A facile microwave-assisted synthesis of 8,9-cycloalkathieno[3,2-e] [1,2,4]triazolo[1,5-c]pyrimidin-5(6H)-ones

被引：3
|
作者：
Kaur, Rajwinder [1 ,2 ]
Kishore, D. Pran [1 ,2 ]
Narayana, B. Lakshmi [1 ,2 ]
Rao, K. Venkat [1 ,2 ]
Balakumar, C. [3 ]
Rajkumar, V. [4 ,5 ]
Rao, A. Raghuram [1 ,2 ]
机构：
[1] Panjab Univ, Univ Inst Pharmaceut Sci, Pharmaceut Chem Div, Chandigarh 160014, India
[2] Panjab Univ, Ctr Adv Study Pharmaceut Sci UGC CAS, Chandigarh 160014, India
[3] Panjab Univ, CPEBS, Chandigarh 160014, India
[4] Panjab Univ, Dept Chem, Chandigarh 160014, India
[5] Panjab Univ, Ctr Adv Study Chem UGC CAS, Chandigarh 160014, India
来源：
JOURNAL OF CHEMICAL SCIENCES | 2011年 / 123卷 / 01期
关键词：
Microwave-irradiation; pyrimidinones; 1,2,4-triazole; aryl hydrazides; condensation; ADENOSINE RECEPTOR ANTAGONISTS; A(2A); POTENT; TRIAZOLOTHIENOPYRIMIDINES; PHARMACOLOGY; NONXANTHINE; DERIVATIVES;
D O I：
10.1007/s12039-011-0067-6
中图分类号：
O6 [化学];
学科分类号：
0703 ;
摘要：
A new series of fused thieno[3,2-e][1,2,4]triazolo[1,5-c]pyrimidinones was synthesized by condensation of ethyl-3-cyano-4,5,6,7-tetrahydrobenzo[b]thiophene-2-yl carbamate with aryl acid hydrazides in quantitative yields using a facile, one-pot procedure under microwave-assisted conditions.
引用
收藏
页码：69 / 73
页数：5
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