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- [21] A phase I/II dose-escalation and expansion study of ZN-c5, an oral selective estrogen receptor degrader (SERD), as monotherapy and in combination with palbociclib in patients with advanced estrogen receptor (ER)+/HER2-breast cancerANNALS OF ONCOLOGY, 2021, 32 : S619 - S619Abramson, V.论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USALinden, H. M.论文数: 0 引用数: 0 h-index: 0机构: Univ Washington, Seattle Canc Care Alliance, Med Ctr, Seattle, WA USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USACrew, K.论文数: 0 引用数: 0 h-index: 0机构: New York Presbyterian Columbia Univ, Med & Epidemiol, Med Ctr, New York, NY USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USAMortimer, J.论文数: 0 引用数: 0 h-index: 0机构: City Hope Comprehens Canc Ctr, Med Oncol & Therapeut Res, Duarte, CA USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USAAlidzanovic, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Clin Ctr Tuzla, Med Oncol, Tuzla, Bosnia & Herceg Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USANangia, J.论文数: 0 引用数: 0 h-index: 0机构: Baylor Coll Med, Breast Oncol, Houston, TX 77030 USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USALayman, R.论文数: 0 引用数: 0 h-index: 0机构: Univ Texas MD Anderson Canc Ctr, Breast Med Oncol Unit 1354, Houston, TX 77030 USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USAVranjes, Z. J.论文数: 0 引用数: 0 h-index: 0机构: Univ Clin Ctr, Republ Srpska Canc Ctr, Banja Luka, Bosnia & Herceg Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USAAndric, Z.论文数: 0 引用数: 0 h-index: 0机构: CHC Bezanijska Kosa, Med Oncol, Belgrade, Serbia Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USAMilovic-Kovacevic, M.论文数: 0 引用数: 0 h-index: 0机构: Inst Oncol & Radiol Serbia, Med Oncol Dept, Belgrade, Serbia Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USATrifunovic, J.论文数: 0 引用数: 0 h-index: 0机构: Oncol Inst Vojvodina, Med Oncol, Sremska Kamenica, Serbia Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USAKarchmit, Y.论文数: 0 引用数: 0 h-index: 0机构: Vitebsk Reg Clin Oncol Dispensary, Med Oncol, Vitebsk, BELARUS Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USASuarez, J.论文数: 0 引用数: 0 h-index: 0机构: Zentalis Pharmaceut, Clin Dev Operat, New York, NY USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USASuster, M.论文数: 0 引用数: 0 h-index: 0机构: Zentalis Pharmaceut, Clin Dev Operat, New York, NY USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USAPtaszynski, M.论文数: 0 引用数: 0 h-index: 0机构: Zentalis Pharmaceut, Clin Dev Operat, New York, NY USA Vanderbilt Ingram Canc Ctr, Hematol Oncol, Nashville, TN USA论文数: 引用数: h-index:机构:
- [22] Dose-escalation study of G1T48, an oral selective estrogen receptor degrader (SERD), in postmenopausal women with ER+/HER2-locally advanced or metastatic breast cancer (ABC)ANNALS OF ONCOLOGY, 2019, 30 : 121 - +Dees, E. C.论文数: 0 引用数: 0 h-index: 0机构: UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USAAftimos, P. G.论文数: 0 引用数: 0 h-index: 0机构: Inst Jules Bordet, Clin Trials Conduct Unit, Brussels, Belgium UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USAvan Oordt, C. W. Menke-van der Houven论文数: 0 引用数: 0 h-index: 0机构: Vrije Univ Amsterdam Med Ctr, Med Oncol, Amsterdam, Netherlands UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USADe Vries, E. G. E.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Groningen UMCG, Medicth Oncol, Groningen, Netherlands UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USANeven, P.论文数: 0 引用数: 0 h-index: 0机构: Univ Leuven, Vesalius Res Ctr VIB, Univ Hosp Leuven, KU Leuven, Leuven, Belgium UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USAPegram, M. D.论文数: 0 引用数: 0 h-index: 0机构: Stanford Comprehens Canc Inst, Med, Stanford, CA USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USAIqbal, R.论文数: 0 引用数: 0 h-index: 0机构: Vrije Univ Amsterdam Med Ctr, Med Oncol, Amsterdam, Netherlands UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USABoers, J.论文数: 0 引用数: 0 h-index: 0机构: Univ Hosp Groningen UMCG, Medicth Oncol, Groningen, Netherlands UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USAXiao, J.论文数: 0 引用数: 0 h-index: 0机构: G1 Therapeut Inc, Biometr, Res Triangle Pk, NC USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USASipes, C.论文数: 0 引用数: 0 h-index: 0机构: G1 Therapeut Inc, Clin Operat, Res Triangle Pk, NC USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USALi, C.论文数: 0 引用数: 0 h-index: 0机构: G1 Therapeut Inc, Clin Pharmacol, Clin Dev, Res Triangle Pk, NC USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USASorrentino, J. A.论文数: 0 引用数: 0 h-index: 0机构: G1 Therapeut Inc, Biomarkers, Clin Dev, Res Triangle Pk, NC USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USAMalik, R.论文数: 0 引用数: 0 h-index: 0机构: G1 Therapeut Inc, Res & Dev, Res Triangle Pk, NC USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USABeelen, A. P.论文数: 0 引用数: 0 h-index: 0机构: G1 Therapeut Inc, Clin Dev, Res Triangle Pk, NC USA UNC Lineberger Comprehens Canc Ctr, Hematol & Oncol, Chapel Hill, NC USA
- [23] A first-in-human phase I study to evaluate the oral selective estrogen receptor degrader (SERD), GDC-0927, in postmenopausal women with estrogen receptor positive (ER+) HER2-negative metastatic breast cancer (BC)CANCER RESEARCH, 2018, 78 (04)Dickler, Maura N.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAVillanueva, Rafael论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFidalgo, Jose Alejandro Perez论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMayer, Ingrid A.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABoni, Valentina论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWiner, Eric P.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAHamilton, Erika P.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABellet, Meritxell论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAUrruticoechea, Ander论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGonzalez-Martin, Antonio论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USACortes, Javier论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMartin, Miguel论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGiltnane, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGates, Mary论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USACheeti, Sravanthi论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFredrickson, Jill论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWang, Xiaojing论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFriedman, Lori S.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USASpoerke, Jill M.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMetcalfe, Ciara论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALiu, Lichuan论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALi, Robert论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMorley, Roland论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMcCurry, Ursula论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAChan, Iris T.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMueller, Lars论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMilan, Sandra论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALauchle, Jennifer论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAHumke, Eric W.论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABardia, Aditya论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA
- [24] A first-in-human phase I study to evaluate the oral selective estrogen receptor degrader (SERD), GDC-9545, in postmenopausal women with estrogen receptor-positive (ER+) HER2-negative (HER2-) metastatic breast cancerCANCER RESEARCH, 2020, 80 (04)Jhaveri, Komal论文数: 0 引用数: 0 h-index: 0机构: Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWiner, Eric Paul论文数: 0 引用数: 0 h-index: 0机构: Dana Farber Canc Inst, Boston, MA 02115 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALim, Elgene论文数: 0 引用数: 0 h-index: 0机构: St Vincents Hosp, Sydney, NSW, Australia Garvan Inst Med Res, Sydney, NSW, Australia Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFidalgo, Jose AlejandroPerez论文数: 0 引用数: 0 h-index: 0机构: Univ Valencia, INCLIVA, CIBERONC, Hosp Clin, Valencia, Spain Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABellet, Meritxell论文数: 0 引用数: 0 h-index: 0机构: Hosp Univ Vall dHebron, Barcelona, Spain Vall dHebron Inst Oncol VHIO, Barcelona, Spain Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMayer, Ingrid Alina论文数: 0 引用数: 0 h-index: 0机构: Vanderbilt Univ, Med Ctr, Nashville, TN USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABoni, Valentina论文数: 0 引用数: 0 h-index: 0机构: START Madrid CIOCC HM Univ Sanchinarro, Madrid, Spain Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAPatel, Jaymin M.论文数: 0 引用数: 0 h-index: 0机构: Beth Israel Deaconess Med Ctr, Boston, MA 02215 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USABardia, Aditya论文数: 0 引用数: 0 h-index: 0机构: Massachusetts Gen Hosp, Canc Ctr, Boston, MA 02114 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGarcia, Jose Manuel论文数: 0 引用数: 0 h-index: 0机构: Hosp Quiron, Barcelona, Spain Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAKabos, Peter论文数: 0 引用数: 0 h-index: 0机构: Univ Colorado, Denver, CO 80202 USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGates, Mary论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAChen, Ya-Chi论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFredrickson, Jill论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAWang, Xiaojing论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAFriedman, Lori Sickels论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USASpoerke, Jill论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGendreau, Steven论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMetcalfe, Ciara论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALiu, Lichuan论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAChang, Ching-Wei论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMonemi, Sharareh论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAGonzalez, Monica论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMcCurry, Ursula论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAMilan, Sandra论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USAHumke, Eric William论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, San Francisco, CA USA Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USALoi, Sherene论文数: 0 引用数: 0 h-index: 0机构: Peter MacCallum Canc Ctr, Melbourne, Vic, Australia Mem Sloan Kettering Canc Ctr, 1275 York Ave, New York, NY 10021 USA
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