The PIM kinase inhibitor TP-3654 demonstrates efficacy in a murine model of myelofibrosis

被引:2
|
作者
Dutta, Avik [1 ]
Nath, Dipmoy [1 ]
Yang, Yue [1 ]
Mohi, Golam [1 ]
机构
[1] Univ Virginia, Charlottesville, VA USA
关键词
D O I
10.1158/1538-7445.AM2018-1874
中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
1874
引用
收藏
页数:2
相关论文
共 50 条
  • [31] Proteasome inhibitor bortezomib can inhibit bone marrow fibrosis development in a murine model of myelofibrosis.
    Wagner-Ballon, O
    Gastinne, T
    Tulliez, M
    Lacout, C
    Pisani, D
    Chagraoui, H
    Villeval, JL
    Vainchenker, W
    Giraudier, S
    BLOOD, 2005, 106 (11) : 726A - 726A
  • [32] AMN107: Efficacy of the selective Bcr-Abl tyrosine kinase inhibitor in a murine model of chronic myelogenous leukemia
    Jensen, Michael R.
    Bruggen, Josef
    Dilea, Clifford
    Mestan, Jurgen
    Manley, Paul W.
    CANCER RESEARCH, 2006, 66 (08)
  • [33] Preclinical efficacy of the novel PIM2 kinase inhibitor, JP_11646, in human acute leukemia models
    Pundt, Krista E.
    Baldino, Carmen M.
    Caserta, Justin
    Dumas, Stephane
    Flanders, Yvonne
    Wang, Eunice S.
    Fetterly, Gerald J.
    CANCER RESEARCH, 2014, 74 (19)
  • [34] Identification of PIM447, a potent and selective proviral insertion site of Moloney murine leukemia (PIM) 1,2 and 3 kinase inhibitor in clinical trials for cancer
    Burger, Matthew
    Nishiguchi, Gisele
    Han, Wooseok
    Lan, Jiong
    Simmons, Robert
    Atallah, Gordana
    Tamez, Victoriano
    Zhang, Yanchen
    Ding, Yu
    Mathur, Michelle
    Muller, Kristine
    Bellamacina, Cornelia
    Lindvall, Mika
    Zang, Richard
    Huh, Kay
    Dai, Yumin
    Ginn, Elaine
    Aycinena, Alex
    Langowski, John
    Lambert, Amy
    Fritsch, Christine
    Kauffmann, Audry
    Pfister, Estelle
    Garcia, Pablo
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2015, 250
  • [35] Development of a murine orthotopic model of leukemia:: Evaluation of TP53 gene therapy efficacy
    Bossi, G
    Scardigli, R
    Musiani, P
    Martinelli, R
    Gentileschi, MP
    Soddu, S
    Sacchi, A
    CANCER GENE THERAPY, 2000, 7 (01) : 135 - 143
  • [36] Development of a murine orthotopic model of leukemia: Evaluation of TP53 gene therapy efficacy
    Gianluca Bossi
    Raffaella Scardigli
    Piero Musiani
    Roberta Martinelli
    Maria Pia Gentileschi
    Silvia Soddu
    Ada Sacchi
    Cancer Gene Therapy, 2000, 7 : 135 - 143
  • [37] The IMPDH inhibitor VX-944 demonstrates in vivo efficacy in an aggressive leukemia model.
    Jain, J
    Ma, JG
    Furey, B
    Recher, C
    Demur, C
    Poondru, S
    Zhang, JB
    Li, SL
    Firestone, B
    Olson, K
    Murphy, M
    Taylor, J
    Henkel, G
    Ball, E
    Yao, YM
    Almquist, S
    Hoover, R
    BLOOD, 2004, 104 (11) : 693A - 694A
  • [38] Discovery of Selective Small Molecule Pan-Pim Kinase Inhibitors with Potent Oral Efficacy in Murine Xenograft Models.
    O'Brien, Sean
    Haddach, Mustapha
    Borsan, Cosmin
    Michaux, Jerome
    Kerdoncuff, Pauline
    Schwaebe, Mike
    Pierre, Fabrice
    Stefan, Eric
    Nedelle, Anne Sophie
    Siddiqui-Jain, Adam
    Streiner, Nicole
    Macalino, Diwata
    Drygin, Denis
    Ho, Caroline
    Bliesath, Josh
    Omori, May
    Stansfield, Ryan
    Phung, Jennifer
    Ryckman, David
    Rice, William
    Anderes, Kenna
    BLOOD, 2009, 114 (22) : 687 - 688
  • [39] TAS5315, A NOVEL BRUTON'S TYROSINE KINASE INHIBITOR, DEMONSTRATES POTENT EFFICACY AGAINST BONE DESTRUCTION IN AN ANIMAL MODEL FOR RHEUMATOID ARTHRITIS
    Noma, Naruto
    Hosoi, Fumihito
    Iguchi, Satoru
    Kaneko, Ryusuke
    Yoshiga, Yohei
    Arima, Yasunobu
    Akasaka, Daichi
    Tanaka, Kenji
    Saito, Akihiro
    Utsugi, Teruhiro
    Ikizawa, Koichi
    ANNALS OF THE RHEUMATIC DISEASES, 2019, 78 : 1092 - 1092
  • [40] TAS5315, A NOVEL BRUTON'S TYROSINE KINASE (BTK) INHIBITOR, DEMONSTRATES POTENT EFFICACY IN MOUSE COLLAGEN-INDUCED ARTHRITIS MODEL
    Hosoi, F.
    Iguchi, S.
    Yoshiga, Y.
    Kaneko, R.
    Nakachi, Y.
    Akasaka, D.
    Yonekura, K.
    Iwasawa, Y.
    Sasaki, E.
    Utsugi, T.
    ANNALS OF THE RHEUMATIC DISEASES, 2015, 74 : 97 - 97