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- [41] Complete response using the EZH2 inhibitor tazemetostat against multiple relapsed follicular lymphoma in the leukemic phaseINTERNATIONAL CANCER CONFERENCE JOURNAL, 2024, 13 (04): : 488 - 492论文数: 引用数: h-index:机构:Nabe, Yoshimi论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, JapanHoraguchi, Ryusuke论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, JapanMinemura, Tomoki论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan论文数: 引用数: h-index:机构:Noguchi, Akira论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Diagnost Pathol, Toyama, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan论文数: 引用数: h-index:机构:Kamihara, Yusuke论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, JapanWada, Akinori论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, JapanFujihira, Takuma论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, JapanSato, Tsutomu论文数: 0 引用数: 0 h-index: 0机构: Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan Toyama Univ Hosp, Dept Hematol, 2630 Sugitani, Toyama 9300152, Japan
- [42] Discovery of IHMT-337 as a potent irreversible EZH2 inhibitor targeting CDK4 transcription for malignanciesSignal Transduction and Targeted Therapy, 8Husheng Mei论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceHong Wu论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceJing Yang论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceBin Zhou论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceAoli Wang论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceChen Hu论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceShuang Qi论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceZongru Jiang论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceFengming Zou论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceBeilei Wang论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceFeiyang Liu论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceYongfei Chen论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceWenchao Wang论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceJing Liu论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical ScienceQingsong Liu论文数: 0 引用数: 0 h-index: 0机构: Chinese Academy of Sciences,Anhui Province Key Laboratory of Medical Physics and Technology, Institute of Health and Medical Technology, Hefei Institutes of Physical Science
- [43] Selective killing of SMARCA2-and SMARCA4-deficient tumors by inhibition of EZH2: In vitro and in vivo preclinical modelsCANCER RESEARCH, 2017, 77Chan-Penebre, Elayne论文数: 0 引用数: 0 h-index: 0Armstrong, Kelli论文数: 0 引用数: 0 h-index: 0Drew, Allison论文数: 0 引用数: 0 h-index: 0Grassian, Alexandra R.论文数: 0 引用数: 0 h-index: 0Feldman, Igor论文数: 0 引用数: 0 h-index: 0Roche, Maria论文数: 0 引用数: 0 h-index: 0Ho, Peter论文数: 0 引用数: 0 h-index: 0Brach, Dorothy论文数: 0 引用数: 0 h-index: 0Raimondi, Alejandra论文数: 0 引用数: 0 h-index: 0Copeland, Robert A.论文数: 0 引用数: 0 h-index: 0Chesworth, Richard论文数: 0 引用数: 0 h-index: 0Smith, Jesse J.论文数: 0 引用数: 0 h-index: 0Ribich, Scott A.论文数: 0 引用数: 0 h-index: 0
- [44] Inhibition of cytoplasmic EZH2 induces antitumor activity through stabilization of the DLC1 tumor suppressor proteinNature Communications, 12Brajendra K. Tripathi论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Meghan F. Anderman论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Disha Bhargava论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Luciarita Boccuzzi论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Xiaolan Qian论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Dunrui Wang论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Marian E. Durkin论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Alex G. Papageorge论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Fernando J. de Miguel论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Katerina Politi论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Kylie J. Walters论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)James H. Doroshow论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)Douglas R. Lowy论文数: 0 引用数: 0 h-index: 0机构: Laboratory of Cellular Oncology,Departments of Pathology and Internal Medicine (Section of Medical Oncology)
- [45] Inhibition of cytoplasmic EZH2 induces antitumor activity through stabilization of the DLC1 tumor suppressor proteinNATURE COMMUNICATIONS, 2021, 12 (01)Tripathi, Brajendra K.论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USAAnderman, Meghan F.论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USABhargava, Disha论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USABoccuzzi, Luciarita论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USAQian, Xiaolan论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USAWang, Dunrui论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USADurkin, Marian E.论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USAPapageorge, Alex G.论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USAde Miguel, Fernando J.论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USAPoliti, Katerina论文数: 0 引用数: 0 h-index: 0机构: Yale Sch Med, Yale Canc Ctr, New Haven, CT USA Yale Sch Med, Sect Med Oncol, Dept Pathol, New Haven, CT USA Yale Sch Med, Sect Med Oncol, Dept Internal Med, New Haven, CT USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USAWalters, Kylie J.论文数: 0 引用数: 0 h-index: 0机构: NCI, Struct Biophys Lab, Ctr Canc Res, Frederick, MD 21701 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USADoroshow, James H.论文数: 0 引用数: 0 h-index: 0机构: NCI, Dev Therapeut Branch, Ctr Canc Res, Frederick, MD 21701 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USALowy, Douglas R.论文数: 0 引用数: 0 h-index: 0机构: NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA NCI, Lab Cellular Oncol, Ctr Canc Res, Bethesda, MD 20892 USA
- [46] Initial testing (stage 1) of tazemetostat (EPZ-6438), a novel EZH2 inhibitor, by the Pediatric Preclinical Testing ProgramPEDIATRIC BLOOD & CANCER, 2017, 64 (03)Kurmasheva, Raushan T.论文数: 0 引用数: 0 h-index: 0机构: Nationwide Childrens Hosp, Columbus, OH USA Nationwide Childrens Hosp, Columbus, OH USASammons, Melissa论文数: 0 引用数: 0 h-index: 0机构: Nationwide Childrens Hosp, Columbus, OH USA Nationwide Childrens Hosp, Columbus, OH USAFavours, Edward论文数: 0 引用数: 0 h-index: 0机构: Nationwide Childrens Hosp, Columbus, OH USA UTHSCSA, Greehey Childrens Canc Res Inst, 8403 Floyd Curl Dr, San Antonio, TX 78229 USA Nationwide Childrens Hosp, Columbus, OH USAWu, Jianwrong论文数: 0 引用数: 0 h-index: 0机构: St Jude Childrens Res Hosp, Memphis, TN 38105 USA Nationwide Childrens Hosp, Columbus, OH USAKurmashev, Dias论文数: 0 引用数: 0 h-index: 0机构: Nationwide Childrens Hosp, Columbus, OH USA UTHSCSA, Greehey Childrens Canc Res Inst, 8403 Floyd Curl Dr, San Antonio, TX 78229 USA Nationwide Childrens Hosp, Columbus, OH USACosmopoulos, Katherine论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Nationwide Childrens Hosp, Columbus, OH USAKeilhack, Heike论文数: 0 引用数: 0 h-index: 0机构: Ribon Therapeut Inc, Lexington, MD USA Nationwide Childrens Hosp, Columbus, OH USAKlaus, Christine R.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Nationwide Childrens Hosp, Columbus, OH USAHoughton, Peter J.论文数: 0 引用数: 0 h-index: 0机构: Nationwide Childrens Hosp, Columbus, OH USA UTHSCSA, Greehey Childrens Canc Res Inst, 8403 Floyd Curl Dr, San Antonio, TX 78229 USA Nationwide Childrens Hosp, Columbus, OH USASmith, Malcolm A.论文数: 0 引用数: 0 h-index: 0机构: NCI, Canc Therapy Evaluat Program, Bethesda, MD 20892 USA Nationwide Childrens Hosp, Columbus, OH USA
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- [48] A selective inhibitor of EZH2 blocks H3K27 methylation and kills mutant lymphoma cellsNature Chemical Biology, 2012, 8 : 890 - 896Sarah K Knutson论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Tim J Wigle论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Natalie M Warholic论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Christopher J Sneeringer论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Christina J Allain论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Christine R Klaus论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Joelle D Sacks论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Alejandra Raimondi论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Christina R Majer论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Jeffrey Song论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Margaret Porter Scott论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Lei Jin论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Jesse J Smith论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Edward J Olhava论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Richard Chesworth论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Mikel P Moyer论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Victoria M Richon论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Robert A Copeland论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Heike Keilhack论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Roy M Pollock论文数: 0 引用数: 0 h-index: 0机构: Epizyme,Kevin W Kuntz论文数: 0 引用数: 0 h-index: 0机构: Epizyme,
- [49] A selective inhibitor of EZH2 blocks H3K27 methylation and kills mutant lymphoma cellsNATURE CHEMICAL BIOLOGY, 2012, 8 (11) : 890 - 896Knutson, Sarah K.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAWigle, Tim J.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAWarholic, Natalie M.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USASneeringer, Christopher J.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAAllain, Christina J.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAKlaus, Christine R.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USASacks, Joelle D.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USARaimondi, Alejandra论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAMajer, Christina R.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USASong, Jeffrey论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAScott, Margaret Porter论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAJin, Lei论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USASmith, Jesse J.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAOlhava, Edward J.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAChesworth, Richard论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAMoyer, Mikel P.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USARichon, Victoria M.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USACopeland, Robert A.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAKeilhack, Heike论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAPollock, Roy M.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USAKuntz, Kevin W.论文数: 0 引用数: 0 h-index: 0机构: Epizyme Inc, Cambridge, MA USA Epizyme Inc, Cambridge, MA USA
- [50] PRC2-mediated repression of SMARCA2 predicts EZH2 inhibitor activity in SWI/SNF mutant tumorsPROCEEDINGS OF THE NATIONAL ACADEMY OF SCIENCES OF THE UNITED STATES OF AMERICA, 2017, 114 (46) : 12249 - 12254Januario, Thomas论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USAYe, Xiaofen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USABainer, Russell论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Bioinformat, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USAAlicke, Bruno论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USASmith, Tunde论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USAHaley, Benjamin论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USAModrusan, Zora论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Mol Biol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USAGould, Stephen论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Translat Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USAYauch, Robert L.论文数: 0 引用数: 0 h-index: 0机构: Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA Genentech Inc, Dept Discovery Oncol, San Francisco, CA 94080 USA