiong论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Shanghai Jiao Tong Univ, Sch Med, Renji Hosp, Dept Lab Med, Shanghai, Peoples R China Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USAWang-Gillam, Andrea论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USALim, Kian-Huat论文数: 0 引用数: 0 h-index: 0机构: Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA Washington Univ, Sch Med, Dept Internal Med, Div Oncol, St Louis, MO 63110 USA
- [22] Amino-alkyl substituted fused imidazoles: potent, selective and orally bioavailable inhibitors of PI3KEJC SUPPLEMENTS, 2010, 8 (07): : 62 - 62Pastor, J.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainMartinez, S.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainAlvarez, R. M.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainVarela, C.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainHernandez, A. I.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainRodriguez, S.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainOyarzabal, J.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainAlbarran, M.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainLink, W.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, SpainBischoff, J. R.论文数: 0 引用数: 0 h-index: 0机构: Spanish Natl Canc Res Ctr, Madrid, Spain Spanish Natl Canc Res Ctr, Madrid, Spain
- [23] Optimization of Orally Bioavailable PI3Kδ Inhibitors and Identification of Vps34 as a Key Selectivity TargetJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (02) : 638 - 655Henley, Zoe A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandAmour, Augustin论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Refractory Resp Inflammat Discovery Performance U, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandBarton, Nick论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Data & Computat Sci Med Sci & Technol, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandBantscheff, Marcus论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Meyerhofstr 1, D-69117 Heidelberg, Germany GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandBergamini, Giovanna论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Meyerhofstr 1, D-69117 Heidelberg, Germany GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandBertrand, Sophie M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandConvery, Maire论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Prot Cellular & Struct Sci, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandDown, Kenneth论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandDuempelfeld, Birgit论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Meyerhofstr 1, D-69117 Heidelberg, Germany GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandEdwards, Chris D.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Drug Metab & Pharmacokinet, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandGrandi, Paola论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Meyerhofstr 1, D-69117 Heidelberg, Germany GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandGore, Paul M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandKeeling, Steve论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandLivia, Stefano论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandMallett, David论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Drug Metab & Pharmacokinet, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandMaxwell, Aoife论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandPrice, Mark论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Vitro Vivo Translat, David Jack Ctr, Pk Rd, Ware SG12 0DP, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandRau, Christina论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Meyerhofstr 1, D-69117 Heidelberg, Germany GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandReinhard, Friedrich B. M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Cellzome GmbH, Meyerhofstr 1, D-69117 Heidelberg, Germany GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandRowedder, James论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Screening Profiling & Mech Biol, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandRowland, Paul论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Prot Cellular & Struct Sci, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandTaylor, Jonathan A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandThomas, Daniel A.论文数: 0 引用数: 0 h-index: 0机构: Arctoris, 120E Olymp Ave,Milton Pk, Abingdon OX14 4SA, Oxon, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandHessel, Edith M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline R&D, Refractory Resp Inflammat Discovery Performance U, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, England GlaxoSmithKline R&D, Global Med Chem, Gunnels Wood Rd, Stevenage SG1 2NY, Herts, EnglandHamblin, J. 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