Isoform-Selective Targeting of Facilitative Glucose Transporters with Small Molecule Inhibitors

被引:0
|
作者
Heitmeier, Monique
Hresko, Richard C.
Shanmugam, Mala
Hruz, Paul W.
机构
关键词
D O I
10.2337/db18-1779-P
中图分类号
R5 [内科学];
学科分类号
1002 ; 100201 ;
摘要
引用
收藏
页数:2
相关论文
共 50 条
  • [41] ISOFORM-SPECIFIC SUBCELLULAR TARGETING OF GLUCOSE TRANSPORTERS IN MOUSE FIBROBLASTS
    HUDSON, AW
    RUIZ, ML
    BIRNBAUM, MJ
    JOURNAL OF CELL BIOLOGY, 1992, 116 (03): : 785 - 797
  • [42] Disturbance of peristalsis in the guinea-pig isolated small intestine by indomethacin, but not cyclo-oxygenase isoform-selective inhibitors
    Shahbazian, A
    Schuligoi, R
    Heinemann, A
    Peskar, BA
    Holzer, P
    BRITISH JOURNAL OF PHARMACOLOGY, 2001, 132 (06) : 1299 - 1309
  • [43] Synthesis and characterization of novel isoform-selective IP6K1 inhibitors
    Wormald, Michael M.
    Ernst, Glen
    Wei, Huijun
    Barrow, James C.
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2019, 29 (19)
  • [44] Isoform-selective targeting of PI3K: time to consider new opportunities?
    Cirillo, Davide
    Diceglie, Marta
    Nazare, Marc
    TRENDS IN PHARMACOLOGICAL SCIENCES, 2023, 44 (09) : 601 - 621
  • [45] Development of an ELISA-Based HDAC Activity Assay for Characterization of Isoform-Selective Inhibitors
    Padige, Geetha
    Negmeldin, Ahmed T.
    Pflum, Mary Kay H.
    JOURNAL OF BIOMOLECULAR SCREENING, 2015, 20 (10) : 1277 - 1285
  • [46] Small molecule inhibitors targeting the cancers
    Liu, Gui-Hong
    Chen, Tao
    Zhang, Xin
    Ma, Xue-Lei
    Shi, Hua-Shan
    MEDCOMM, 2022, 3 (04):
  • [47] 7-Substituted-sulfocoumarins are isoform-selective, potent carbonic anhydrase II inhibitors
    Tanc, Muhammet
    Carta, Fabrizio
    Bozdag, Murat
    Scozzafava, Andrea
    Supuran, Claudiu T.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2013, 21 (15) : 4502 - 4510
  • [48] Investigation of the binding of isoform-selective inhibitors to prostaglandin endoperoxide synthases using fluorescence spectroscopy
    Lanzo, CA
    Beechem, JM
    Talley, J
    Marnett, LJ
    BIOCHEMISTRY, 1998, 37 (01) : 217 - 226
  • [49] Design and Synthesis of Simplified Largazole Analogues as Isoform-Selective Human Lysine Deacetylase Inhibitors
    Reddy, Damodara N.
    Ballante, Flavio
    Chuang, Timothy
    Pirolli, Adele
    Marrocco, Biagina
    Marshall, Garland R.
    JOURNAL OF MEDICINAL CHEMISTRY, 2016, 59 (04) : 1613 - 1633
  • [50] Rational design and crystallographic analysis of novel isoform-selective TRKA inhibitors for cancer therapy
    Wang, Guan
    Wu, Yongya
    Wu, Chengyong
    Shuai, Wen
    Jiang, Tingting
    Wang, Aoxue
    Bu, Faqian
    Sun, Qiu
    Ouyang, Liang
    ACTA PHARMACEUTICA SINICA B, 2023, 13 (01) : 440 - 443