Synthesis, Characterization and Biological Evaluation of Thiazole Containing Chromones and Pyrazole Derivatives

被引:0
|
作者
Darekar, Nirmala R. [1 ,2 ]
Takate, Sushama J. [2 ]
Akolkar, Hemantkumar N. [4 ]
Salve, Supriya P. [2 ]
Karale, Bhausaheb K. [1 ]
Mhaske, Sadhana D. [2 ,3 ]
机构
[1] Radhabai Kale Mahila Mahavidyalaya, Dept Chem, Ahmednagar, Maharashtra, India
[2] New Arts Sci & Commerce Coll, Dept Chem, Ahmednagar, Maharashtra, India
[3] Dadapatil Rajale Arts Sci & Commerce Coll, Dept Chem, Ahmednagar, Maharashtra, India
[4] Abasaheb Marathe Arts & New Commerce, Dept Chem, Sci Coll, Rajapur, Maharashtra, India
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中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
A novel series of 2-(4-methylthiazol-5-yl)-4H-chromen-4-ones (5) and 2-(5-(4-methylthiazol-5-yl)-1Hpyrazol-3-yl)phenols (6) were synthesized by using 4-methylthiazole-5-carboxylic acid 1 and substituted 2-hydroxy acetophenone 2. All the synthesized compounds were characterized with the help of spectral techniques and screened for their antimicrobial activities.
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页码:433 / 438
页数:6
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