Discovery of potent, selective, and brain-penetrant apoptosis signal-regulating kinase 1 (ASK1) inhibitors

被引:0
|
作者
de Turiso, Felix Gonzalez Lopez [1 ]
Himmelbauer, Martin [1 ]
Jones, John [1 ]
Xin, Zhili [1 ]
Gilfillan, Rab [1 ]
机构
[1] Biogen, Med Chem, Cambridge, MA USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
237-MEDI
引用
收藏
页数:1
相关论文
共 50 条
  • [31] Apoptosis signal-regulating kinase 1 (ASK1) induces neuronal differentiation and survival of PC12 cells
    Takeda, K
    Hatai, T
    Hamazaki, TS
    Nishitoh, H
    Saitoh, M
    Ichijo, H
    JOURNAL OF BIOLOGICAL CHEMISTRY, 2000, 275 (13) : 9805 - 9813
  • [32] Apoptosis signal-regulating kinase 1 (Ask1) targeted small interfering RNA on ischemic neuronal cell death
    Kim, Hyun-Woo
    Cho, Kyoung-Joo
    Lee, Su Kyoung
    Kim, Gyung W.
    BRAIN RESEARCH, 2011, 1412 : 73 - 78
  • [33] INHIBITION OF APOPTOSIS SIGNAL-REGULATING KINASE 1 (ASK1) REDUCES MYOCARDIAL ISCHEMIA-REPERFUSION INJURY IN THE MOUSE
    Toldo, Stefano
    Breckenridge, David
    Mezzaroma, Eleonora
    Van Tassell, Benjamin
    Kannan, Harsha R.
    Shryock, John
    Voelkel, Norbert F.
    Abbate, Antonio
    JOURNAL OF THE AMERICAN COLLEGE OF CARDIOLOGY, 2012, 59 (13) : E548 - E548
  • [34] Regulation of Degradation of Apoptosis Signal-Regulating Kinase 1 (ASK1) by Its Novel Interaction Partner, Gα13
    Kutuzov, M. A.
    Andreeva, A. V.
    Voyno-Yasenctskaya, T. A.
    MOLECULAR BIOLOGY OF THE CELL, 2006, 17
  • [35] REDUCTION OF HEPATOCYTE INJURY BY SRT-015, A NOVEL INHIBITOR OF APOPTOSIS SIGNAL-REGULATING KINASE 1 (ASK1).
    Plonowski, Artur
    Elias, Kathleen
    Brown, Samuel D.
    Veidal, Sanne
    Rigbolt, Kristoffer
    Feigh, Michael
    Porter, Terence
    McDonnell, Neil
    HEPATOLOGY, 2020, 72 : 1031 - 1031
  • [36] TOXI 10-Apoptosis signal-regulating kinase 1 (ASK1) is a sensor-trigger for stress signaling
    Codreanu, Simona G.
    Myers, Jeremy S.
    Wong, Hansen L.
    Liebler, Daniel C.
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238
  • [37] Impact of mitochondrial reactive oxygen species (ROS) and apoptosis signal-regulating kinase 1 (ASK1) in insulin resistance
    Nishikawa, T
    Imoto, K
    Sonoda, K
    Kukidome, D
    Fujisawa, K
    Yano, M
    Senokuchi, T
    Motoshima, H
    Taguchi, T
    Matsumura, T
    Araki, E
    DIABETES, 2005, 54 : A320 - A321
  • [38] Role of Apoptosis Signal-regulating Kinase-1 (ASK1) in Influenza A Virus-induced Lung Injury
    Gordon, E. M.
    Dong, B.
    Hollifield, M.
    Valenca, S. Dos Santos
    Garvy, B.
    Waters, C. M.
    AMERICAN JOURNAL OF RESPIRATORY AND CRITICAL CARE MEDICINE, 2023, 207
  • [39] Apoptosis Signal-Regulating Kinase 1 (ASK1) Is a Novel Regulator of Heparin-Induced Thrombocytopenia and Thrombosis in Mice
    Patel, Pravin
    Zhou, Yuhang
    McKenzie, Steven Edward
    Naik, Ulhas P.
    BLOOD, 2017, 130
  • [40] Modified Cyclophilin a Inhibits ER-Stress-Induced Apoptosis through Apoptosis Signal-Regulating Kinase 1(ASK1) Signaling
    Kim, Hunsung
    Choe, Wonchae
    FREE RADICAL BIOLOGY AND MEDICINE, 2012, 53 : S45 - S45