Discovery of novel and orally active inhibitors of lck kinase.

被引:0
|
作者
Goldberg, D [1 ]
Butz, T [1 ]
Cardozo, M [1 ]
Eckner, R [1 ]
Hammach, A [1 ]
Huang, J [1 ]
Jakes, S [1 ]
Kapadia, S [1 ]
Lukas, S [1 ]
Morwick, T [1 ]
Moss, N [1 ]
Panzenbeck, M [1 ]
Patel, U [1 ]
Peet, G [1 ]
Peterson, J [1 ]
Prokopowicz, A [1 ]
Snow, RJ [1 ]
Takahashi, H [1 ]
Tan, J [1 ]
Tschantz, M [1 ]
Wang, XJ [1 ]
Xiang, P [1 ]
Zinter, R [1 ]
机构
[1] Boehringer Ingelheim Pharmaceut Inc, Ridgefield, CT 06877 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
24-MEDI
引用
收藏
页码:U643 / U643
页数:1
相关论文
共 50 条
  • [31] Discovery of a Novel Class of Orally Active Antifungal β-1,3-D-Glucan Synthase Inhibitors
    Walker, Scott S.
    Xu, Yiming
    Triantafyllou, Ilias
    Waldman, Michelle F.
    Mendrick, Cara
    Brown, Nathaniel
    Mann, Paul
    Chau, Andrew
    Patel, Reena
    Bauman, Nicholas
    Norris, Christine
    Antonacci, Barry
    Gurnani, Maya
    Cacciapuoti, Anthony
    McNicholas, Paul M.
    Wainhaus, Samuel
    Herr, R. Jason
    Kuang, Rongze
    Aslanian, Robert G.
    Ting, Pauline C.
    Black, Todd A.
    ANTIMICROBIAL AGENTS AND CHEMOTHERAPY, 2011, 55 (11) : 5099 - 5106
  • [32] Discovery of Novel Benzoxazinones as Potent and Orally Active Long Chain Fatty Acid Elongase 6 Inhibitors
    Mizutani, Takashi
    Ishikawa, Shiho
    Nagase, Tsuyoshi
    Takahashi, Hidekazu
    Fujimura, Takashi
    Sasaki, Takahide
    Nagumo, Akira
    Shimamura, Ken
    Miyamoto, Yasuhisa
    Kitazawa, Hidefumi
    Kanesaka, Maki
    Yoshimoto, Ryo
    Aragane, Katsumi
    Tokita, Shigeru
    Sato, Nagaaki
    JOURNAL OF MEDICINAL CHEMISTRY, 2009, 52 (22) : 7289 - 7300
  • [33] Discovery of orally active selective inhibitors of Plk1[p]
    Pinder, Joanne L.
    Durrant, Steven
    Everitt, Simon
    Mortimore, Michael
    Keily, Shazia
    Knegtel, Ronald
    O'Donnell, Michael
    Brenchley, Guy
    Charrier, Jean-Damien
    Golec, Julian
    Kay, David
    Mak, Chau
    Ramaya, Sharn
    Rutherford, Alistair
    Studley, John
    Virani, Anisa
    Weber, Peter
    Young, Stephen C.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243
  • [34] Discovery of Orally Active Hydroxyethylamine Based SPPL2a Inhibitors
    Velcicky, Juraj
    Mathison, Casey J. N.
    Nikulin, Victor
    Pflieger, Daniel
    Epple, Robert
    Azimioara, Mihai
    Cow, Christopher
    Michellys, Pierre-Yves
    Rigollier, Pascal
    Beisner, Daniel R.
    Bodendorf, Ursula
    Guerini, Danilo
    Liu, Bo
    Wen, Ben
    Zaharevitz, Samantha
    Brandl, Trixi
    ACS MEDICINAL CHEMISTRY LETTERS, 2019, 10 (06): : 887 - 892
  • [35] Discovery of orally active butyrolactam 11β-HSD1 inhibitors
    Yeh, Vince S. C.
    Kurukulasuriya, Ravi
    Fung, Steven
    Monzon, Katina
    Chiou, William
    Wang, Jiahong
    Stolarik, Deanne
    Imade, Hovis
    Shapiro, Robin
    Knourek-Segel, Victoria
    Bush, Eugene
    Wilcox, Denise
    Nguyen, Phong T.
    Brune, Michael
    Jacobson, Peer
    Link, J. T.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2006, 16 (21) : 5555 - 5560
  • [36] Discovery of new orally active phosphodiesterase (PDE4) inhibitors
    Ochiai, H
    Ishida, A
    Ohtani, T
    Kusumi, K
    Kishikawa, K
    Yamamoto, S
    Takeda, H
    Obata, T
    Nakai, H
    Toda, M
    CHEMICAL & PHARMACEUTICAL BULLETIN, 2004, 52 (09) : 1098 - 1104
  • [37] Discovery of potent and orally active tricyclic-based FBPase inhibitors
    Tsukada, Tomoharu
    Kanno, Osamu
    Yamane, Takahiro
    Tanaka, Jun
    Yoshida, Taishi
    Okuno, Akira
    Shiiki, Takeshi
    Takahashi, Mizuki
    Nishi, Takahide
    BIOORGANIC & MEDICINAL CHEMISTRY, 2010, 18 (14) : 5346 - 5351
  • [38] Discovery of sulfonylalkylamides: A new class of orally active factor Xa inhibitors
    Imaeda, Yasuhiro
    Miyawaki, Toshio
    Sakamoto, Hiroki
    Itoh, Fumio
    Konishi, Noriko
    Hiroe, Katsuhiko
    Kawamura, Masaki
    Tanaka, Toshimasa
    Kubo, Keiji
    BIOORGANIC & MEDICINAL CHEMISTRY, 2008, 16 (05) : 2243 - 2260
  • [39] Discovery of novel sphingosine kinase 1 inhibitors
    Xiang, Yibin
    Asmussen, Gary
    Booker, Michael
    Hirth, Bradford
    Kane, John L., Jr.
    Liao, Junkai
    Noson, Kevin D.
    Yee, Christopher
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (21) : 6119 - 6121
  • [40] Discovery of novel TAM family kinase inhibitors
    Zhang, Zaihui
    Li, Rick
    Lee, Erica
    Hu, Yuxiang
    Yan, Jun
    Sanghera, Jasbinder
    CANCER RESEARCH, 2014, 74 (19)