Design and synthesis of transition state analog inhibitors of thymidine phosphorylase.

被引:0
|
作者
Kalman, TI [1 ]
Lai, L [1 ]
机构
[1] SUNY Buffalo, Dept Med Chem, Buffalo, NY 14260 USA
关键词
D O I
暂无
中图分类号
O6 [化学];
学科分类号
0703 ;
摘要
50-MEDI
引用
收藏
页码:U545 / U545
页数:1
相关论文
共 50 条
  • [1] Transition state of thymidine phosphorylase.
    Birck, MR
    Schramm, VL
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2003, 226 : U173 - U173
  • [2] The synthesis of possible transition state analogue inhibitors of thymidine phosphorylase
    Evans, Gary B.
    Gainsford, Graeme J.
    Schramm, Vern L.
    Tyler, Peter C.
    TETRAHEDRON LETTERS, 2015, 56 (02) : 406 - 409
  • [3] Synthesis and evaluation of multisubstrate bicyclic pyrimidine nucleoside inhibitors of human thymidine phosphorylase.
    Allan, AL
    Gladstone, PL
    Price, MLP
    Hopkins, SA
    Juarez, JC
    Doñate, F
    Ternansky, RJ
    Ganem, B
    Li, YB
    Wang, WR
    Ealick, SE
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U200 - U200
  • [4] Synthesis and evaluation of multisubstrate bicyclic pyrimidine nucleoside inhibitors of human thymidine phosphorylase.
    Allan, AL
    Gladstone, PL
    Price, MLP
    Hopkins, SA
    Juarez, JC
    Doñate, F
    Ternansky, RJ
    Ganem, B
    Li, YB
    Wang, WR
    Ealick, SE
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2005, 229 : U206 - U206
  • [5] Kinetic isotope effects of thymidine phosphorylase.
    Rezaei, M
    Kearny, M
    Kline, PC
    BIOCHEMISTRY, 2000, 39 (06) : 1551 - 1551
  • [6] Kinetic isotope effects of thymidine phosphorylase.
    Rezaei, M
    Kearny, M
    Kline, PC
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2000, 219 : U130 - U131
  • [7] Purine nucleoside phosphorylase. Transition state structure, transition state inhibitors and one-third-the-sites reactivity
    Miles, RW
    Tyler, PC
    Furneaux, RH
    Bagdassarian, CK
    Schramm, VL
    ENZYMATIC MECHANISMS, 1999, 27 : 32 - 47
  • [8] Rational design and synthesis of thymidine phosphorylase inhibitors.
    McNally, VA
    Williams, KJ
    Bryce, R
    Stratford, IJ
    Jaffar, M
    Freeman, S
    CLINICAL CANCER RESEARCH, 2001, 7 (11) : 3748S - 3748S
  • [9] Transition state of thymidine phosphorylase
    Birck, MTR
    Schramm, VL
    BIOCHEMISTRY, 2003, 42 (28) : 8625 - 8625
  • [10] Design and synthesis of prodrugs of thymidine phosphorylase inhibitors for xanthine oxidase biotransformation
    Reigan, P
    Chinje, E
    Douglas, KT
    Freeman, S
    Gbaj, A
    Stratford, IJ
    EUROPEAN JOURNAL OF CANCER, 2002, 38 : S122 - S123