Small-Molecule CFTR Activators for Dry Eye Therapy

被引:0
|
作者
Flores, Alyssa M. [1 ,2 ]
Phuan, Puay W. [1 ]
Verkman, Alan S. [1 ]
Levin, Marc H. [2 ]
机构
[1] Univ Calif San Francisco, Med & Physiol, San Francisco, CA 94143 USA
[2] Univ Calif San Francisco, Ophthalmol, San Francisco, CA 94143 USA
关键词
D O I
暂无
中图分类号
R77 [眼科学];
学科分类号
100212 ;
摘要
4807
引用
收藏
页数:2
相关论文
共 50 条
  • [31] Small-molecule CFTR inhibitors slow cyst growth in polycystic kidney disease
    Yang, Baoxue
    Sonawane, Nitin D.
    Zhao, Dan
    Somlo, Stefan
    Verkman, A. S.
    JOURNAL OF THE AMERICAN SOCIETY OF NEPHROLOGY, 2008, 19 (07): : 1300 - 1310
  • [32] Dissecting Dynamic Allosteric Pathways Using Chemically Related Small-Molecule Activators
    Lisi, George P.
    Manley, Gregory A.
    Hendrickson, Heidi
    Rivalta, Ivan
    Batista, Victor S.
    Loria, J. Patrick
    STRUCTURE, 2016, 24 (07) : 1155 - 1166
  • [33] Correcting CFTR folding defects by small-molecule correctors to cure cystic fibrosis
    Mijnders, Marjolein
    Kleizen, Bertrand
    Braakman, Ineke
    CURRENT OPINION IN PHARMACOLOGY, 2017, 34 : 83 - 90
  • [34] Small-molecule targeting of translation initiation for cancer therapy
    Aktas, Bertal H.
    Qiao, Yuan
    Ozdelen, Esra
    Schubert, Roland
    Sevinc, Sema
    Harbinski, Fred
    Grubissich, Luciano
    Singer, Samuel
    Halperin, Jose A.
    ONCOTARGET, 2013, 4 (10) : 1606 - 1617
  • [35] Small-molecule activators of AMP-activated protein kinase as modulators of energy metabolism
    Novikova D.S.
    Garabadzhiu A.V.
    Melino G.
    Barlev N.A.
    Tribulovich V.G.
    Russian Chemical Bulletin, 2015, 64 (7) : 1497 - 1517
  • [36] Development of small-molecule inhibitors of autophagy as anticancer therapy
    Yuan, Junying
    Vakifahmetoglu-Norberg, Helin
    Xia, Hongguang
    Liu, Junli
    Li, Ying
    Kim, Minsu
    Ma, Dawei
    CANCER RESEARCH, 2012, 72
  • [37] Discovery of novel small-molecule aldehyde dehydrogenase 2 activators based on drug repurposing
    Tian, Wei
    Sun, Xiangpei
    Gao, Xing
    Wang, Wentao
    Chen, Zhuo
    Chen, Xin
    Zheng, Canhui
    JOURNAL OF SAUDI CHEMICAL SOCIETY, 2023, 27 (06)
  • [38] Small-molecule activators of AMP-activated protein kinase as modulators of energy metabolism
    Novikova, D. S.
    Garabadzhiu, A. V.
    Melino, G.
    Barlev, N. A.
    Tribulovich, V. G.
    RUSSIAN CHEMICAL BULLETIN, 2015, 64 (07) : 1497 - 1517
  • [39] Discovery of small-molecule Bax activators for the treatment of triple-negative breast cancer
    Liu, Gang
    Li, Dengfeng
    Chen, Haiying
    Ding, Ye
    She, Qiang
    Zhou, Jia
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 2018, 256
  • [40] Discovery and optimization of small molecule Bax activators for cancer therapy
    Liu, Gang
    Kim, Hyejin
    Ding, Chunyong
    Yu, Zhuo
    Wang, Hong
    Chen, Haiying
    Shen, Qiang
    Zhou, Jia
    CANCER RESEARCH, 2019, 79 (13)