New synthesis of fused pyrimidine derivatives via ortho-(isocyanomethyl)nitroaromatic compounds

被引：5

作者：

Ostrowski, S ^{[1
]}

机构：

[1] Polish Acad Sci, Inst Organ Chem, PL-01224 Warsaw, Poland

来源：

JOURNAL OF CHEMICAL RESEARCH-S | 1998年 / 01期

关键词：

D O I：

10.1039/a703092d

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

An efficient synthesis of functionalized fused pyrimidine derivatives from the respective ortho-(isocyanomethyl)nitroarenes is described: hydrolysis of the isocyano group in the title isocyanides followed by catalytic reduction of the nitro group and subsequent cyclocondensation of the diamine formed with orthoesters leads to the final products.

引用

页码：14 / 15

页数：3

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