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- [1] Discovery of a small molecule SIRT1 activator for the treatment of prostate cancerABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Kong, Yali论文数: 0 引用数: 0 h-index: 0机构: Georgetown Univ, Med Ctr, Drug Discovery Program, Washington, DC 20057 USA Georgetown Univ, Med Ctr, Drug Discovery Program, Washington, DC 20057 USAZhang, Li论文数: 0 引用数: 0 h-index: 0机构: Georgetown Univ, Med Ctr, Drug Discovery Program, Washington, DC 20057 USAPreet, Anju论文数: 0 引用数: 0 h-index: 0机构: Georgetown Univ, Med Ctr, Drug Discovery Program, Washington, DC 20057 USAAvantaggiati, Maria L.论文数: 0 引用数: 0 h-index: 0机构: Georgetown Univ, Med Ctr, Drug Discovery Program, Washington, DC 20057 USABrown, Milton L.论文数: 0 引用数: 0 h-index: 0机构: Georgetown Univ, Med Ctr, Drug Discovery Program, Washington, DC 20057 USA Georgetown Univ, Med Ctr, Drug Discovery Program, Washington, DC 20057 USA
- [2] Identification of a small molecule activator of SIRT1 gene expressionAGING-US, 2013, 5 (03): : 174 - 182Cho, Si-Young论文数: 0 引用数: 0 h-index: 0机构: Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South Korea Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South KoreaCho, Miook论文数: 0 引用数: 0 h-index: 0机构: Albert Einstein Coll Med, Dept Genet, Bronx, NY 10461 USA Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South KoreaSeo, Dae Bang论文数: 0 引用数: 0 h-index: 0机构: Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South Korea Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South KoreaLee, Sang Jun论文数: 0 引用数: 0 h-index: 0机构: Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South Korea Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South KoreaSuh, Yousin论文数: 0 引用数: 0 h-index: 0机构: Albert Einstein Coll Med, Dept Genet, Bronx, NY 10461 USA Albert Einstein Coll Med, Dept Med, Bronx, NY 10461 USA Guangdong Med Coll, Inst Aging Res, Dongguan, Peoples R China Amorepacific Corp, R&D Ctr, Gyeonggi Do 446729, South Korea
- [3] Crystallographic Structure of a Small Molecule SIRT1 Activator/Enzyme ComplexBIOPHYSICAL JOURNAL, 2014, 106 (02) : 646A - 646ADai, Han论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAZhao, Huizhen论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAJiang, Yong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USASweitzer, Sharon M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAPietrak, Beth论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USASchwartz, Benjamin论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAMiller, William论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAHu, Erding论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USAEllis, James L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA USA GlaxoSmithKline, Collegeville, PA USA
- [4] AROuSing SIRT1: Identification of a novel endogenous SIRT1 activatorMOLECULAR CELL, 2007, 28 (03) : 354 - 356Verdin, Eric论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Gladstone Inst Virol & Immunol, San Francisco, CA 94158 USA Univ Calif San Francisco, Gladstone Inst Virol & Immunol, San Francisco, CA 94158 USA
- [5] Crystallographic structure of a small molecule SIRT1 activator-enzyme complexNATURE COMMUNICATIONS, 2015, 6Dai, Han论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USACase, April W.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USARiera, Thomas V.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAConsidine, Thomas论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USALee, Jessica E.论文数: 0 引用数: 0 h-index: 0机构: ExSAR Corp, Monmouth Jct, NJ 08852 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAHamuro, Yoshitomo论文数: 0 引用数: 0 h-index: 0机构: ExSAR Corp, Monmouth Jct, NJ 08852 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAZhao, Huizhen论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAJiang, Yong论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USASweitzer, Sharon M.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAPietrak, Beth论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USASchwartz, Benjamin论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USABlum, Charles A.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USADisch, Jeremy S.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USACaldwell, Richard论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USASzczepankiewicz, Bruce论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAOalmann, Christopher论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USANg, Pui Yee论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAWhite, Brian H.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USACasaubon, Rebecca论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USANarayan, Radha论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAKoppetsch, Karsten论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USABourbonais, Francis论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAWu, Bo论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Hefei Inst Phys Sci, High Field Magnet Lab, Hefei 230031, Anhui, Peoples R China GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAWang, Junfeng论文数: 0 引用数: 0 h-index: 0机构: Chinese Acad Sci, Hefei Inst Phys Sci, High Field Magnet Lab, Hefei 230031, Anhui, Peoples R China GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAQian, Dongming论文数: 0 引用数: 0 h-index: 0机构: Viva Biotech, Shanghai 201203, Peoples R China GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAJiang, Fan论文数: 0 引用数: 0 h-index: 0机构: Viva Biotech, Shanghai 201203, Peoples R China GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAMao, Cheney论文数: 0 引用数: 0 h-index: 0机构: Viva Biotech, Shanghai 201203, Peoples R China GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAWang, Minghui论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAHu, Erding论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline, Collegeville, PA 19426 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAWu, Joe C.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAPerni, Robert B.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAVlasuk, George P.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USAEllis, James L.论文数: 0 引用数: 0 h-index: 0机构: GlaxoSmithKline Co, Sirtris, Cambridge, MA 02139 USA GlaxoSmithKline, 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- [9] Small molecule activators of SIRT1 as therapeutics for the treatment of type 2 diabetesNature, 2007, 450 : 712 - 716Jill C. Milne论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicinePhilip D. Lambert论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineSimon Schenk论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineDavid P. Carney论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineJesse J. Smith论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineDavid J. Gagne论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineLei Jin论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineOlivier Boss论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineRobert B. Perni论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineChi B. Vu论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineJean E. Bemis论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineRoger Xie论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineJeremy S. Disch论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicinePui Yee Ng论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineJoseph J. Nunes论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineAmy V. Lynch论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineHongying Yang论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineHeidi Galonek论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineKristine Israelian论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineWendy Choy论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineAndre Iffland论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineSiva Lavu论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineOliver Medvedik论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineDavid A. Sinclair论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineJerrold M. Olefsky论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineMichael R. Jirousek论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicinePeter J. Elliott论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of MedicineChristoph H. Westphal论文数: 0 引用数: 0 h-index: 0机构: Sirtris Pharmaceuticals Inc.,Division of Endocrinology and Metabolism, Department of Medicine
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