A facile and chemoselective synthesis of 1,4-benzodiazepin-2-ones and dienyl thiazolidin-4-ones

被引：12

作者：

Kuila, Bilash ^{[1
]}

Kumar, Yogesh ^{[1
]}

Mahajan, Dinesh ^{[2
]}

Kumar, Kapil ^{[3
]}

Singh, Prabhpreet ^{[3
]}

Bhargava, Gaurav ^{[1
]}

机构：

[1] IK Gujral Punjab Tech Univ, Dept Appl Sci, Kapurthala 144603, Punjab, India

[2] Sphaera Pharma Pvt Ltd, IMT Manesar, Plot 32,Sec 5, Gurgaon 122051, Haryana, India

[3] Guru Nanak Dev Univ, Dept Chem, Amritsar 143005, Punjab, India

来源：

RSC ADVANCES | 2016年 / 6卷 / 62期

关键词：

LACTAM SYNTHON METHOD; BETA-LACTAMS; DIASTEREOSELECTIVE SYNTHESIS; BUILDING-BLOCKS; INHIBITORS; DERIVATIVES; POTENT; 1,4-BENZODIAZEPINE-2,5-DIONES; PEPTIDOMIMETICS; 2-AZETIDINONES;

D O I：

10.1039/c6ra10021j

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

An efficient protocol for chemoselective synthesis of previously unknown 1,4-benzodiazepin-2-ones and dienyl thiazolidin-4-one carboxylates in excellent yields by ring transformation reactions of functionally decorated 2-azetidin-3-thiazolidin-4-ones is reported.

引用

页码：S7485 / S7489

页数：5

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