共 50 条
- [31] Structure-Based Design of Potent and Selective Ligands at the Four Adenosine ReceptorsMOLECULES, 2017, 22 (11):Jespers, Willem论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, Sweden Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, SwedenOliveira, Ana论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, Sweden Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, SwedenPrieto-Diaz, Ruben论文数: 0 引用数: 0 h-index: 0机构: Univ Santiago Compostela, Fac Farm, Dept Quim Organ, Ctr Singular Invest Quim Biol & Mat Mol CIQUS, Santiago De Compostela 15782, Spain Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, SwedenMajellaro, Maria论文数: 0 引用数: 0 h-index: 0机构: Univ Santiago Compostela, Fac Farm, Dept Quim Organ, Ctr Singular Invest Quim Biol & Mat Mol CIQUS, Santiago De Compostela 15782, Spain Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, SwedenAqvist, Johan论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, Sweden Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, SwedenSotelo, Eddy论文数: 0 引用数: 0 h-index: 0机构: Univ Santiago Compostela, Fac Farm, Dept Quim Organ, Ctr Singular Invest Quim Biol & Mat Mol CIQUS, Santiago De Compostela 15782, Spain Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, SwedenGutierrez-de-Teran, Hugo论文数: 0 引用数: 0 h-index: 0机构: Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, Sweden Uppsala Univ, Dept Cell & Mol Biol, Biomed Ctr BMC, BOX 596, SE-75124 Uppsala, Sweden
- [32] Preclinical evaluation of AMG 925, a FLT3/CDK4 dual kinase inhibitor.MOLECULAR CANCER THERAPEUTICS, 2013, 12 (11)Dai, Kang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAKeegan, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USALi, Zhihong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAJi, Ma论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USALi, Gong论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAEksterowicz, John论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USASuzanne, Coberly论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAHollenback, David论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAWeidner, Margret论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAHuard, Justin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USALiang, Lingming论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAAlba, Grace论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAOrf, Jessica论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USALo, Mei-Chu论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAZhao, Sharon论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USANgo, Rachel论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAChen, Ada论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USALiu, Lily论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USACarlson, Timothy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAMcgee, Lawrence R.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAMedina, Julio论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAKamb, Alexander论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USAVlickramasinghe, Dineli论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA USA Amgen Inc, San Francisco, CA USA
- [33] Structure-based inhibitor designVITAMINS AND HORMONES - ADVANCES IN RESEARCH AND APPLICATIONS, VOL 58, 2000, 58 : 149 - +Craig, SP论文数: 0 引用数: 0 h-index: 0机构: Univ N Carolina, Sch Pharm, Lab Mol Parasitol & Drug Design, Chapel Hill, NC 27599 USA Univ N Carolina, Sch Pharm, Lab Mol Parasitol & Drug Design, Chapel Hill, NC 27599 USAEakin, AE论文数: 0 引用数: 0 h-index: 0机构: Univ N Carolina, Sch Pharm, Lab Mol Parasitol & Drug Design, Chapel Hill, NC 27599 USA Univ N Carolina, Sch Pharm, Lab Mol Parasitol & Drug Design, Chapel Hill, NC 27599 USA
- [34] Structure-Based Design of a Potent, Selective, and Brain Penetrating PDE2 Inhibitor with Demonstrated Target EngagementACS MEDICINAL CHEMISTRY LETTERS, 2014, 5 (09): : 1049 - 1053Buijnsters, Peter论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumDe Angelis, Meri论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumLanglois, Xavier论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumRombouts, Frederik J. R.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumSanderson, Wendy论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Discovery Sci, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumTresadern, Gary论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Discovery Sci, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumRitchie, Alison论文数: 0 引用数: 0 h-index: 0机构: BioFocus, Saffron Walden CB10 1XL, Essex, England Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumTrabanco, Andres A.论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumVanHoof, Greet论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Discovery Sci, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumVan Roosbroeck, Yves论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, Belgium Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, BelgiumAndres, Jose-Ignacio论文数: 0 引用数: 0 h-index: 0机构: Janssen Res & Dev, Neurosci Med Chem, Toledo 45007, Spain Janssen Res & Dev, Neurosci Med Chem, B-2340 Beerse, Belgium
- [35] Metamorphosis of paroxetine into a highly potent and selective GRK2 inhibitor via structure-based drug designABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2017, 253Waldschmidt, Helen论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USAHoman, Kristoff论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmacol, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Biol Chem, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USACruz-Rodriguez, Osvaldo论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmacol, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Biol Chem, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, PhD Program Chem Biol, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USACato, Marilyn论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmacol, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Biol Chem, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USABouley, Renee论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmacol, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Biol Chem, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USAWilson, Michael论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USACannavo, Alessandro论文数: 0 引用数: 0 h-index: 0机构: Temple Univ, Ctr Translat Med, Philadelphia, PA 19122 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USASong, Jianliang论文数: 0 引用数: 0 h-index: 0机构: Temple Univ, Ctr Translat Med, Philadelphia, PA 19122 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USACheung, Joseph论文数: 0 引用数: 0 h-index: 0机构: Temple Univ, Ctr Translat Med, Philadelphia, PA 19122 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USAKirchhoff, Paul论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USA论文数: 引用数: h-index:机构:Tesmer, John论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Pharmacol, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Biol Chem, Inst Life Sci, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USALarsen, Scott论文数: 0 引用数: 0 h-index: 0机构: Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USA Univ Michigan, Dept Med Chem, Vahlteich Med Chem Core, Ann Arbor, MI 48109 USA
- [36] Structure-based library design and the discovery of a potent and selective mast cell β-tryptase inhibitor as an oral therapeutic agentBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (02) : 1049 - 1054Liang, Guyan论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAAldous, Suzanne论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAMerriman, Gregory论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USALevell, Julian论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAPribish, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USACairns, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAChen, Xin论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAMaignan, Sebastien论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAMathieu, Magali论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USATsay, Joseph论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USASides, Keith论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USARebello, Sam论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAWhitely, Brian论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAMorize, Isabelle论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USAPauls, Henry W.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, New York, NY 10154 USA Bristol Myers Squibb Co, New York, NY 10154 USA
- [37] Structure-Based Design of a Potent and Selective Covalent Inhibitor for SRC Kinase That Targets a P-Loop CysteineJOURNAL OF MEDICINAL CHEMISTRY, 2020, 63 (04) : 1624 - 1641Du, Guangyan论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USARao, Suman论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAGurbani, Deepak论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAHenning, Nathaniel J.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAJiang, Jie论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAChe, Jianwei论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAYang, Annan论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAFicarro, Scott B.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAMarto, Jarrod A.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAAguirre, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Med Oncol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USASorger, Peter K.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Lab Syst Biol, Boston, MA 02115 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAWestover, Kenneth D.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAZhang, Tinghu论文数: 0 引用数: 0 h-index: 0机构: Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA Univ Texas Southwestern Med Ctr Dallas, Dept Radiat Oncol, Dallas, TX 75390 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02215 USA Univ Texas Southwestern Med Ctr Dallas, Dept Biochem, Dallas, TX 75390 USA
- [38] Cell death induction in resting lymphocytes by pan-Cdk inhibitor, but not by Cdk4/6 selective inhibitorINVESTIGATIONAL NEW DRUGS, 2011, 29 (05) : 921 - 931Kobayashi, Makiko论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, Japan Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, JapanTakahashi-Suzuki, Ikuko论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, Japan Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, JapanShimomura, Toshiyasu论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, Japan Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, JapanIwasawa, Yoshikazu论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Res Inst, Merck Res Labs, Dept Chem, Tsukuba, Ibaraki 3002611, Japan Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, JapanHirai, Hiroshi论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, Japan Banyu Tsukuba Res Inst, Merck Res Labs, Dept Oncol, Tsukuba, Ibaraki 3002611, Japan
- [39] Cell death induction in resting lymphocytes by pan-Cdk inhibitor, but not by Cdk4/6 selective inhibitorInvestigational New Drugs, 2011, 29 : 921 - 931Makiko Kobayashi论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Research Institute,Department of Oncology, Merck Research LaboratoriesIkuko Takahashi-Suzuki论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Research Institute,Department of Oncology, Merck Research LaboratoriesToshiyasu Shimomura论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Research Institute,Department of Oncology, Merck Research LaboratoriesYoshikazu Iwasawa论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Research Institute,Department of Oncology, Merck Research LaboratoriesHiroshi Hirai论文数: 0 引用数: 0 h-index: 0机构: Banyu Tsukuba Research Institute,Department of Oncology, Merck Research Laboratories
- [40] Discovery and structure-based design of 4,6-diaminonicotinamides as potent and selective IRAK4 inhibitorsBIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2017, 27 (21) : 4908 - 4913Bhide, Rajeev S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USAKeon, Alec论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USAWeigelt, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Mol Struct & Design, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USASack, John S.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Mol Struct & Design, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USASchmidt, Robert J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USALin, Shuqun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USAXiao, Hai-Yun论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USASpergel, Steven H.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USAKempson, James论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USAPitts, William J.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USACarman, Julie论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Immunosci Biol, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USAPoss, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA Bristol Myers Squibb Co, Discovery Chem, Res & Dev, Route 206 & Prov Line Rd, Princeton, NJ 08543 USA