Synthesis of furo[3,4-c]quinolin-3(1H)-one derivatives through TMG catalyzed intramolecular aza-MBH reaction based on the furanones

被引：11

作者：

Yin, Dawei ^{[1
]}

Wang, Wei ^{[1
]}

Peng, Yangqiu ^{[1
]}

Ge, Zemei ^{[1
]}

Cheng, Tieming ^{[1
]}

Wang, Xin ^{[1
]}

Li, Runtao ^{[1
]}

机构：

[1] Peking Univ, Sch Pharmaceut Sci, State Key Lab Nat & Biomimet Drugs, Beijing 100191, Peoples R China

来源：

RSC ADVANCES | 2015年 / 5卷 / 22期

基金：

中国国家自然科学基金;

关键词：

BAYLIS-HILLMAN REACTION; INHIBITORS; ALKALOIDS; QUINOLINE;

D O I：

10.1039/c4ra13796e

中图分类号：

O6 [化学];

学科分类号：

0703 ;

摘要：

The first TMG catalyzed intramolecular aza-MBH reaction based on furanone derivatives was developed and successfully applied in the synthesis of a novel fused heterocyclic scaffold, furo[3,4-c]quinolin-3-(1H)-ones in moderate to good yields.

引用

页码：17296 / 17299

页数：4

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