Pth15: An interfacial inhibitor of HIV-1 integrase that efficiently blocks HIV-1 replication

被引:0
|
作者
Gros, Edwige [1 ]
Guiot, Edwire [1 ]
Agopian, Audrey [1 ]
Deprez, Eric [2 ]
Mouscadet, Jean Francois [2 ]
Witvrouw, Myriam [3 ]
Divita, Gilles [1 ]
机构
[1] CNRS, CRBM, UMR 5237, F-34033 Montpellier, France
[2] CNRS, LBPA, UMR 8113, Cachan, France
[3] LMVD Univ Leuven, Louvain, Belgium
关键词
D O I
10.1016/j.antiviral.2008.01.044
中图分类号
R9 [药学];
学科分类号
1007 ;
摘要
30
引用
收藏
页码:A28 / A28
页数:1
相关论文
共 50 条
  • [21] Suppression of HIV replication using RNA interference against HIV-1 integrase
    Lau, Tat San
    Li, Yonggang
    Kameoka, Masanori
    Ng, Tzi Bun
    Wan, David Chi Cheong
    FEBS LETTERS, 2007, 581 (17) : 3253 - 3259
  • [22] Interfacial peptide inhibitors of HIV-1 integrase activity and dimerization
    Zhao, L
    Chmielewski, JA
    BIOPOLYMERS, 2003, 71 (03) : 397 - 397
  • [23] Interfacial peptide inhibitors of HIV-1 integrase activity and dimerization
    Zhao, L
    O'Reilly, MK
    Shultz, MD
    Chmielewski, J
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2003, 13 (06) : 1175 - 1177
  • [24] Peptide HIV-1 Integrase Inhibitors from HIV-1 Gene Products
    Suzuki, Shintaro
    Urano, Emiko
    Hashimoto, Chic
    Tsutsumi, Hiroshi
    Nakahara, Toru
    Tanaka, Tomohiro
    Nakanishi, Yuta
    Maddali, Kasthuraiah
    Han, Yan
    Hamatake, Makiko
    Miyauchi, Kosuke
    Pommie, Yves
    Beutler, John A.
    Sugiura, Wataru
    Fuji, Hideyoshi
    Hoshino, Tyuji
    Itotani, Kyoko
    Nomura, Wataru
    Narumi, Tetsuo
    Yamamoto, Naoki
    Komano, Jun A.
    Tamamura, Hirokazu
    JOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (14) : 5356 - 5360
  • [25] Development of an HIV-1 integrase genotyping assay for HIV-1 subtype AE
    Liu, Yang
    Margot, Nicolas
    Kitrinos, Kathryn M.
    Callebaut, Christian
    JOURNAL OF MEDICAL VIROLOGY, 2019, 91 (05) : 890 - 893
  • [26] Raltegravir: the first HIV-1 integrase strand transfer inhibitor in the HIV armamentarium
    Nguyen, Bach-Yen T.
    Isaacs, Robin D.
    Teppler, Hedy
    Leavitt, Randi Y.
    Sklar, Peter
    Iwamoto, Marian
    Wenning, Larissa A.
    Miller, Michael D.
    Chen, Joshua
    Kemp, Ramon
    Xu, Wei
    Fromtling, Robert A.
    Vacca, Joseph P.
    Young, Steven D.
    Rowley, Michael
    Lower, Michael W.
    Gottesdiener, Keith M.
    Hazuda, Daria J.
    PHARMACEUTICAL SCIENCE TO IMPROVE THE HUMAN CONDITION: WINNERS AND FINALIST CANDIDATES OF THE PRIX GALIEN USA, INTERNATIONAL, AND PRO BONO HUMANITARIAN AWARDS 2010, 2011, 1222 : 83 - 89
  • [27] Styrylquinoline derivatives:: A new class of potent HIV-1 integrase inhibitors that block HIV-1 replication in CEM cells
    Mekouar, K
    Mouscadet, JF
    Desmaële, D
    Subra, F
    Leh, H
    Savouré, D
    Auclair, C
    d'Angelo, J
    JOURNAL OF MEDICINAL CHEMISTRY, 1998, 41 (15) : 2846 - 2857
  • [28] HIV-1 inhibitor
    Lloyd, AW
    DRUG DISCOVERY TODAY, 1996, 1 (04) : 170 - 170
  • [29] The total synthesis of fukiic acid, an HIV-1 integrase inhibitor
    Queffelec, Clmence
    Bailly, Fabrice
    Mbemba, Gladys
    Mouscadet, Jean-Francois
    Debyser, Zeger
    Witvrouw, Myriarn
    Cotelle, Philippe
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2008, 43 (10) : 2268 - 2271
  • [30] Emerging patterns and implications of HIV-1 integrase inhibitor resistance
    Geretti, Anna Maria
    Armenia, Daniele
    Ceccherini-Silberstein, Francesca
    CURRENT OPINION IN INFECTIOUS DISEASES, 2012, 25 (06) : 677 - 686