Use of fret based technology to identify allosteric modulators for GPCRS: Application to metabotropic glutamate receptors

被引：0
|
作者：
Hubert, N [1 ]
Franchet, C [1 ]
Neuville, P [1 ]
机构：
[1] Faust Pharmaceut, Illkirch Graffenstaden, France
来源：
NEUROPHARMACOLOGY | 2005年 / 49卷
关键词：
D O I：
暂无
中图分类号：
Q189 [神经科学];
学科分类号：
071006 ;
摘要：
61
引用
收藏
页码：250 / 250
页数：1
相关论文
共 50 条
  • [21] Enlightening allosteric properties of metabotropic glutamate receptors
    Pin, J. -P.
    EUROPEAN BIOPHYSICS JOURNAL WITH BIOPHYSICS LETTERS, 2013, 42 : S159 - S159
  • [22] Selective Actions of Novel Allosteric Modulators Reveal Functional Heteromers of Metabotropic Glutamate Receptors in the CNS
    Yin, Shen
    Noetzel, Meredith J.
    Johnson, Kari A.
    Zamorano, Rocio
    Jalan-Sakrikar, Nidhi
    Gregory, Karen J.
    Conn, P. Jeffrey
    Niswender, Colleen M.
    JOURNAL OF NEUROSCIENCE, 2014, 34 (01): : 79 - 94
  • [23] Control of autoimmune inflammation using liposomes to deliver positive allosteric modulators of metabotropic glutamate receptors
    Gammon, Joshua M.
    Adapa, Arjun R.
    Jewell, Christopher M.
    JOURNAL OF BIOMEDICAL MATERIALS RESEARCH PART A, 2017, 105 (11) : 2977 - 2985
  • [24] Fragment-Based Approaches for Allosteric Metabotropic Glutamate Receptor (mGluR) Modulators
    Orgovan, Zoltan
    Ferenczy, Gyorgy G.
    Keseru, Gyorgy M.
    CURRENT TOPICS IN MEDICINAL CHEMISTRY, 2019, 19 (19) : 1768 - 1781
  • [25] Allosteric Modulators of Metabotropic Glutamate Receptor 5 for Treatment of Schizophrenia
    Conn, P. J.
    Stauffer, S. R.
    Zhou, S.
    Manka, J.
    Williams, R.
    Noetzel, M. J.
    Gregory, K. J.
    Vinson, P.
    Niswender, C. M.
    Jones, C. K.
    Steckler, T.
    MacDonald, G.
    Lindsley, C. W.
    CURRENT NEUROPHARMACOLOGY, 2011, 9 : 11 - 12
  • [26] Design and synthesis of novel metabotropic glutamate receptor allosteric modulators
    Stankiewicz, Anna
    Bugno, Ryszard
    Branski, Piotr
    Bojarski, Andrzej J.
    PHARMACOLOGICAL REPORTS, 2012, 64 (02) : 473 - 474
  • [27] Conformational fingerprinting of allosteric modulators in metabotropic glutamate receptor 2
    Liauw, Brandon Wey-Hung
    Foroutan, Arash
    Schamber, Michael R.
    Lu, Weifeng
    Afsari, Hamid Samareh
    Vafabakhsh, Reza
    ELIFE, 2022, 11
  • [28] Design and synthesis of novel metabotropic glutamate receptor allosteric modulators
    Anna Stankiewicz
    Ryszard Bugno
    Piotr Brański
    Andrzej J. Bojarski
    Pharmacological Reports, 2012, 64 : 473 - 474
  • [29] Allosteric modulation of metabotropic glutamate receptors by chloride ions
    Tora, Amelie S.
    Rovira, Xavier
    Dione, Ibrahima
    Bertrand, Hugues-Olivier
    Brabet, Isabelle
    De Koninck, Yves
    Doyon, Nicolas
    Pin, Jean-Philippe
    Acher, Francine
    Goudet, Cyril
    FASEB JOURNAL, 2015, 29 (10): : 4174 - 4188
  • [30] New insights into the activation mechanism of metabotropic glutamate receptors:: What we learned from the allosteric modulators
    Pin, JP
    Goudet, C
    Hlavackova, V
    Kniazeff, J
    Maurel, D
    Prézeau, L
    Blahos, J
    NEUROPHARMACOLOGY, 2005, 49 : 265 - 265
12345