Penetration of 3'-amino 3'-deoxythymidine, a cytotoxic metabolite of zidovudine, into the cerebrospinal fluid of HIV-1 infected patients

被引:0
|
作者
Hoetelmans, RMW
Kraaijeveld, CL
Meenhorst, PL
Mulder, JW
Burger, DM
Koks, CHW
Beijnen, JH
机构
[1] SLOTERVAART HOSP,DEPT PHARM,NL-1066 EC AMSTERDAM,NETHERLANDS
[2] SLOTERVAART HOSP,DEPT NEUROL,NL-1066 EC AMSTERDAM,NETHERLANDS
[3] SLOTERVAART HOSP,DEPT INTERNAL MED,NL-1066 EC AMSTERDAM,NETHERLANDS
[4] UNIV NIJMEGEN HOSP,DEPT CLIN PHARM,NL-6500 HB NIJMEGEN,NETHERLANDS
关键词
D O I
暂无
中图分类号
R392 [医学免疫学]; Q939.91 [免疫学];
学科分类号
100102 ;
摘要
引用
收藏
页码:P23 / P23
页数:1
相关论文
共 50 条
  • [21] Biomarkers of neuronal injury and amyloid metabolism in the cerebrospinal fluid of patients infected with HIV-1 subtypes B and C
    de Almeida, Sergio Monteiro
    Ribeiro, Clea E.
    Rotta, Indianara
    Piovesan, Mauro
    Tang, Bin
    Vaida, Florin
    Raboni, Sonia Mara
    Letendre, Scott
    Potter, Michael
    Batistela Fernandes, Meire S.
    Ellis, Ronald J.
    JOURNAL OF NEUROVIROLOGY, 2018, 24 (01) : 28 - 40
  • [22] CEREBROSPINAL-FLUID ANTICARDIOLIPIN ANTIBODIES IN PATIENTS WITH HIV-1 INFECTION
    BREY, RL
    ARROYO, R
    BOSWELL, RN
    JOURNAL OF ACQUIRED IMMUNE DEFICIENCY SYNDROMES, 1991, 4 (04) : 435 - 441
  • [23] Cerebrospinal-fluid HIV-1 RNA and drug concentrations after treatment with lamivudine plus zidovudine or stavudine
    Foudraine, NA
    Hoetelmans, RMW
    Lange, JMA
    de Wolf, F
    van Benthem, BHB
    Mass, JJ
    Keet, IPM
    Portegies, P
    LANCET, 1998, 351 (9115): : 1547 - 1551
  • [24] Pharmacokinetics of hydroxyurea in plasma and cerebrospinal fluid of HIV-1-infected patients
    Gwilt, PR
    Manouilov, KK
    McNabb, J
    Swindells, SS
    JOURNAL OF CLINICAL PHARMACOLOGY, 2003, 43 (09): : 1003 - 1007
  • [25] SOLID-STATE AND SOLUTION CONFORMATION OF 3'-AMINO-3'-DEOXYTHYMIDINE, PRECURSOR TO A NONCOMPETITIVE INHIBITOR OF HIV-1 REVERSE-TRANSCRIPTASE
    KOVACS, T
    PARKANYI, L
    PELCZER, I
    CERVANTESLEE, F
    PANNELL, KH
    TORRENCE, PF
    JOURNAL OF MEDICINAL CHEMISTRY, 1991, 34 (08) : 2595 - 2600
  • [26] Therapeutic concentrations of indinavir in cerebrospinal fluid of HIV-1-infected patients
    Brinkman, K
    Kroon, F
    Hugen, PWH
    Burger, DM
    AIDS, 1998, 12 (05) : 537 - 537
  • [27] Efficacy and safety of zidovudine, lamivudine, and tenofovir combination in antiretroviral naive, HIV-1 infected patients
    Rey, D
    Krebs, M
    Partisani, M
    Hess-Kempf, G
    Cheneau, C
    Priester, M
    Bernard-Henry, C
    De Mautort, E
    Lang, JM
    INTERNATIONAL JOURNAL OF ANTIMICROBIAL AGENTS, 2004, 24 : S120 - S120
  • [28] AROMATIC AMINO-ACID PHOSPHORAMIDATE DIESTERS AND TRIESTERS OF 3'-AZIDO-3'-DEOXYTHYMIDINE (AZT) ARE NONTOXIC INHIBITORS OF HIV-1 REPLICATION
    WAGNER, CR
    MCINTEE, EJ
    SCHINAZI, RF
    ABRAHAM, TW
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 1995, 5 (16) : 1819 - 1824
  • [29] The effect of zidovudine on skeletal muscle mtDNA in HIV-1 infected patients with mild or no muscle dysfunction
    Casademont, J
    Barrientos, A
    Grau, JM
    Pedrol, E
    Estivill, X
    UrbanoMarquez, A
    Nunes, V
    BRAIN, 1996, 119 : 1357 - 1364
  • [30] Inhibition of the initiation of HIV-1 reverse transcription by 3′-azido-3′-deoxythymidine -: Comparison with elongation
    Rigourd, M
    Lanchy, JM
    Le Grice, SFJ
    Ehresmann, B
    Ehresmann, C
    Marquet, R
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2000, 275 (35) : 26944 - 26951