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- [21] Variants in the GPR40 gene and association with type 2 diabetesDIABETOLOGIA, 2006, 49 : 37 - 37Kalis, M.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, SwedenLeveen, P.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, SwedenLyssenko, V.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, SwedenAlmgren, P.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, SwedenOlde, B.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, SwedenOwman, C.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, SwedenGroop, L.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, SwedenCilio, C. M.论文数: 0 引用数: 0 h-index: 0机构: Lund Univ, Dept Clin Sci, Cellular Autoimmun Unit, Malmo, Sweden
- [22] GPR40 agonists for the treatment of type 2 diabetes: life after 'TAKing' a hitDIABETES OBESITY & METABOLISM, 2015, 17 (07): : 622 - 629Mancini, A. D.论文数: 0 引用数: 0 h-index: 0机构: CRCHUM, Montreal Diabet Res Ctr, Montreal, PQ, Canada Univ Montreal, Dept Med, Montreal, PQ H3C 3J7, Canada CRCHUM, Montreal Diabet Res Ctr, Montreal, PQ, Canada论文数: 引用数: h-index:机构:
- [23] Discovery and development of CPL207280 as new GPR40/FFA1 agonistEUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2021, 226Mach, Mateusz论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandBazydlo-Guzenda, Katarzyna论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Med Univ Warsaw, Postgrad Sch Mol Med, 61 Zwirki & Wigury St, PL-02091 Warsaw, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandBuda, Pawel论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandMatloka, Mikolaj论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandDzida, Radoslaw论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandStelmach, Filip论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandGalazka, Kinga论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandWasinska-Kalwa, Malgorzata论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandSmuga, Damian论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandHolowinska, Dagmara论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandDawid, Urszula论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandGurba-Bryskiewicz, Lidia论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandWisniewski, Krzysztof论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandDubiel, Krzysztof论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandPieczykolan, Jerzy论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, PolandWieczorek, Maciej论文数: 0 引用数: 0 h-index: 0机构: Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland Celon Pharma SA, R&D Ctr, Marymoncka 15, PL-05152 Kazun Nowy, Poland
- [24] Discovery of TUG-770: A Highly Potent Free Fatty Acid Receptor 1 (FFA1/GPR40) Agonist for Treatment of Type 2 DiabetesACS MEDICINAL CHEMISTRY LETTERS, 2013, 4 (05): : 441 - 445Christiansen, Elisabeth论文数: 0 引用数: 0 h-index: 0机构: Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, Denmark Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, Denmark论文数: 引用数: h-index:机构:Urban, Christian论文数: 0 引用数: 0 h-index: 0机构: Univ Dusseldorf, Inst Pharmaceut & Med Chem, D-40225 Dusseldorf, Germany Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkHudson, Brian D.论文数: 0 引用数: 0 h-index: 0机构: Univ Glasgow, Coll Med Vet & Life Sci, Inst Mol Cell & Syst Biol, Glasgow G12 8QQ, Lanark, Scotland Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkWargent, Edward T.论文数: 0 引用数: 0 h-index: 0机构: Univ Buckingham, Clore Lab, Buckingham MK18 1EG, England Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkGrundmann, Manuel论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Inst Pharmaceut Biol, D-53115 Bonn, Germany Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkJenkins, Laura论文数: 0 引用数: 0 h-index: 0机构: Univ Glasgow, Coll Med Vet & Life Sci, Inst Mol Cell & Syst Biol, Glasgow G12 8QQ, Lanark, Scotland Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkZaibi, Mohamed论文数: 0 引用数: 0 h-index: 0机构: Univ Buckingham, Clore Lab, Buckingham MK18 1EG, England Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkStocker, Claire J.论文数: 0 引用数: 0 h-index: 0机构: Univ Buckingham, Clore Lab, Buckingham MK18 1EG, England Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkUllrich, Susanne论文数: 0 引用数: 0 h-index: 0机构: Univ Tubingen, Dept Internal Med 4, Div Endocrinol Diabetol Vasc Med Nephrol & Clin C, D-72076 Tubingen, Germany Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkKostenis, Evi论文数: 0 引用数: 0 h-index: 0机构: Univ Bonn, Inst Pharmaceut Biol, D-53115 Bonn, Germany Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkKassack, Matthias U.论文数: 0 引用数: 0 h-index: 0机构: Univ Dusseldorf, Inst Pharmaceut & Med Chem, D-40225 Dusseldorf, Germany Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkMilligan, Graeme论文数: 0 引用数: 0 h-index: 0机构: Univ Glasgow, Coll Med Vet & Life Sci, Inst Mol Cell & Syst Biol, Glasgow G12 8QQ, Lanark, Scotland Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkCawthorne, Michael A.论文数: 0 引用数: 0 h-index: 0机构: Univ Buckingham, Clore Lab, Buckingham MK18 1EG, England Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, DenmarkUlven, Trond论文数: 0 引用数: 0 h-index: 0机构: Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, Denmark Univ Southern Denmark, Dept Phys Chem & Pharm, DK-5230 Odense M, Denmark
- [25] AMG 837: A potent, orally bioavailable, partial allosteric agonist of GPR40ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2012, 243Houze, Jonathan B.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAZhu, Liusheng论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASun, Ying论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAAkerman, Michelle论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAQiu, Wei论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAZhang, Alex J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASharma, Rajiv论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASchmitt, Michael论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAWang, Yingcai论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USALiu, Jiwen论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAMedina, Julio C.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAReagan, Jeff D.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USALuo, Jian论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USATonn, George论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAZhang, Jane论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAGuo, Qi论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USASwaminath, Gayathri论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USALu, Jenny Y. -L.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAChen, Michael论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USALopez, Edwin论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USANguyen, Kathy论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAYang, Li论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USATang, Liang论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USATian, Hui论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USAShuttleworth, Steven J.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USALin, Daniel C. -H.论文数: 0 引用数: 0 h-index: 0机构: Amgen Inc, San Francisco, CA 94080 USA Amgen Inc, San Francisco, CA 94080 USA
- [26] Discovery of DS-1558: A Potent and Orally Bioavailable GPR40 AgonistACS MEDICINAL CHEMISTRY LETTERS, 2015, 6 (03): : 266 - 270Takano, Rieko论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanYoshida, Masao论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanInoue, Masahiro论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanHonda, Takeshi论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanNakashima, Ryutaro论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanMatsumoto, Koji论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanYano, Tatsuya论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanOgata, Tsuneaki论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanWatanabe, Nobuaki论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanHirouchi, Masakazu论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanYoneyama, Tomoko论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo RD Novare Co Ltd, Drug Discovery & Biomed Technol Unit, Edogawa Ku, Tokyo 1348630, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanIto, Shuichiro论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo RD Novare Co Ltd, Drug Discovery & Biomed Technol Unit, Edogawa Ku, Tokyo 1348630, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, JapanToda, Narihiro论文数: 0 引用数: 0 h-index: 0机构: Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan Daiichi Sankyo Co Ltd, R&D Div, Shinagawa Ku, Tokyo 1408710, Japan
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