Discovery and functional characterization of small molecule inhibitors of SWI/SNFATPase activity in BRG1/SMARCA4-Deficient non small cell lung cancers

被引:0
|
作者
Jagani, Z. [1 ]
Chenail, G. [1 ]
Xiang, K. [1 ]
Bushold, G. [1 ]
Bhang, C. [1 ]
Li, A. [1 ]
Vattay, A. [1 ]
Gilbert, T. [1 ]
Zhu, J. [2 ]
Terranova, R. [3 ]
Dubost, V. [3 ]
Huet, F. [4 ]
Farley, D. [5 ]
Cantwell, J. [6 ]
Ruddy, D. [1 ]
Rakiec, D. [1 ]
Shirley, M. [1 ]
Elliott, G. [1 ]
Nakajima, K. [7 ]
Papillon, J. [7 ]
机构
[1] Novartis Inst BioMed Res, Oncol, Cambridge, MA USA
[2] Novartis Inst BioMed Res, Sci Data Analyt, Cambridge, MA USA
[3] Novartis Inst BioMed Res, Preclin Safety, Basel, Switzerland
[4] Novartis Inst BioMed Res, PreClin Safety, Cambridge, MA USA
[5] Novartis Inst BioMed Res, Chem Biol & Therapeut, Cambridge, MA USA
[6] Novartis Inst BioMed Res, Prot Sci, Emeryville, CA USA
[7] Novartis Inst BioMed Res, Global Discovery Chem, Cambridge, MA USA
关键词
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中图分类号
R73 [肿瘤学];
学科分类号
100214 ;
摘要
19 (PB-199
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收藏
页码:E23 / E23
页数:1
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