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- [1] Phase II trial of the PI3 kinase inhibitor buparlisib (BKM-120) with or without enzalutamide in men with metastatic castration resistant prostate cancerEUROPEAN JOURNAL OF CANCER, 2017, 81 : 228 - 236Armstrong, Andrew J.论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Med, Durham, NC USA Duke Univ, Dept Surg, Durham, NC USA Duke Univ, Dept Pharmacol, Durham, NC USA Duke Univ, Dept Canc Biol, Div Med Oncol, Duke Canc Inst, Durham, NC USA Duke Univ, Dept Med, Durham, NC USAHalabi, Susan论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Biostat, Durham, NC USA Duke Univ, Dept Med, Durham, NC USAHealy, Patrick论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Biostat, Durham, NC USA Duke Univ, Dept Med, Durham, NC USAAlumkal, Joshi J.论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Knight Canc Inst, Portland, OR 97201 USA Duke Univ, Dept Med, Durham, NC USAWinters, Carolyn论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Med, Durham, NC USA Duke Univ, Dept Surg, Durham, NC USA Duke Univ, Dept Pharmacol, Durham, NC USA Duke Univ, Dept Canc Biol, Div Med Oncol, Duke Canc Inst, Durham, NC USA Duke Univ, Dept Med, Durham, NC USAKephart, Julie论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Med, Durham, NC USA Duke Univ, Dept Surg, Durham, NC USA Duke Univ, Dept Pharmacol, Durham, NC USA Duke Univ, Dept Canc Biol, Div Med Oncol, Duke Canc Inst, Durham, NC USA Duke Univ, Dept Med, Durham, NC USABitting, Rhonda L.论文数: 0 引用数: 0 h-index: 0机构: Wake Forest Univ, Winston Salem, NC 27109 USA Duke Univ, Dept Med, Durham, NC USAHobbs, Carey论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Med, Durham, NC USA Duke Univ, Dept Surg, Durham, NC USA Duke Univ, Dept Pharmacol, Durham, NC USA Duke Univ, Dept Canc Biol, Div Med Oncol, Duke Canc Inst, Durham, NC USA Duke Univ, Dept Med, Durham, NC USASoleau, Colleen F.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Seattle, WA 98195 USA Duke Univ, Dept Med, Durham, NC USA论文数: 引用数: h-index:机构:Slottke, Rachel论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth & Sci Univ, Knight Canc Inst, Portland, OR 97201 USA Duke Univ, Dept Med, Durham, NC USAMundy, Kelly论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Med, Durham, NC USA Duke Univ, Dept Surg, Durham, NC USA Duke Univ, Dept Pharmacol, Durham, NC USA Duke Univ, Dept Canc Biol, Div Med Oncol, Duke Canc Inst, Durham, NC USA Duke Univ, Dept Med, Durham, NC USAYu, Evan Y.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Seattle, WA 98195 USA Duke Univ, Dept Med, Durham, NC USAGeorge, Daniel J.论文数: 0 引用数: 0 h-index: 0机构: Duke Univ, Dept Med, Durham, NC USA Duke Univ, Dept Surg, Durham, NC USA Duke Univ, Dept Pharmacol, Durham, NC USA Duke Univ, Dept Canc Biol, Div Med Oncol, Duke Canc Inst, Durham, NC USA Duke Univ, Dept Med, Durham, NC USA
- [2] Discovery of BKM120, a pan class I PI3 kinase inhibitor in phase I/II clinical trialsABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2010, 240Burger, Matthew T.论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAPecchi, Sabina论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAWagman, Allan论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USANi, Zhi-Jie论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAKnapp, Mark论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAAtallah, Gordana论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAPfister, Keith论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USANg, Simon论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USASmith, Aaron论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAPick, Teresa论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAFrazier, Kelly论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAVerhagen, Joelle论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAZhang, Yanchen论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USABartulis, Sarah论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAHendricksen, Tom论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAIwanowicz, Edwin论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAHazenadar, Joshua论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAHuh, Kay论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAAshash, Ahmad论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAXin, Xiaohua论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAMenezes, Daniel论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAMerritt, Hanne论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAWiesmann, Marion论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USAVoliva, Charles论文数: 0 引用数: 0 h-index: 0机构: Novartis Inst Biomed Res, Emeryville, CA USA Novartis Inst Biomed Res, Emeryville, CA USA
- [3] A phase Ib trial of enzalutamide with venetoclax in metastatic castration-resistant prostate cancer (mCRPC).JOURNAL OF CLINICAL ONCOLOGY, 2020, 38 (15)Gopalakrishnan, Dharmesh论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USAKirk, Jason论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USADavis, John论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USAGeorge, Saby论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USALevine, Ellis Glenn论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USABeumer, Jan Hendrik论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USAAppleman, Leonard Joseph论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USATang, Dean论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USAChatta, Gurkamal S.论文数: 0 引用数: 0 h-index: 0机构: Roswell Park Comprehens Canc Ctr, Buffalo, NY USA
- [4] Phase 2 study of the pan-isoform PI3 kinase inhibitor BKM120 in metastatic urothelial carcinoma patients.JOURNAL OF CLINICAL ONCOLOGY, 2015, 33 (07)Iyer, Gopa论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USATully, Christopher Michael论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAGarcia-Grossman, Ilana Rebecca论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAScott, Sasinya N.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USABoyd, Mariel Elena论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAMccoy, Asia S.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USABerger, Michael F.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USAAl-Ahmadie, Hikmat论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USASolit, David B.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USARosenberg, Jonathan E.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USABajorin, Dean F.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, New York, NY 10021 USA
- [5] Phase II trial of the phosphatidyinositol-3 kinase (PI3K) inhibitor BKM120 in recurrent glioblastoma (GBM)JOURNAL OF CLINICAL ONCOLOGY, 2013, 31 (15)Wen, Patrick Y.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAYung, W. K. Alfred论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAMellinghoff, Ingo K.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USALamborn, Kathleen论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USARamkissoon, Shakti论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USACloughesy, Timothy Francis论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USARinne, Mikael论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAOmuro, Antonio Marcilio Padula论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USADeAngelis, Lisa Marie论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAGilbert, Mark R.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAChi, Andrew S.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USABatchelor, Tracy论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAColman, Howard论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAChang, Susan Marina论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAMassacesi, Cristian论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USADiTomaso, Emmanuelle论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAPrados, Michael论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USAReardon, David A.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USALigon, Keith L.论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA
- [6] Phase I/II trial of enzalutamide (Enz) plus mifepristone (Mif) for metastatic castration-resistant prostate cancer (mCRPC)JOURNAL OF CLINICAL ONCOLOGY, 2020, 38 (06)Serritella, Anthony论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USAShevrin, Daniel H.论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USAHeath, Elisabeth I.论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USAWade, James Lloyd论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USAMartinez, Elia论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USAKarrison, Theodore论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USAStadler, Walter Michael论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USASzmulewitz, Russell Zelig论文数: 0 引用数: 0 h-index: 0机构: Univ Chicago, Med Ctr, Chicago, IL 60637 USA
- [7] Optimal sequencing of enzalutamide and abiraterone in men with metastatic castration-resistant prostate cancer (mCRPC)JOURNAL OF CLINICAL ONCOLOGY, 2016, 34 (02)Maughan, Benjamin Louis论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Medcl Ctr, Baltimore, MD USASuzman, Daniel L.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Medcl Ctr, Baltimore, MD USANadal, Rosa Maria论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Medcl Ctr, Baltimore, MD USABassi, Sunakshi论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Medcl Ctr, Baltimore, MD USAAntonarakis, Emmanuel S.论文数: 0 引用数: 0 h-index: 0机构: Johns Hopkins Medcl Ctr, Baltimore, MD USA
- [8] Phase II study of sorafenib and docetaxel in men with metastatic castration resistant prostate cancer (mCRPC)JOURNAL OF CLINICAL ONCOLOGY, 2009, 27 (15)Cetnar, J. P.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USARosen, M. A.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAVaughn, D. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAHaas, N. B.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USATroxel, A. B.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USASong, H.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAAdluru, G.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAFlaherty, K. T.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAO'Dwyer, P. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USAAmaravadi, R. K.论文数: 0 引用数: 0 h-index: 0机构: Univ Penn, Philadelphia, PA 19104 USA Univ Penn, Philadelphia, PA 19104 USA
- [9] PHASE 3 TRIAL OF PEMBROLIZUMAB AND ENZALUTAMIDE VERSUS ENZALUTAMIDE IN PATIENTS WITH METASTATIC CASTRATION-RESISTANT PROSTATE CANCER (MCRPC) (KEYNOTE-641)JOURNAL FOR IMMUNOTHERAPY OF CANCER, 2020, 8 : A210 - A210Graff, Julie Nicole论文数: 0 引用数: 0 h-index: 0机构: Oregon Hlth, Knight Canc Inst, Portland, OR USA Oregon Hlth, Knight Canc Inst, Portland, OR USABurgents, Joseph论文数: 0 引用数: 0 h-index: 0机构: Merck & Co Inc, Kenilworth, NJ USA Oregon Hlth, Knight Canc Inst, Portland, OR USALiang, Li Wen论文数: 0 引用数: 0 h-index: 0机构: MSD China, Beijing, Peoples R China Oregon Hlth, Knight Canc Inst, Portland, OR USAStenzl, Arnulf论文数: 0 引用数: 0 h-index: 0机构: Eberhard Karls Univ Tuebingen, Tubingen, Germany Oregon Hlth, Knight Canc Inst, Portland, OR USA
- [10] Randomized phase II study of olaparib with or without cediranib in men with metastatic castration-resistant prostate cancer (mCRPC)JOURNAL OF CLINICAL ONCOLOGY, 2020, 38 (06)Kim, Joseph W.论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAMcKay, Rana R.论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USATaplin, Mary-Ellen论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USADavis, Nancy B.论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAMonk, Paul论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAAppleman, Leonard Joseph论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USALara, Primo论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAVaishampayan, Ulka N.论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAZhang, Jingsong论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAPaul, Asit K.论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USABubley, Glenn论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAVan Allen, Eliezer Mendel论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAHuang, Ying论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAZhang, Zhenwei论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USALoda, Massimo论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAShapiro, Geoffrey论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USALoRusso, Patricia论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAIvy, S. Percy论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USAPetrylak, Daniel Peter论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USA