共 50 条
- [31] Design, synthesis and enzymatic evaluation of 6-bridged imidazolyluracil derivatives as inhibitors of human thymidine phosphorylaseJOURNAL OF PHARMACY AND PHARMACOLOGY, 2007, 59 (04) : 537 - 547McNally, Virginia A.Rajabi, MehdiGbaj, AbdulStratford, Ian J.Edwards, Philip N.Douglas, Kenneth T.Bryce, Richard A.Jaffar, MohammedFreeman, Sally
- [32] Synthesis of a series of transition state analog inhibitors of guanine deaminase (guanase)ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2009, 238Chakraborty, SaibalHosmane, Ramchandra
- [33] Rational design of bis-indolylmethane-oxadiazole hybrids as inhibitors of thymidine phosphorylaseBIOORGANIC & MEDICINAL CHEMISTRY, 2018, 26 (12) : 3654 - 3663Taha, MuhammadRashid, UmerImran, SyahrulAli, Muhammad
- [34] DESIGN OF HIV PROTEASE INHIBITORS BASED ON THE TRANSITION-STATE ANALOG CONCEPTJOURNAL OF PHARMACOBIO-DYNAMICS, 1992, 15 (07): : S91 - S91MIMOTO, TIMAI, JKISANUKI, STANAKA, SHATTORI, NTAKAHASHI, OKATOH, RYUMISAKI, TSAKIKAWA, HAKAJI, KKISO, Y
- [35] CHARACTERIZATION OF PYROGLUTAMYL AMINOPEPTIDASE AND DESIGN OF POTENTIAL TRANSITION-STATE ANALOG INHIBITORSABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1988, 196 : 86 - MEDISVOBODA, KSCURRIE, BL
- [36] Synthesis and evaluation of multisubstrate bicyclic pyrimidine nucleoside inhibitors of human thymidine phosphorylaseJOURNAL OF MEDICINAL CHEMISTRY, 2006, 49 (26) : 7807 - 7815Allan, Amy L.Gladstone, Patricia L.Price, Melissa L. P.Hopkins, Stephanie A.Juarez, Jose C.Donate, FernandoTernansky, Robert J.Shaw, David E.Ganem, BruceLi, YingboWang, WeiruEalick, Steven
- [37] TRANSITION-STATE AND MULTISUBSTRATE ANALOG INHIBITORSENZYME KINETICS AND MECHANISM, PT D, 1995, 249 : 284 - 312RADZICKA, AWOLFENDEN, R
- [38] Design and Synthesis of Potent "Sulfur-Free" Transition State Analogue Inhibitors of 5′-Methylthioadenosine Nucleosidase and 5′-Methylthioadenosine PhosphorylaseJOURNAL OF MEDICINAL CHEMISTRY, 2010, 53 (18) : 6730 - 6746Longshaw, Alistair I.Adanitsch, FlorianGutierrez, Jemy A.Evans, Gary B.Tyler, Peter C.Schramm, Vern I.
- [39] Synthesis of transition state analogue inhibitors for purine nucleoside phosphorylase and N-riboside hydrolasesTETRAHEDRON, 2000, 56 (19) : 3053 - 3062Evans, GBFurneaux, RHGainsford, GJSchramm, VLTyler, PC
- [40] Design of Novel Inhibitors of Human Thymidine Phosphorylase: Synthesis, Enzyme Inhibition, in Vitro Toxicity, and Impact on Human Glioblastoma CancerJOURNAL OF MEDICINAL CHEMISTRY, 2019, 62 (03) : 1231 - 1245de Moura Sperotto, Nathalia D.Roth, Candida DevesRodrigues-Junior, Valnes S.Neves, Christiano EvPaula, Favero ReisdorferDadda, Adilio da SilvaBergo, Pedrode Freitas, Talita FreitasMacchi, Fernanda SouzaMoura, SidneiDuarte de Souza, Ana PaulaCampos, Maria MarthaBizarro, Cristiano ValimSantos, Diogenes SantiagoBasso, Luiz AugustoMachado, Pablo