Inhibition of the recruitment of inflammatory cells by the tachykinin NK3 receptor antagonist, SR 142801, in a murine model of asthma

被引：0
|
作者：
Nenan, S. [1 ]
Germain, N. [1 ]
Lagente, V. [1 ]
Emonds-Alt, X. [2 ]
Advenier, C. [3 ]
Boichot, E. [1 ]
机构：
[1] Univ Rennes 1, Fac Pharm, INSERM, U456, F-35014 Rennes, France
[2] Sanofi Synthelabo Rech, Montpellier, France
[3] Univ Paris 05, Lab Pharmacol, F-75270 Paris 06, France
来源：
FUNDAMENTAL & CLINICAL PHARMACOLOGY | 2001年 / 15卷
关键词：
D O I：
暂无
中图分类号：
R9 [药学];
学科分类号：
1007 ;
摘要：
引用
收藏
页码：118 / 118
页数：1
相关论文
共 44 条
  • [21] Effect of local administration of a non-peptide NK3 receptor antagonist, SR 142801, on Clostridium difficile-induced diarrhea in guinea pigs.
    Theodorou, V
    Marche, P
    Corthier, G
    Edmonds-Alt, X
    Fioramonti, J
    Bueno, L
    GASTROENTEROLOGY, 1998, 114 (04) : A423 - A423
  • [22] Permissive role of neurokinin NK3 receptors in NK1 receptor-mediated activation of the locus coeruleus revealed by SR 142801
    Bert, L
    Rodier, D
    Bougault, I
    Allouard, N
    Le-Fur, G
    Soubrié, P
    Steinberg, R
    SYNAPSE, 2002, 43 (01) : 62 - 69
  • [23] Depression of windup of spinal neurons in the neonatal rat spinal cord in vitro by an NK3 tachykinin receptor antagonist
    Barbieri, M
    Nistri, A
    JOURNAL OF NEUROPHYSIOLOGY, 2001, 85 (04) : 1502 - 1511
  • [24] Pharmacological characterization of SR 142801: A new non-peptide antagonist of the neurokinin NK-3 receptor
    NguyenLe, XK
    Nguyen, QT
    Gobeil, F
    Pheng, LH
    EmondsAlt, X
    Breliere, JC
    Regoli, D
    PHARMACOLOGY, 1996, 52 (05) : 283 - 291
  • [25] Inhibition of the inflammatory response to antigen challenge in the hamster cheek pouch by the tachykinin NK1 receptor antagonist SR140333
    Hall, JM
    Palframan, R
    Reynia, S
    Brain, SD
    BRITISH JOURNAL OF PHARMACOLOGY, 1996, 119 : P274 - P274
  • [26] ANTAGONISM BY SR-142801, A NONPEPTIDE NK3 RECEPTOR ANTAGONIST, OF SENKTIDE-EVOKED INCREASE IN FIRING RATE IN GUINEA-PIG LOCUS-COERULEUS SLICES
    MICHAUD, JC
    SOUBRIE, P
    LEFUR, G
    BRITISH JOURNAL OF PHARMACOLOGY, 1995, 115 : P107 - P107
  • [27] Modifications by the NK1, NK2 and NK3 tachykinin antagonists (SR140333, SR48968, SR142801, respectively) of the NMDA-evoked release of [3H]acetylcholine in striatal compartments of the rat
    Gauchy, C
    Blanchet, F
    Perez, S
    Glowinski, J
    Kemel, ML
    Soubrie, P
    JOURNAL OF NEUROCHEMISTRY, 1997, 69 : S70 - S70
  • [28] Mapping the binding pocket of a novel, high-affinity, slow dissociating tachykinin NK3 receptor antagonist: Biochemical and electrophysiological characterization
    Malherbe, Pad
    Knoflach, Frederic
    Marcuz, Anne
    Bohnert, Claudia
    Weber, Michael
    Knust, Henner
    Ratni, Hasane
    Spooren, Will
    Ballard, Theresa M.
    Bissantz, Caterina
    NEUROPHARMACOLOGY, 2014, 86 : 259 - 272
  • [29] Involvement of enhanced neurokinin NK3 receptor expression in the severe asthma guinea pig model
    Mukaiyama, O
    Morimoto, K
    Nosaka, E
    Takahashi, S
    Yamashita, M
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2004, 498 (1-3) : 287 - 294
  • [30] CHARACTERIZATION OF TACHYKININ MEDIATED CALCIUM MOBILIZATION IN CHO-K1 CELLS EXPRESSING HUMAN NK3 RECEPTOR
    LALWANI, ND
    BROTT, D
    WU, LH
    CHUNG, FZ
    FASEB JOURNAL, 1994, 8 (07): : A1301 - A1301
12345