Acute effects of an inverse agonist selective for α5 GABAA receptors on rat behaviour in the forced swim test

被引:0
|
作者
Samardzic, J. [1 ]
Batinic, B. [2 ]
Biawat, P. [3 ]
Obradovic, D. I. [1 ]
Cook, J. M. [3 ]
Savic, M. M. [2 ]
机构
[1] Univ Belgrade, Dept Pharmacol Clin Pharmacol & Toxicol, Fac Med, Belgrade, Serbia
[2] Univ Belgrade, Dept Pharmacol, Fac Pharm, Belgrade, Serbia
[3] Univ Wisconsin, Dept Chem & Biochem, Milwaukee, WI 53201 USA
关键词
D O I
10.1016/S0924-977X(12)70269-9
中图分类号
R74 [神经病学与精神病学];
学科分类号
摘要
引用
收藏
页码:S187 / S188
页数:2
相关论文
共 50 条
  • [21] Selective antagonism of 5α-reduced neurosteroid effects at GABAA receptors
    Mennerick, S
    He, YJ
    Jiang, X
    Manion, BD
    Wang, MD
    Shute, A
    Benz, A
    Evers, AS
    Covey, DF
    Zorumski, CF
    MOLECULAR PHARMACOLOGY, 2004, 65 (05) : 1191 - 1197
  • [22] Estrogen effects on the forced swim test differ in two outbred rat strains
    Koss, Wendy A.
    Einat, Haim
    Schloesser, Robert J.
    Manji, Husseini K.
    Rubinow, David R.
    PHYSIOLOGY & BEHAVIOR, 2012, 106 (02) : 81 - 86
  • [23] The 5-HT3 receptor agonist attenuates the action of antidepressants in the forced swim test in rats
    Nakagawa, Y
    Ishima, T
    Takashima, T
    BRAIN RESEARCH, 1998, 786 (1-2) : 189 - 193
  • [24] The antidepressant activity of inositol in the forced swim test involves 5-HT2 receptors
    Einat, H
    Clenet, F
    Shaldubina, A
    Belmaker, RH
    Bourin, M
    BEHAVIOURAL BRAIN RESEARCH, 2001, 118 (01) : 77 - 83
  • [25] INVERSE AGONIST OF α5 GABAA RECEPTORS HAD PREVENTIVE BUT NOT THERAPEUTIC EFFECTS ON ISOFLURANE-INDUCED MEMORY IMPAIRMENTS IN AGED RATS
    Liu, Yue
    Du, Lei
    Yin, Yiqing
    Zhao, Zifang
    ANESTHESIA AND ANALGESIA, 2018, 126 (04): : 49 - 51
  • [26] Preclinical and clinical pharmacology of the GABAA receptor α5 subtype-selective inverse agonist α5IA
    Atack, John R.
    PHARMACOLOGY & THERAPEUTICS, 2010, 125 (01) : 11 - 26
  • [27] EVALUATION OF ANTIDEPRESSANT-LIKE EFFECTS OF MELATONIN IN FEMALE RAT IN FORCED SWIM TEST
    Zahra, el Mrabet fatima
    Ouichou, Ali
    Mesfioui, Abdehalim
    DRUG METABOLISM REVIEWS, 2010, 42 : 108 - 109
  • [28] Effects of postnatal cocaine exposure and environmental enrichment on rat behavior in a forced swim test
    Magalhaes, A
    Summavielle, T
    Tavares, MA
    de Sousa, L
    CURRENT STATUS OF DRUG DEPENDENCE / ABUSE STUDIES: CELLULAR AND MOLECULAR MECHANISMS OF DRUGS OF ABUSE AND NEUROTOXICITY, 2004, 1025 : 619 - 629
  • [29] Antidepressant-like effects of neurokinin receptor antagonists in the forced swim test in the rat
    Dableh, LJ
    Yashpal, K
    Rochford, J
    Henry, JL
    EUROPEAN JOURNAL OF PHARMACOLOGY, 2005, 507 (1-3) : 99 - 105
  • [30] Divergent Metabolic Effects of Acute Versus Chronic Repeated Forced Swim Stress in the Rat
    Rabasa, Cristina
    Askevik, Kaisa
    Schele, Erik
    Hu, Min
    Vogel, Heike
    Dickson, Suzanne L.
    OBESITY, 2019, 27 (03) : 427 - 433