共 50 条
- [1] The development of a selective CDK7 inhibitor with anti-tumor activityCANCER RESEARCH, 2009, 69Coombes, Raoul论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandCheiper论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandJogalekar, Ashutosh S.论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandBrackow, Jan论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandAli, Simak论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandHeathcote, Dean论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandKroll, Sebastian论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandBodo, S.论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandSiwicka, Aleksandra论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandPeriyasamy, Manikandan论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandTolhurst, Robert论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandKanneganti, Seshu论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandSnyder, James论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandLiotta, Dennis论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandAboagye, Eric论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, EnglandBarrett, Anthony论文数: 0 引用数: 0 h-index: 0机构: Univ London Imperial Coll Sci Technol & Med, London, England
- [2] SY-5609, an orally available selective CDK7 inhibitor demonstrates broad anti-tumor activity in vivoCANCER RESEARCH, 2019, 79 (13)Hu, Shanhu论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMarineau, Jason论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAHamman, Kristin论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USABradley, Michael论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USASavinainen, Anneli论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAAlnemy, Sydney论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USARajagopal, Nisha论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAOrlando, David论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAChuaqui, Claudio论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAOlson, Eric论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USA
- [3] Q901; a highly selective covalent cdk7 inhibitor inducing substantial anti-tumor effect in a broad spectrum of solid tumor lineagesCANCER RESEARCH, 2022, 82 (12)Yu, Donghoon论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaJeon, Yeejin论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaLee, Seung-Joo论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaKim, Jaeseung论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South KoreaNam, Kiyean论文数: 0 引用数: 0 h-index: 0机构: Qurient Co Ltd, Seoul, South Korea Qurient Co Ltd, Seoul, South Korea
- [4] An oral and selective CDK12 inhibitor demonstrates robust anti-tumor activityCANCER RESEARCH, 2022, 82 (12)Hu, Shanhu论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMoebius, David论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USADworakowski, Wojciech论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USACooper, Elliott论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USALaPlaca, Derek论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAAlnemy, Sydney论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAPerera, Phone论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAMarineau, Jason论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAChuaqui, Claudio论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USACarulli, John P.论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USAOlson, Eric论文数: 0 引用数: 0 h-index: 0机构: Syros Pharmaceut, Cambridge, MA USA Syros Pharmaceut, Cambridge, MA USA
- [5] A selective, potent, and orally bioavailable CDK7 inhibitor demonstrates superior anti-cancer activity in colorectal cancer modelsCANCER RESEARCH, 2024, 84 (07)Park, Heuijoon论文数: 0 引用数: 0 h-index: 0Seo, Kyoungwan论文数: 0 引用数: 0 h-index: 0Yu, Jihyun论文数: 0 引用数: 0 h-index: 0Kim, Jieun论文数: 0 引用数: 0 h-index: 0Joo, Min Sung论文数: 0 引用数: 0 h-index: 0Kim, Sungeun论文数: 0 引用数: 0 h-index: 0Lee, Joonhyung论文数: 0 引用数: 0 h-index: 0Lee, Jeonghyeon论文数: 0 引用数: 0 h-index: 0Kim, Eun-Jung论文数: 0 引用数: 0 h-index: 0Nam, Joonwoo论文数: 0 引用数: 0 h-index: 0Han, Wooseok论文数: 0 引用数: 0 h-index: 0
- [6] Potent anti-tumor activity of AUR102, a selective covalent inhibitor of CDK7EUROPEAN JOURNAL OF CANCER, 2020, 138 : S47 - S47Satyam, L. K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaPoddutoori, R.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Med Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaThiyagarajan, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaMukherjee, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Computat Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaKaza, L. N.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaCharamanna, K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Toxicol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaMarappan, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Biochem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaSamiulla, D.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaTiwari, N. K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaDevaraja, T.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Med Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaAravind, A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Pharmacol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaDhudashiya, A. A.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaBooher, R.论文数: 0 引用数: 0 h-index: 0机构: Exelixis Inc, Alameda, CA USA Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaDaginakatte, G.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Pharmacol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaAntony, T.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Biochem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaChelur, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Toxicol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaNellore, K.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaGiri, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Drug Metab & Pharmacokinet, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaRamachandra, M.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, IndiaSamajdar, S.论文数: 0 引用数: 0 h-index: 0机构: Aurigene Discovery Technol Ltd, Med Chem, Bangalore, Karnataka, India Aurigene Discovery Technol Ltd, Cell & Mol Biol, Bangalore, Karnataka, India
- [7] Synergistic Anti-Tumor Effect of Combining Selective CDK7 and BRD4 Inhibition in NeuroblastomaFRONTIERS IN ONCOLOGY, 2022, 11Gao, Yang论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA Boston Childrens Hosp, Boston, MA 02115 USA Harvard Med Sch, Dept Pediat, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA论文数: 引用数: h-index:机构:Nasholm, Nicole论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Pediat, San Francisco, CA 94143 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USADas, Sanjukta论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA Boston Childrens Hosp, Boston, MA 02115 USA Harvard Med Sch, Dept Pediat, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAKwiatkowski, Nicholas论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAAbraham, Brian J.论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Dept Computat Biol, 332 N Lauderdale St, Memphis, TN 38105 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAZhang, Tinghu论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAGray, Nathanael S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Canc Biol, Boston, MA 02115 USA Harvard Med Sch, Dept Biol Chem & Mol Pharmacol, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USAGustafson, Clay论文数: 0 引用数: 0 h-index: 0机构: Univ Calif San Francisco, Helen Diller Family Comprehens Canc Ctr, Dept Pediat, San Francisco, CA 94143 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA论文数: 引用数: h-index:机构:George, Rani E.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA Boston Childrens Hosp, Boston, MA 02115 USA Harvard Med Sch, Dept Pediat, Boston, MA 02115 USA Dana Farber Canc Inst, Dept Pediat Hematol Oncol, Boston, MA 02115 USA
- [8] In vivo anti-tumor efficacy of UD-017, a novel highly selective & orally available CDK7 inhibitor, in colorectal cancer cells xenograft modelsCANCER RESEARCH, 2017, 77Aga, Yasuhiro论文数: 0 引用数: 0 h-index: 0Ogi, Sayaka论文数: 0 引用数: 0 h-index: 0Tokunaga, Yasunori论文数: 0 引用数: 0 h-index: 0Ogawa, Ayumi论文数: 0 引用数: 0 h-index: 0Onuma, Kazuhiro论文数: 0 引用数: 0 h-index: 0Matsushita, Takashi论文数: 0 引用数: 0 h-index: 0Sunamoto, Hidetoshi论文数: 0 引用数: 0 h-index: 0Hasegawa, Tom论文数: 0 引用数: 0 h-index: 0Ushiyama, Shigeru论文数: 0 引用数: 0 h-index: 0
- [9] ICEC0942, an orally bioavailable selective inhibitor of CDK7 for breast cancerBREAST CANCER RESEARCH AND TREATMENT, 2016, 159 (01) : 195 - 195Ali, Simak论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Surg & Canc, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandPatel, Hetal论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Surg & Canc, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandPeriyasamy, Manikandan论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Surg & Canc, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandBondke, Alexander论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Chem, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandSlafer, Brian W.论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Chem, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandOttaviani, Silvia论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Surg & Canc, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandHarrod, Alison论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Surg & Canc, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandBuluwela, Laki论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Surg & Canc, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandFuchter, Matthew J.论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Chem, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandBarrett, Anthony G. M.论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Chem, London, England Imperial Coll London, Dept Surg & Canc, London, EnglandCoombes, R. Charles论文数: 0 引用数: 0 h-index: 0机构: Imperial Coll London, Dept Surg & Canc, London, England Imperial Coll London, Dept Surg & Canc, London, England
- [10] SY-1365, a potent and selective CDK7 inhibitor, exhibits promising anti-tumor activity in multiple preclinical models of aggressive solid tumorsCANCER RESEARCH, 2017, 77Hu, Shanhu论文数: 0 引用数: 0 h-index: 0Ke, Nan论文数: 0 引用数: 0 h-index: 0Ren, Yixuan论文数: 0 引用数: 0 h-index: 0Miljovska, Sofija论文数: 0 引用数: 0 h-index: 0Rajagopal, Nisha论文数: 0 引用数: 0 h-index: 0McKeown, Michael论文数: 0 引用数: 0 h-index: 0Orlando, David论文数: 0 引用数: 0 h-index: 0Sprott, Kevin论文数: 0 引用数: 0 h-index: 0Choi, Yoon J.论文数: 0 引用数: 0 h-index: 0Olson, Eric论文数: 0 引用数: 0 h-index: 0Fritz, Christian C.论文数: 0 引用数: 0 h-index: 0