New fragment analogues of antistasin's (ATS) active site - Design, synthesis and structure-activity relationship

被引:0
|
作者
Danalev, D. L. [1 ]
Vezenkov, L. T. [1 ]
机构
[1] Univ Chem Technol & Met, Dept Organ Chem, Sofia, Bulgaria
关键词
D O I
暂无
中图分类号
Q5 [生物化学]; Q7 [分子生物学];
学科分类号
071010 ; 081704 ;
摘要
引用
收藏
页码:171 / 171
页数:1
相关论文
共 50 条
  • [31] Structure-activity relationship of antileishmanials neolignan analogues
    Aveniente, Mario
    Pinto, Eduardo F.
    Santos, Lourivaldo S.
    Rossi-Bergmann, Bartira
    Barata, Lauro E. S.
    BIOORGANIC & MEDICINAL CHEMISTRY, 2007, 15 (23) : 7337 - 7343
  • [32] Structure-activity relationship studies of curcumin analogues
    Fuchs, James R.
    Pandit, Bulbul
    Bhasin, Deepak
    Etter, Jonathan P.
    Regan, Nicholas
    Abdelhamid, Dalia
    Li, Chenglong
    Lin, Jiayuh
    Li, Pui-Kai
    BIOORGANIC & MEDICINAL CHEMISTRY LETTERS, 2009, 19 (07) : 2065 - 2069
  • [33] Synthesis and structure-activity relationship studies of novel tubulysin U analogues - effect on cytotoxicity of structural variations in the tubuvaline fragment
    Shankar, Sreejith P.
    Jagodzinska, Monika
    Malpezzi, Luciana
    Lazzari, Paolo
    Manca, Ilaria
    Greig, Iain R.
    Sani, Monica
    Zanda, Matteo
    ORGANIC & BIOMOLECULAR CHEMISTRY, 2013, 11 (14) : 2273 - 2287
  • [34] Structure-Activity Relationship of Imidazopyridinium Analogues as Antagonists of Neuropeptide S Receptor
    Patnaik, Samarjit
    Marugan, Juan J.
    Liu, Ke
    Zheng, Wei
    Southall, Noel
    Dehdashti, Seameen J.
    Thorsell, Annika
    Heilig, Markus
    Bell, Lauren
    Zook, Michelle
    Eskay, Bob
    Brimacombe, Kyle R.
    Austin, Christopher P.
    JOURNAL OF MEDICINAL CHEMISTRY, 2013, 56 (22) : 9045 - 9056
  • [35] Chromone-Fused Cytosine Analogues: Synthesis, Biological Activity, and Structure-Activity Relationship
    Haveliwala, Dhaval D.
    Kamdar, Nimesh R.
    Mistry, Prashant T.
    Patel, Saurabh K.
    NUCLEOSIDES NUCLEOTIDES & NUCLEIC ACIDS, 2014, 33 (02): : 80 - 91
  • [36] Synthesis and Structure-Activity Relationship of Xenocoumacin 1 and Analogues as Inhibitors of Ribosomal Protein Synthesis
    Zumbrunn, Cornelia
    Krusi, Daniela
    Stamm, Christina
    Caspers, Patrick
    Ritz, Daniel
    Rueedi, Georg
    CHEMMEDCHEM, 2021, 16 (05) : 891 - 897
  • [37] SYNTHESIS AND STRUCTURE-ACTIVITY RELATIONSHIP OF NEW BISPHOSPHONATE DERIVATIVE
    TAKEUCHI, M
    SAKAMOTO, S
    KAWAMUKI, K
    KUDO, M
    ABE, T
    FUJITA, S
    MURASE, K
    ISOMURA, Y
    ABSTRACTS OF PAPERS OF THE AMERICAN CHEMICAL SOCIETY, 1990, 199 : 53 - MEDI
  • [38] Synthesis of isocryptolepine analogues and their structure-activity relationship studies as antiplasmodial and antiproliferative agents
    Aroonkit, Pasuk
    Thongsornkleeb, Charnsak
    Tummatorn, Jumreang
    Krajangsri, Suppachai
    Mungthin, Mathirut
    Ruchirawat, Somsak
    EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY, 2015, 94 : 56 - 62
  • [39] Synthesis and structure-activity relationship of teixobactin analogues via convergent Ser ligation
    Jin, Kang
    Po, Kathy Hiu Laam
    Wang, Shengxi
    Reuven, Jonathan Avraham
    Wai, Chi Nga
    Lau, Ho Ting
    Chan, Ting Ho
    Chen, Sheng
    Li, Xuechen
    BIOORGANIC & MEDICINAL CHEMISTRY, 2017, 25 (18) : 4990 - 4995
  • [40] Superoxide dismutase mimetics: Synthesis and structure-activity relationship study of MnTBAP analogues
    Gauuan, PJF
    Trova, MP
    Gregor-Boros, L
    Bocckino, SB
    Crapo, JD
    Day, BJ
    BIOORGANIC & MEDICINAL CHEMISTRY, 2002, 10 (09) : 3013 - 3021