An improved two-step regioselective synthesis of naphth[1,2,-b]- and naphth[2,1-b]oxepin-5-ones

被引:0
|
作者
Tandon, VK [1 ]
Chhor, RB [1 ]
Goswamy, GK [1 ]
机构
[1] Univ Lucknow, Dept Chem, Lucknow 226007, Uttar Pradesh, India
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中图分类号
O62 [有机化学];
学科分类号
070303 ; 081704 ;
摘要
An improved regioselective synthesis of naphth[1,2-b]oxepin-5-one 1 and naphth[2, 1-b]oxepin-5-one 2 has been described. The key step is one-step regioselective synthesis of 4-naphthoxybutanoic acids 3 and 4, formed from the corresponding naphthols, and their cyclisation to naphthoxepinones 1 and 2.
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页码:1027 / 1029
页数:3
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