Conformationally restricted tryptamine sulfonamides as novel and selective 5-HT6 receptor antagonists

被引:0
|
作者
Konda, Jagadishbabu [1 ]
Kambhampati, Rama Sastry [1 ]
Kothmirkar, Prabhakar [1 ]
Bandyala, Trinath Reddy [1 ]
Yarra, Sivasekhar N. K. [1 ]
Arepalli, Sobhanadri [1 ]
Rasheed, M. Abdul [1 ]
Shinde, Anil K. [1 ]
Nirogi, Ramakrishna
机构
[1] Suven Life Sci Ltd, Discovery Res Med Chem, Hyderabad 500034, Andhra Pradesh, India
来源
ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY | 2009年 / 237卷
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
104-MEDI
引用
收藏
页数:1
相关论文
共 50 条
  • [11] Amino aryl sulfonamides as novel and potent 5-ht6 receptor ligands
    Nirogi, Ramakrishna
    Kambhampati, Ramasastry
    Bandyala, Trinathreddy
    Konda, Jagadishbabu
    Arepalli, Sobhanadri
    Reballi, Veena
    Kothmirkar, Prabhakar
    Pamuleti, Narasimhareddy G.
    Shinde, Anil
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240
  • [12] Novel brain penetrant benzofuropiperidine 5-HT6 receptor antagonists
    Sundar, Babu G.
    Bailey, Thomas R.
    Dunn, Derek D.
    Bacon, Edward R.
    Salvino, Joseph M.
    Morton, George C.
    Aimone, Lisa D.
    Huang Zeqi
    Mathiasen, Joanne R.
    Dicamillo, Amy
    Huffman, Mark J.
    McKenna, Beth A.
    Kopec, Karla
    Lu, Lily D.
    Brown, Rebecca
    Qian, Jie
    Angeles, Thelma
    Connors, Thomas
    Spais, Chrysanthe
    Holskin, Beverly
    Galinis, Deborah
    Duzic, Emir
    Schaffhauser, Herve
    Rosse, Gerard C.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2012, 22 (01) : 120 - 123
  • [13] Conformationally constrained N1-arylsulfonyltryptamine derivatives as 5-HT6 receptor antagonists
    Cole, DC
    Lennox, WJ
    Stock, JR
    Ellingboe, JW
    Mazandarani, H
    Smith, DL
    Zhang, GM
    Tawa, GJ
    Schechter, LE
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (21) : 4780 - 4785
  • [14] New aryl sulfonamides compounds as potent and selective 5-ht6 receptor ligands
    Shinde, Anil
    Reballi, Veena
    Tiriveedhi, Vinay
    Gudla, Parandhama
    Kota, Laxman
    Chindhe, Anil
    Rambabu, Namala
    Kambhampati, Ramasastry
    Nirogi, Ramakrishna
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240
  • [15] Selective 5-HT6 antagonists for cognitive disorders
    Langston, S
    DRUG DISCOVERY TODAY, 2001, 6 (09) : 489 - 489
  • [16] Synthesis and structure-activity relationship of novel conformationally restricted analogues of serotonin as 5-HT6 receptor ligands
    Nirogi, Ramakrishna V. S.
    Kambhampati, Ramasastri
    Kothmirkar, Prabhakar
    Konda, Jagadishbabu
    Bandyala, Thrinath Reddy
    Gudla, Parandhama
    Arepalli, Sobhanadri
    Gangadasari, Narasimhareddy P.
    Shinde, Anil K.
    Deshpande, Amol D.
    Dwarampudi, Adireddy
    Chindhe, Anil K.
    Dubey, Pramod Kumar
    JOURNAL OF ENZYME INHIBITION AND MEDICINAL CHEMISTRY, 2012, 27 (03) : 443 - 450
  • [17] Bicyclic heteroarylpiperazines as selective brain penetrant 5-HT6 receptor antagonists
    Ahmed, M
    Briggs, MA
    Bromidge, SM
    Buck, T
    Campbell, L
    Deeks, NJ
    Garner, A
    Gordon, L
    Hamprecht, DW
    Holland, V
    Johnson, CN
    Medhurst, AD
    Mitchell, DJ
    Moss, SF
    Powles, J
    Seal, JT
    Stean, TO
    Stemp, G
    Thompson, M
    Trail, B
    Upton, N
    Winborn, K
    Witty, DR
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2005, 15 (21) : 4867 - 4871
  • [18] MEDI 40-Tetrahydro carbazoles: Novel, potent and selective 5-HT6 receptor antagonists
    Kambhampati, Rama Sastry
    Konda, Jagadish B.
    Kothmirkar, Prabhakar
    Bandyala, Trinath R.
    Yarra, Sivasekhar N. K.
    Arepalli, Sobhanadri
    Shinde, Anil K.
    Nirogi, Ramakrishna V. S.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2007, 234
  • [19] IDENTIFICATION OF NOVEL INDANYLAMIDINOHYDRAZONES AS 5-HT6 ANTAGONISTS
    Mesquida, Neus
    Lopez-Perez, Sara
    Dinares, Immaculada
    Frigola, Jordi
    Merce, Ramon
    Holenz, Joerg
    Perez, Raquel
    Burgueno, Javier
    Alcalde, Ermitas
    DRUGS OF THE FUTURE, 2009, 34 : 126 - 126
  • [20] Tetrahydrocarbazole derivatives as novel and selective 5-HT6 receptor ligands
    Konda, Jagadishbabu
    Kambhampati, Ramasastry
    Kothmirkar, Prabhakar
    Arepalli, Sobhanadri
    Bandyala, Trinath Reddy
    Gudla, Parandhama
    Shinde, Anil K.
    Nirogi, Ramakrishna
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238